|
CA2726861C
(en)
|
2008-02-13 |
2014-05-27 |
Intarcia Therapeutics, Inc. |
Devices, formulations, and methods for delivery of multiple beneficial agents
|
|
AU2010272944B2
(en)
|
2009-07-13 |
2015-11-19 |
Zealand Pharma A/S |
Acylated glucagon analogues
|
|
RU2547990C2
(ru)
|
2009-09-28 |
2015-04-10 |
Интарсия Терапьютикс, Инк. |
Быстрое достижение и/или прекращение существенной стабильной доставки лекарственного средства
|
|
JP6006118B2
(ja)
|
2009-12-16 |
2016-10-12 |
ノヴォ ノルディスク アー/エス |
Glp−1アナログ及び誘導体
|
|
JP6039569B2
(ja)
*
|
2010-11-09 |
2016-12-07 |
ノヴォ ノルディスク アー/エス |
二重アシル化されたglp−1誘導体
|
|
SI2651398T1
(en)
|
2010-12-16 |
2018-04-30 |
Novo Nordisk A/S |
SOLID COMPOSITIONS CONTAINING GLP-1 AGONIST AND SOL N- (8- (2-HYDROXYBENZOIL) AMINO) CAPRICULATE ACIDS
|
|
US20120208755A1
(en)
*
|
2011-02-16 |
2012-08-16 |
Intarcia Therapeutics, Inc. |
Compositions, Devices and Methods of Use Thereof for the Treatment of Cancers
|
|
PL2696687T3
(pl)
|
2011-04-12 |
2017-06-30 |
Novo Nordisk A/S |
Pochodne podwójnie acylowanej GLP-1
|
|
BR112014001274A2
(pt)
|
2011-07-18 |
2017-04-18 |
Arts Biologics As |
composto de hormônio luteinizante, e, composição farmacêutica
|
|
JP6126097B2
(ja)
*
|
2011-09-06 |
2017-05-10 |
ノヴォ ノルディスク アー/エス |
Glp−1誘導体
|
|
CN110041399B
(zh)
|
2011-12-29 |
2023-12-12 |
诺沃—诺迪斯克有限公司 |
包含非成蛋白质性的氨基酸的二肽
|
|
US9452225B2
(en)
|
2012-03-01 |
2016-09-27 |
Novo Nordisk A/S |
GLP-1 prodrugs
|
|
PT2827845T
(pt)
|
2012-03-22 |
2019-03-29 |
Novo Nordisk As |
Composições compreendendo um agente de entrega e sua preparação
|
|
HRP20181447T1
(hr)
|
2012-03-22 |
2018-11-02 |
Novo Nordisk A/S |
Pripravci glp-1 peptida i njihova priprava
|
|
IN2014MN02304A
(https=)
|
2012-05-03 |
2015-08-07 |
Zealand Pharma As |
|
|
CN104411322B
(zh)
*
|
2012-05-08 |
2017-05-24 |
诺和诺德股份有限公司 |
双酰化glp‑1衍生物
|
|
EP2846823B1
(en)
|
2012-05-08 |
2019-12-04 |
Novo Nordisk A/S |
Double-acylated glp-1 derivatives
|
|
EP2851429B1
(en)
|
2012-05-18 |
2019-07-24 |
Adda Biotech Inc. |
Protein and protein conjugate for diabetes treatment, and applications thereof
|
|
JP6517690B2
(ja)
|
2012-06-20 |
2019-05-22 |
ノヴォ ノルディスク アー/エス |
ペプチド及び送達剤を含む錠剤製剤
|
|
EP2866825B1
(en)
|
2012-07-01 |
2020-04-08 |
Novo Nordisk A/S |
Use of long-acting glp-1 peptides
|
|
IN2015DN00544A
(https=)
|
2012-07-23 |
2015-06-26 |
Zealand Pharma As |
|
|
FR2994848B1
(fr)
|
2012-08-30 |
2014-08-22 |
Univ Paris Curie |
Traitement de l'arthrose par les hormones incretines ou leurs analogues
|
|
TWI608013B
(zh)
|
2012-09-17 |
2017-12-11 |
西蘭製藥公司 |
升糖素類似物
|
|
UA116217C2
(uk)
|
2012-10-09 |
2018-02-26 |
Санофі |
Пептидна сполука як подвійний агоніст рецепторів glp1-1 та глюкагону
|
|
EP2915817B1
(en)
*
|
2012-10-31 |
2018-06-20 |
Hybio Pharmaceutical Co., Ltd. |
Method for preparing exenatide
|
|
AU2013366692B2
(en)
|
2012-12-21 |
2017-11-23 |
Sanofi |
Dual GLP1/GIP or trigonal GLP1/GIP/Glucagon agonists
|
|
KR102272671B1
(ko)
*
|
2013-05-02 |
2021-07-06 |
노보 노르디스크 에이/에스 |
Glp-1 화합물의 경구 투여
|
|
JP6475233B2
(ja)
*
|
2013-06-20 |
2019-02-27 |
ノヴォ ノルディスク アー/エス |
Glp−1誘導体及びその使用
|
|
EP3016975B1
(en)
|
2013-07-04 |
2019-01-16 |
Novo Nordisk A/S |
Derivatives of glp-1 like peptides, and uses thereof
|
|
EP3033112B1
(en)
|
2013-08-15 |
2020-10-07 |
Novo Nordisk A/S |
Glp-1 derivatives, and uses thereof
|
|
JP6822839B2
(ja)
|
2013-09-13 |
2021-01-27 |
ザ・スクリップス・リサーチ・インスティテュート |
修飾された治療剤、及びその組成物
|
|
US9988429B2
(en)
|
2013-10-17 |
2018-06-05 |
Zealand Pharma A/S |
Glucagon analogues
|
|
PL3057984T3
(pl)
|
2013-10-17 |
2018-12-31 |
Zealand Pharma A/S |
Acylowane analogi glukagonu
|
|
WO2015067715A2
(en)
|
2013-11-06 |
2015-05-14 |
Zealand Pharma A/S |
Gip-glp-1 dual agonist compounds and methods
|
|
CN105829339B
(zh)
|
2013-11-06 |
2021-03-12 |
西兰制药公司 |
胰高血糖素-glp-1-gip三重激动剂化合物
|
|
US10626156B2
(en)
|
2013-12-06 |
2020-04-21 |
Jie Han |
Bioreversable promoieties for nitrogen-containing and hydroxyl-containing drugs
|
|
EP3080154B1
(en)
|
2013-12-13 |
2018-02-07 |
Sanofi |
Dual glp-1/gip receptor agonists
|
|
EP3080152A1
(en)
|
2013-12-13 |
2016-10-19 |
Sanofi |
Non-acylated exendin-4 peptide analogues
|
|
WO2015086728A1
(en)
|
2013-12-13 |
2015-06-18 |
Sanofi |
Exendin-4 peptide analogues as dual glp-1/gip receptor agonists
|
|
WO2015086733A1
(en)
|
2013-12-13 |
2015-06-18 |
Sanofi |
Dual glp-1/glucagon receptor agonists
|
|
KR102455171B1
(ko)
|
2013-12-18 |
2022-10-14 |
더 스크립스 리서치 인스티튜트 |
변형된 치료제, 스테이플드 펩티드 지질 접합체, 및 이의 조성물
|
|
TW201625669A
(zh)
|
2014-04-07 |
2016-07-16 |
賽諾菲公司 |
衍生自艾塞那肽-4(Exendin-4)之肽類雙重GLP-1/升糖素受體促效劑
|
|
TW201625668A
(zh)
|
2014-04-07 |
2016-07-16 |
賽諾菲公司 |
作為胜肽性雙重glp-1/昇糖素受體激動劑之艾塞那肽-4衍生物
|
|
TW201625670A
(zh)
|
2014-04-07 |
2016-07-16 |
賽諾菲公司 |
衍生自exendin-4之雙重glp-1/升糖素受體促效劑
|
|
ES2741507T3
(es)
*
|
2014-04-07 |
2020-02-11 |
Novo Nordisk As |
Compuestos de glp-1 acilados doblemente
|
|
EP3973994A1
(en)
|
2014-06-12 |
2022-03-30 |
RA Pharmaceuticals, Inc. |
Modulation of complement activity
|
|
US9932381B2
(en)
|
2014-06-18 |
2018-04-03 |
Sanofi |
Exendin-4 derivatives as selective glucagon receptor agonists
|
|
US9889085B1
(en)
|
2014-09-30 |
2018-02-13 |
Intarcia Therapeutics, Inc. |
Therapeutic methods for the treatment of diabetes and related conditions for patients with high baseline HbA1c
|
|
KR102620911B1
(ko)
|
2014-10-29 |
2024-01-05 |
질랜드 파마 에이/에스 |
Gip 효능제 화합물 및 방법
|
|
JP6730278B2
(ja)
*
|
2014-11-27 |
2020-07-29 |
ノヴォ ノルディスク アー/エス |
Glp−1誘導体及びその使用
|
|
WO2016097108A1
(en)
|
2014-12-17 |
2016-06-23 |
Novo Nordisk A/S |
Glp-1 derivatives and uses thereof
|
|
US9937222B2
(en)
|
2015-01-28 |
2018-04-10 |
Ra Pharmaceuticals, Inc. |
Modulators of complement activity
|
|
JP7211704B2
(ja)
*
|
2015-01-29 |
2023-01-24 |
ノヴォ ノルディスク アー/エス |
Glp-1アゴニスト及び腸溶コーティングを含む錠剤
|
|
US20180263915A1
(en)
*
|
2015-01-29 |
2018-09-20 |
Novo Nordisk A/S |
Pharmaceutical Composition for Oral GLP-1 Administration Comprising a Tablet Core and Immediate Release Coating
|
|
DK3283507T3
(da)
|
2015-04-16 |
2020-01-02 |
Zealand Pharma As |
Acyleret glucagonanalog
|
|
RU2730996C2
(ru)
|
2015-06-03 |
2020-08-26 |
Интарсия Терапьютикс, Инк. |
Системы установки и извлечения имплантата
|
|
AU2016270373A1
(en)
|
2015-06-05 |
2018-01-04 |
Vertex Pharmaceuticals Incorporated |
Triazoles for the treatment of demyelinating diseases
|
|
AR105319A1
(es)
|
2015-06-05 |
2017-09-27 |
Sanofi Sa |
Profármacos que comprenden un conjugado agonista dual de glp-1 / glucagón conector ácido hialurónico
|
|
EP3319968A1
(en)
|
2015-07-06 |
2018-05-16 |
Rodin Therapeutics, Inc. |
Heterobicyclic n-aminophenyl-amides as inhibitors of histone deacetylase
|
|
WO2017007756A1
(en)
|
2015-07-06 |
2017-01-12 |
Rodin Therapeutics, Inc |
Hetero-halo inhibitors of histone deacetylase
|
|
TW201706291A
(zh)
|
2015-07-10 |
2017-02-16 |
賽諾菲公司 |
作為選擇性肽雙重glp-1/升糖素受體促效劑之新毒蜥外泌肽(exendin-4)衍生物
|
|
CN106496322A
(zh)
*
|
2015-09-07 |
2017-03-15 |
江苏恒瑞医药股份有限公司 |
人胰岛素或其类似物的酰化衍生物的制备方法
|
|
EP3368556B1
(en)
*
|
2015-10-28 |
2024-04-10 |
Tufts University |
Novel polypeptides with improved proteolytic stability, and methods of preparing and using same
|
|
RU2733720C2
(ru)
|
2015-12-16 |
2020-10-06 |
Ра Фармасьютикалз, Инк. |
Модуляторы активности комплемента
|
|
GB2551945B
(en)
*
|
2015-12-18 |
2021-09-08 |
Heptares Therapeutics Ltd |
Novel GLP-1 receptor agonist peptides
|
|
US10946074B2
(en)
|
2016-03-03 |
2021-03-16 |
Novo Nordisk A/S |
GLP-1 derivatives and uses thereof
|
|
KR102574993B1
(ko)
|
2016-05-16 |
2023-09-06 |
인타르시아 세라퓨틱스 인코포레이티드 |
글루카곤-수용체 선택적 폴리펩티드 및 이들의 이용 방법
|
|
USD860451S1
(en)
|
2016-06-02 |
2019-09-17 |
Intarcia Therapeutics, Inc. |
Implant removal tool
|
|
USD840030S1
(en)
|
2016-06-02 |
2019-02-05 |
Intarcia Therapeutics, Inc. |
Implant placement guide
|
|
CN107561168A
(zh)
*
|
2016-06-30 |
2018-01-09 |
山东新时代药业有限公司 |
一种聚乙二醇化促胰岛素分泌肽类似物的分析检测方法
|
|
ES2828526T3
(es)
|
2016-11-07 |
2021-05-26 |
Novo Nordisk As |
Esteres activos DCHBS de compuestos PEG y sus usos
|
|
WO2018106646A1
(en)
|
2016-12-06 |
2018-06-14 |
Vertex Pharmaceuticals Incorporated |
Aminotriazoles for the treatment of demyelinating diseases
|
|
WO2018106641A1
(en)
|
2016-12-06 |
2018-06-14 |
Vertex Pharmaceuticals Incorporated |
Pyrazoles for the treatment of demyelinating diseases
|
|
WO2018106643A1
(en)
|
2016-12-06 |
2018-06-14 |
Vertex Pharmaceuticals Incorporated |
Heterocyclic azoles for the treatment of demyelinating diseases
|
|
KR20190093196A
(ko)
|
2016-12-07 |
2019-08-08 |
라 파마슈티컬스 인코포레이티드 |
보체 활성의 조절인자
|
|
JP7286542B2
(ja)
|
2017-01-03 |
2023-06-05 |
インターシア セラピューティクス,インコーポレイティド |
Glp-1受容体アゴニストの持続的投与及び薬物の同時投与を含む方法
|
|
HUE057849T2
(hu)
|
2017-01-11 |
2022-06-28 |
Alkermes Inc |
Hiszton deacetiláz biciklusos gátlói
|
|
FR3061715B1
(fr)
|
2017-01-12 |
2021-07-30 |
Institut National Univ Jean Francois Champollion |
Peptide immunomodulateur
|
|
MX2019010651A
(es)
*
|
2017-03-08 |
2020-01-13 |
Intarcia Therapeutics Inc |
Aparato y métodos para administración de un compuesto nauseogénico desde un dispositivo de administración de fármacos.
|
|
TWI797133B
(zh)
|
2017-06-09 |
2023-04-01 |
丹麥商諾佛 儂迪克股份有限公司 |
用於經口投予的固體組成物
|
|
LT3664802T
(lt)
|
2017-08-07 |
2022-06-27 |
Alkermes, Inc. |
Bicikliniai histonų deacetilazės inhibitoriai
|
|
KR102665710B1
(ko)
|
2017-08-24 |
2024-05-14 |
노보 노르디스크 에이/에스 |
Glp-1 조성물 및 그 용도
|
|
KR102396217B1
(ko)
*
|
2017-09-19 |
2022-05-09 |
임문워크 아이엔씨 |
알부민과의 결합 친화성이 증대된 약학 구조물
|
|
CA3078652A1
(en)
|
2017-10-12 |
2019-04-18 |
Novo Nordisk A/S |
Semaglutide in medical therapy
|
|
JP6898518B2
(ja)
|
2018-02-02 |
2021-07-07 |
ノヴォ ノルディスク アー/エス |
Glp−1アゴニスト、n−(8−(2−ヒドロキシベンゾイル)アミノ)カプリル酸の塩及び滑沢剤を含む固形組成物
|
|
MX2020010505A
(es)
|
2018-04-05 |
2021-01-15 |
Sun Pharmaceutical Ind Ltd |
Analogos novedosos de glp-1.
|
|
US11633459B2
(en)
|
2018-05-04 |
2023-04-25 |
Novo Nordisk A/S |
GIP derivatives and uses thereof
|
|
TWI829687B
(zh)
|
2018-05-07 |
2024-01-21 |
丹麥商諾佛 儂迪克股份有限公司 |
包含glp-1促效劑與n-(8-(2-羥基苯甲醯基)胺基)辛酸之鹽的固體組成物
|
|
CN109134257A
(zh)
*
|
2018-10-08 |
2019-01-04 |
扬州工业职业技术学院 |
一种两步法制备高纯度十二烷基二酸单叔丁酯的方法
|
|
CN109111361A
(zh)
*
|
2018-10-08 |
2019-01-01 |
扬州工业职业技术学院 |
一种一步法高效制备十二烷基二酸单叔丁酯的方法
|
|
WO2020118843A1
(zh)
*
|
2018-12-12 |
2020-06-18 |
四川利通科创生物医药科技有限公司 |
一种glp-1突变体及其制备方法和用途
|
|
MA54807A
(fr)
|
2019-01-24 |
2022-04-27 |
Novo Nordisk As |
Compacteur à rouleaux et procédé de granulation à sec utilisant un compacteur à rouleaux
|
|
WO2020180534A1
(en)
|
2019-03-01 |
2020-09-10 |
President And Fellows Of Harvard College |
Methods and compositions for protein delivery
|
|
KR20220004066A
(ko)
|
2019-04-03 |
2022-01-11 |
프레지던트 앤드 펠로우즈 오브 하바드 칼리지 |
약물 전달용 이온성 액체
|
|
JP2022535411A
(ja)
|
2019-06-04 |
2022-08-08 |
ラ ファーマシューティカルズ インコーポレイテッド |
補体阻害剤による炎症性疾患治療
|
|
WO2021070202A1
(en)
*
|
2019-10-09 |
2021-04-15 |
Prasad Alaparthi Lakshmi |
A method for preparing glp-1 analogue by solid-phase peptide synthesis
|
|
IL291876A
(en)
|
2019-11-06 |
2022-06-01 |
Novo Nordisk As |
Receptor agonists in glp-1 type dementia
|
|
WO2021089752A1
(en)
|
2019-11-07 |
2021-05-14 |
Novo Nordisk A/S |
Solid compositions comprising a glp-1 agonist, an sglt2 inhibitor and a salt of n-(8-(2-hydroxybenzoyl)amino)caprylic acid
|
|
CA3158963A1
(en)
|
2019-11-22 |
2021-05-27 |
Samir Mitragotri |
Ionic liquids for drug delivery
|
|
MX2022006861A
(es)
|
2019-12-04 |
2022-07-11 |
Scripps Research Inst |
Agonistas del receptor glp2 y metodos de uso.
|
|
EP4085077A4
(en)
|
2019-12-31 |
2024-01-17 |
Beijing QL Biopharmaceutical Co., Ltd. |
Fusion proteins of glp-1 and gdf15 and conjugates thereof
|
|
JP7761567B2
(ja)
|
2020-02-18 |
2025-10-28 |
ノヴォ ノルディスク アー/エス |
医薬製剤
|
|
GB202003762D0
(en)
*
|
2020-03-16 |
2020-04-29 |
Heptares Therapeutics Ltd |
GLP receptor agonists
|
|
CN115461044B
(zh)
|
2020-04-29 |
2025-06-10 |
诺和诺德股份有限公司 |
包含glp-1激动剂和组氨酸的固体组合物
|
|
CN114222755B
(zh)
*
|
2020-05-29 |
2024-06-11 |
北京拓界生物医药科技有限公司 |
Glp-1和gip受体双重激动剂化合物及其应用
|
|
EP4181946A1
(en)
*
|
2020-07-18 |
2023-05-24 |
Dr. Reddy's Laboratories Ltd. |
Improved purification process of semaglutide
|
|
EP4185607A1
(en)
|
2020-07-22 |
2023-05-31 |
Novo Nordisk A/S |
Co-agonists at glp-1 and gip receptors suitable for oral delivery
|
|
CN114729060B
(zh)
*
|
2020-09-30 |
2022-11-25 |
北京质肽生物医药科技有限公司 |
多肽缀合物和使用方法
|
|
WO2022096636A1
(en)
|
2020-11-06 |
2022-05-12 |
Novo Nordisk A/S |
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|
|
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|
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|
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|
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|
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