JP2011500562A5 - - Google Patents
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- Publication number
- JP2011500562A5 JP2011500562A5 JP2010528867A JP2010528867A JP2011500562A5 JP 2011500562 A5 JP2011500562 A5 JP 2011500562A5 JP 2010528867 A JP2010528867 A JP 2010528867A JP 2010528867 A JP2010528867 A JP 2010528867A JP 2011500562 A5 JP2011500562 A5 JP 2011500562A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- alkenyl
- compound according
- compound
- ring members
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 C*1C=C(*)C(C)(C)CC1 Chemical compound C*1C=C(*)C(C)(C)CC1 0.000 description 3
- ZRVYMRHQWZKLKY-UHFFFAOYSA-N CC1(COC)CCCC1 Chemical compound CC1(COC)CCCC1 ZRVYMRHQWZKLKY-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US99878607P | 2007-10-10 | 2007-10-10 | |
| US60/998,786 | 2007-10-10 | ||
| US6872408P | 2008-03-06 | 2008-03-06 | |
| US61/068,724 | 2008-03-06 | ||
| PCT/US2008/011422 WO2009048527A1 (en) | 2007-10-10 | 2008-10-03 | Substituted biphenyl gpr40 modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011500562A JP2011500562A (ja) | 2011-01-06 |
| JP2011500562A5 true JP2011500562A5 (enExample) | 2011-11-17 |
| JP5591706B2 JP5591706B2 (ja) | 2014-09-17 |
Family
ID=40338063
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010528867A Expired - Fee Related JP5591706B2 (ja) | 2007-10-10 | 2008-10-03 | 置換ビフェニルｇｐｒ４０調節因子 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US8030354B2 (enExample) |
| EP (1) | EP2205548A1 (enExample) |
| JP (1) | JP5591706B2 (enExample) |
| KR (1) | KR20100090249A (enExample) |
| CN (1) | CN102083783A (enExample) |
| AR (1) | AR068840A1 (enExample) |
| AU (1) | AU2008311355B2 (enExample) |
| BR (1) | BRPI0818253A2 (enExample) |
| CA (1) | CA2702047C (enExample) |
| CL (1) | CL2008002997A1 (enExample) |
| CO (1) | CO6270312A2 (enExample) |
| CR (1) | CR11420A (enExample) |
| IL (1) | IL204635A0 (enExample) |
| MA (1) | MA31841B1 (enExample) |
| MX (1) | MX2010003876A (enExample) |
| PE (1) | PE20091222A1 (enExample) |
| TN (1) | TN2010000125A1 (enExample) |
| TW (1) | TW200927091A (enExample) |
| WO (1) | WO2009048527A1 (enExample) |
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| US8476287B2 (en) | 2009-12-25 | 2013-07-02 | Mochida Pharmaceutical Co., Ltd. | 3-hydroxy-5-arylisothiazole derivative |
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| WO2013045413A1 (en) | 2011-09-27 | 2013-04-04 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
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| RU2015106909A (ru) | 2012-08-02 | 2016-09-27 | Мерк Шарп И Доум Корп. | Антидиабетические трициклические соединения |
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| KR101942752B1 (ko) * | 2012-11-05 | 2019-01-28 | 주식회사 엘지화학 | Ｇｐｒ120 효능제로서의 티오아릴 유도체 |
| PT2920165T (pt) | 2012-11-16 | 2016-12-20 | Bristol Myers Squibb Co | Moduladores de diidropirazol gpr40 |
| BR112015019836A2 (pt) | 2013-02-22 | 2017-07-18 | Merck Sharp & Dohme | composto, composição farmacêutica, e, uso de um composto |
| CA2905428A1 (en) * | 2013-03-14 | 2014-10-02 | Bristol-Myers Squibb Company | Bicyclo [2.2.1] acid gpr120 modulators |
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| JP6397410B2 (ja) * | 2013-08-09 | 2018-09-26 | 武田薬品工業株式会社 | 芳香環化合物 |
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| WO2015089809A1 (en) | 2013-12-19 | 2015-06-25 | Merck Sharp & Dohme Corp. | Antidiabetic substituted heteroaryl compounds |
| EP3102198B1 (en) | 2014-02-06 | 2020-08-26 | Merck Sharp & Dohme Corp. | Antidiabetic compounds |
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| EP3177282B1 (en) | 2014-08-08 | 2021-10-06 | Merck Sharp & Dohme Corp. | Antidiabetic bicyclic compounds |
| US10100042B2 (en) | 2014-08-08 | 2018-10-16 | Merck Sharp & Dohme Corp. | [5,6]—fused bicyclic antidiabetic compounds |
| WO2016019587A1 (en) | 2014-08-08 | 2016-02-11 | Merck Sharp & Dohme Corp. | [7, 6]-fused bicyclic antidiabetic compounds |
| US10968193B2 (en) | 2014-08-08 | 2021-04-06 | Merck Sharp & Dohme Corp. | Antidiabetic bicyclic compounds |
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| WO2017172505A1 (en) | 2016-03-29 | 2017-10-05 | Merck Sharp & Dohme Corp. | Antidiabetic bicyclic compounds |
| US11072602B2 (en) | 2016-12-06 | 2021-07-27 | Merck Sharp & Dohme Corp. | Antidiabetic heterocyclic compounds |
| WO2018118670A1 (en) | 2016-12-20 | 2018-06-28 | Merck Sharp & Dohme Corp. | Antidiabetic spirochroman compounds |
| JPWO2018181847A1 (ja) | 2017-03-31 | 2020-03-05 | 武田薬品工業株式会社 | 芳香環化合物 |
| AR111199A1 (es) | 2017-03-31 | 2019-06-12 | Takeda Pharmaceuticals Co | Compuesto aromático agonista de gpr40 |
| US11225471B2 (en) | 2017-11-16 | 2022-01-18 | Merck Sharp & Dohme Corp. | Antidiabetic bicyclic compounds |
| WO2019160882A1 (en) | 2018-02-13 | 2019-08-22 | Gilead Sciences, Inc. | Pd-1/pd-l1 inhibitors |
| WO2019204609A1 (en) | 2018-04-19 | 2019-10-24 | Gilead Sciences, Inc. | Pd-1/pd-l1 inhibitors |
| BR112020026746A2 (pt) | 2018-07-13 | 2021-03-30 | Gilead Sciences, Inc. | Composto, composição farmacêutica, métodos para inibir pd-1, pd-l1 e/ou a interação de pd-1/pd-l1 e para tratar câncer, e, kit para tratar ou prevenir câncer ou uma doença ou condição. |
| CN112955435B (zh) | 2018-10-24 | 2024-09-06 | 吉利德科学公司 | Pd-1/pd-l1抑制剂 |
| US20220152164A1 (en) * | 2019-03-22 | 2022-05-19 | Kallyope, Inc. | Gpcr combination therapies |
| PH12022552277A1 (en) | 2020-02-28 | 2024-03-04 | Kallyope Inc | Gpr40 agonists |
| US20240002354A1 (en) * | 2020-08-05 | 2024-01-04 | Rezubio Pharmaceuticals Co., Ltd | Antidiabetic compounds and compositions |
| EP4463451A4 (en) * | 2022-01-14 | 2026-01-14 | Rezubio Pharmaceuticals Co Ltd | ANTIDIABETIC COMPOUNDS AND COMPOSITIONS |
| WO2024075696A1 (ja) | 2022-10-03 | 2024-04-11 | 公立大学法人横浜市立大学 | 二環性構造を有するイミダゾピリジン誘導体 |
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| US7572934B2 (en) | 2007-04-16 | 2009-08-11 | Amgen Inc. | Substituted biphenyl GPR40 modulators |
-
2008
- 2008-10-03 BR BRPI0818253-1A patent/BRPI0818253A2/pt not_active Application Discontinuation
- 2008-10-03 MX MX2010003876A patent/MX2010003876A/es active IP Right Grant
- 2008-10-03 JP JP2010528867A patent/JP5591706B2/ja not_active Expired - Fee Related
- 2008-10-03 CN CN2008801199462A patent/CN102083783A/zh active Pending
- 2008-10-03 AU AU2008311355A patent/AU2008311355B2/en not_active Ceased
- 2008-10-03 EP EP08837085A patent/EP2205548A1/en not_active Withdrawn
- 2008-10-03 CA CA2702047A patent/CA2702047C/en not_active Expired - Fee Related
- 2008-10-03 US US12/287,036 patent/US8030354B2/en active Active
- 2008-10-03 WO PCT/US2008/011422 patent/WO2009048527A1/en not_active Ceased
- 2008-10-03 KR KR1020107010209A patent/KR20100090249A/ko not_active Withdrawn
- 2008-10-09 PE PE2008001746A patent/PE20091222A1/es not_active Application Discontinuation
- 2008-10-09 TW TW097139006A patent/TW200927091A/zh unknown
- 2008-10-09 CL CL2008002997A patent/CL2008002997A1/es unknown
- 2008-10-09 AR ARP080104409A patent/AR068840A1/es not_active Application Discontinuation
-
2010
- 2010-03-21 IL IL204635A patent/IL204635A0/en unknown
- 2010-03-22 TN TNP2010000125A patent/TN2010000125A1/fr unknown
- 2010-05-06 CO CO10054070A patent/CO6270312A2/es not_active Application Discontinuation
- 2010-05-10 MA MA32826A patent/MA31841B1/fr unknown
- 2010-05-10 CR CR11420A patent/CR11420A/es not_active Application Discontinuation
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