AR083019A1 - Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para tratar enfermedades de la retina, articulo de fabricacion y composicion farmaceutica que lo comprenden - Google Patents

Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para tratar enfermedades de la retina, articulo de fabricacion y composicion farmaceutica que lo comprenden

Info

Publication number
AR083019A1
AR083019A1 ARP110103391A ARP110103391A AR083019A1 AR 083019 A1 AR083019 A1 AR 083019A1 AR P110103391 A ARP110103391 A AR P110103391A AR P110103391 A ARP110103391 A AR P110103391A AR 083019 A1 AR083019 A1 AR 083019A1
Authority
AR
Argentina
Prior art keywords
imidazol
methylphenyl
methanol
prepare
pharmaceutical composition
Prior art date
Application number
ARP110103391A
Other languages
English (en)
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44675870&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR083019(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of AR083019A1 publication Critical patent/AR083019A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/4174Arylalkylimidazoles, e.g. oxymetazolin, naphazoline, miconazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Uso de un compuesto derivado de [3-(1-(1H-imidazol-4-il)etil)-2-metilfenil]metanol de la fórmula, (1), (2) ó (3) sus enantiómeros individuales, sus diastereoisómeros individuales, sus hidratos, sus solvatos, sus formas cristalinas, sus isómeros individuales, sus tautómeros individuales o una sal farmacéuticamente aceptable de los mismos, en donde R1 es H o alquilo C1-3; R2 es H o alquilo C1-3; R3 es H, alquilo C1-10, heterociclo o arilo; y R es alquilo C1-10, heterociclo o arilo; para preparar un medicamento útil para tratar enfermedades de la retina. Articulo de fabricación y composición farmacéutica que comprenden dicho compuesto.
ARP110103391A 2010-09-16 2011-09-16 Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para tratar enfermedades de la retina, articulo de fabricacion y composicion farmaceutica que lo comprenden AR083019A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US38337010P 2010-09-16 2010-09-16

Publications (1)

Publication Number Publication Date
AR083019A1 true AR083019A1 (es) 2013-01-23

Family

ID=44675870

Family Applications (4)

Application Number Title Priority Date Filing Date
ARP110103391A AR083019A1 (es) 2010-09-16 2011-09-16 Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para tratar enfermedades de la retina, articulo de fabricacion y composicion farmaceutica que lo comprenden
ARP110103392A AR083020A1 (es) 2010-09-16 2011-09-16 Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para tratar enfermedades y afecciones de la piel, articulo de fabricacion y composicion farmaceutica que lo comprenden
ARP110103390A AR083018A1 (es) 2010-09-16 2011-09-16 Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para la reduccion de la presion intraocular, articulo de fabricacion y composicion farmaceutica que lo comprenden
ARP110103389A AR083017A1 (es) 2010-09-16 2011-09-16 Prodrogas de ester de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol

Family Applications After (3)

Application Number Title Priority Date Filing Date
ARP110103392A AR083020A1 (es) 2010-09-16 2011-09-16 Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para tratar enfermedades y afecciones de la piel, articulo de fabricacion y composicion farmaceutica que lo comprenden
ARP110103390A AR083018A1 (es) 2010-09-16 2011-09-16 Uso de un compuesto de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol para preparar un medicamento util para la reduccion de la presion intraocular, articulo de fabricacion y composicion farmaceutica que lo comprenden
ARP110103389A AR083017A1 (es) 2010-09-16 2011-09-16 Prodrogas de ester de [3-(1-(1h-imidazol-4-il)etil)-2-metilfenil]metanol

Country Status (29)

Country Link
US (9) US8492422B2 (es)
EP (13) EP2616068B1 (es)
JP (4) JP6073229B2 (es)
KR (7) KR102139905B1 (es)
CN (5) CN103200942A (es)
AR (4) AR083019A1 (es)
AU (4) AU2011301847B2 (es)
BR (4) BR112013006362A2 (es)
CA (8) CA3122745A1 (es)
CL (4) CL2013000735A1 (es)
CY (3) CY1121024T1 (es)
DK (9) DK2616068T3 (es)
ES (10) ES2684055T3 (es)
HK (5) HK1185539A1 (es)
HU (5) HUE047476T2 (es)
IL (4) IL225282A0 (es)
MX (4) MX2013003008A (es)
MY (4) MY173846A (es)
NZ (1) NZ608751A (es)
PL (7) PL3050564T3 (es)
PT (7) PT3053576T (es)
RU (4) RU2013116405A (es)
SG (4) SG188570A1 (es)
SI (5) SI3338777T1 (es)
TR (1) TR201909249T4 (es)
TW (4) TW201240661A (es)
UA (1) UA112973C2 (es)
WO (4) WO2012037484A1 (es)
ZA (4) ZA201302193B (es)

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BR112014001501A2 (pt) * 2011-07-22 2017-02-14 Allergan Inc moduladores alfa-2 adrenérgicos para tratamento de distúrbios visuais mediados por projeções visuais centrais do olho
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CN108310442B (zh) * 2017-01-17 2021-08-27 台北科技大学 眼科用组合物
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CN108872431B (zh) * 2018-07-09 2021-03-23 成都倍特药业股份有限公司 一种检测4-(1-(2,5-二甲基苯基)乙基)-1h-咪唑或/和其盐酸盐的方法
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EP3348264B1 (en) 2020-01-01
IL225282A0 (en) 2013-06-27
EP3078376B1 (en) 2019-03-27
PT3348264T (pt) 2020-04-02
ES2904479T3 (es) 2022-04-05
AU2011301901B2 (en) 2016-02-11
HUE038698T2 (hu) 2018-11-28
HUE039090T2 (hu) 2018-12-28
KR101952457B1 (ko) 2019-02-26
PT3053576T (pt) 2018-10-08
US20120142746A1 (en) 2012-06-07
HK1185541A1 (zh) 2014-02-21
ES2593612T3 (es) 2016-12-12
RU2013116405A (ru) 2014-10-27
SG188572A1 (en) 2013-04-30
ZA201302288B (en) 2013-11-27
AR083017A1 (es) 2013-01-23
BR112013006362A2 (pt) 2016-06-28
JP2013537236A (ja) 2013-09-30
RU2013116403A (ru) 2014-10-27
HK1185540A1 (zh) 2014-02-21
ES2781681T3 (es) 2020-09-04
CA2811559A1 (en) 2012-03-22
MY191369A (en) 2022-06-20
DK3078376T3 (da) 2019-06-24
CN103200941B (zh) 2015-12-16
EP3659600A1 (en) 2020-06-03
KR102354097B1 (ko) 2022-01-20
ZA201302193B (en) 2013-11-27
US8492557B2 (en) 2013-07-23
US20130296394A1 (en) 2013-11-07
DK3338777T3 (da) 2020-04-20
KR101840500B1 (ko) 2018-03-20
DK3636263T3 (da) 2022-01-10
IL225281A0 (en) 2013-06-27
EP3078376A1 (en) 2016-10-12
DK3050563T3 (en) 2018-08-13
NZ608751A (en) 2015-04-24
CY1121024T1 (el) 2019-12-11
PT3050564T (pt) 2019-12-11
AR083020A1 (es) 2013-01-23
PL3348264T3 (pl) 2020-08-24
BR112013006352A2 (pt) 2016-06-28
WO2012037484A1 (en) 2012-03-22
CL2013000735A1 (es) 2013-11-29
ZA201302194B (en) 2013-11-27
CL2013000734A1 (es) 2013-11-08
EP2616069A1 (en) 2013-07-24
RU2612351C2 (ru) 2017-03-07
PT3338777T (pt) 2020-05-06
MY161607A (en) 2017-04-28
SI3053576T1 (sl) 2018-11-30
CY1122809T1 (el) 2021-05-05
JP6045495B2 (ja) 2016-12-14
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IL225280A0 (en) 2013-06-27
PL3053576T3 (pl) 2018-11-30
ES2687420T3 (es) 2018-10-25
HK1257416A1 (zh) 2019-10-18
ES2788051T3 (es) 2020-10-20
DK3348264T3 (da) 2020-03-23
EP3050564B1 (en) 2019-09-04
AU2011301856A1 (en) 2013-05-02
DK2616068T3 (en) 2016-08-29
JP2013537237A (ja) 2013-09-30
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AU2011301932C1 (en) 2016-09-01
MX2013003009A (es) 2013-06-28
EP3338777A1 (en) 2018-06-27
KR20130105658A (ko) 2013-09-25
RU2013116763A (ru) 2014-10-27
CA3122745A1 (en) 2012-03-22
TW201240662A (en) 2012-10-16
CL2013000733A1 (es) 2013-08-23
PL2616068T3 (pl) 2016-11-30
CA2812191C (en) 2021-04-13
KR20200091507A (ko) 2020-07-30
PL3050564T3 (pl) 2020-06-01
KR102104760B1 (ko) 2020-04-27
EP2616067B1 (en) 2016-05-18
WO2012037490A1 (en) 2012-03-22
WO2012037499A1 (en) 2012-03-22
KR101840501B1 (ko) 2018-05-04
US20160354346A1 (en) 2016-12-08
US8492422B2 (en) 2013-07-23
US8853251B2 (en) 2014-10-07
US20150148394A1 (en) 2015-05-28
EP3636263A1 (en) 2020-04-15
AU2011301847A1 (en) 2013-05-02
PT2616068T (pt) 2016-09-13
AU2011301856C1 (en) 2016-09-08
EP3348264A1 (en) 2018-07-18
TR201909249T4 (tr) 2019-07-22
EP2616069B1 (en) 2016-11-16
BR112013006355A2 (pt) 2016-06-28
SI3050563T1 (sl) 2018-10-30
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CA2812197C (en) 2024-01-02
CN105412092B (zh) 2020-11-17
PT3050563T (pt) 2018-10-01
SG188570A1 (en) 2013-04-30
IL225278A0 (en) 2013-06-27
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MX2013003008A (es) 2013-06-28
HUE047476T2 (hu) 2020-04-28
CN103200942A (zh) 2013-07-10
US20120149746A1 (en) 2012-06-14
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US8653123B2 (en) 2014-02-18
TW201305116A (zh) 2013-02-01
US20120122945A1 (en) 2012-05-17
EP2616068B1 (en) 2016-07-13
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EP3698789A1 (en) 2020-08-26
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SG188573A1 (en) 2013-04-30
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AU2011301901A1 (en) 2013-05-02
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US20130289088A1 (en) 2013-10-31
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ZA201302291B (en) 2013-11-27
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US20120136036A1 (en) 2012-05-31
AU2011301847B2 (en) 2016-02-11
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