JP5591706B2 - 置換ビフェニルｇｐｒ４０調節因子 - Google Patents

置換ビフェニルｇｐｒ４０調節因子 Download PDF

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JP5591706B2
JP5591706B2 JP2010528867A JP2010528867A JP5591706B2 JP 5591706 B2 JP5591706 B2 JP 5591706B2 JP 2010528867 A JP2010528867 A JP 2010528867A JP 2010528867 A JP2010528867 A JP 2010528867A JP 5591706 B2 JP5591706 B2 JP 5591706B2
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alkyl
compound
formula
methyl
mmol
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JP2011500562A (ja
JP2011500562A5 (enExample
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ブラウン，シヨーン・ピー
ツアオ，チオン
ドランスフイールド，ポール・ジエイ
ドウ，シヤオフイ
ハウズ，ジヨナサン
ジアオ，シエン・ユイン
キム，ヨン−ジエ
コーン，トツド・ジエイ
ライ，スウジエン
リー，アン−ロン
リン，ダニエル
ルオ，ジエン
メデイナ，ジユリオ・シー
レーガン，ジエフリー・デイー
パツタロポン，バテイー
シユワルツ，マルグリツト
シエン，ワン
スウ，ヨンリー
スワミナス，ガヤスリ
ビモルラターナ，マルク
ワン，シアン
シオン，ユイメイ
ヤン，リー
ユイ，ミン
ジヤン，ジエ
ジユウ，リウシユヨン
フウ，ズーツオ
リウ，ジウエン
ワン，インツアイ
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アムジエン・インコーポレーテツド
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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
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  • Furan Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
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JP2010528867A 2007-10-10 2008-10-03 置換ビフェニルｇｐｒ４０調節因子 Expired - Fee Related JP5591706B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US99878607P 2007-10-10 2007-10-10
US60/998,786 2007-10-10
US6872408P 2008-03-06 2008-03-06
US61/068,724 2008-03-06
PCT/US2008/011422 WO2009048527A1 (en) 2007-10-10 2008-10-03 Substituted biphenyl gpr40 modulators

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JP2011500562A JP2011500562A (ja) 2011-01-06
JP2011500562A5 JP2011500562A5 (enExample) 2011-11-17
JP5591706B2 true JP5591706B2 (ja) 2014-09-17

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US (1) US8030354B2 (enExample)
EP (1) EP2205548A1 (enExample)
JP (1) JP5591706B2 (enExample)
KR (1) KR20100090249A (enExample)
CN (1) CN102083783A (enExample)
AR (1) AR068840A1 (enExample)
AU (1) AU2008311355B2 (enExample)
BR (1) BRPI0818253A2 (enExample)
CA (1) CA2702047C (enExample)
CL (1) CL2008002997A1 (enExample)
CO (1) CO6270312A2 (enExample)
CR (1) CR11420A (enExample)
IL (1) IL204635A0 (enExample)
MA (1) MA31841B1 (enExample)
MX (1) MX2010003876A (enExample)
PE (1) PE20091222A1 (enExample)
TN (1) TN2010000125A1 (enExample)
TW (1) TW200927091A (enExample)
WO (1) WO2009048527A1 (enExample)

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CN101868452B (zh) 2007-10-10 2014-08-06 诺华股份有限公司 螺环吡咯烷类与其对抗hcv和hiv感染的应用
EP2260017A1 (en) * 2008-03-06 2010-12-15 Amgen, Inc Conformationally constrained carboxylic acid derivatives useful for treating metabolic disorders
CA2739888C (en) * 2008-10-15 2013-11-19 Amgen Inc. Spirocyclic gpr40 modulators
AR074760A1 (es) 2008-12-18 2011-02-09 Metabolex Inc Agonistas del receptor gpr120 y usos de los mismos en medicamentos para el tratamiento de diabetes y el sindrome metabolico.
EA201290574A1 (ru) 2009-12-25 2012-12-28 Мотида Фармасьютикал Ко., Лтд. Новое производное 3-гидрокси-5-арилизотиазола
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2582674B1 (en) * 2010-06-16 2014-10-01 Cymabay Therapeutics, Inc. Gpr120 receptor agonists and uses thereof
US8299117B2 (en) 2010-06-16 2012-10-30 Metabolex Inc. GPR120 receptor agonists and uses thereof
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
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