JP2009535352A5 - - Google Patents

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JP2009535352A5
JP2009535352A5 JP2009507893A JP2009507893A JP2009535352A5 JP 2009535352 A5 JP2009535352 A5 JP 2009535352A5 JP 2009507893 A JP2009507893 A JP 2009507893A JP 2009507893 A JP2009507893 A JP 2009507893A JP 2009535352 A5 JP2009535352 A5 JP 2009535352A5
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hiv
compound
pharmaceutically acceptable
group
acceptable salt
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JP2009507893A
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JP2009535352A (ja
JP5214590B2 (ja
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Priority claimed from US11/733,283 external-priority patent/US7807671B2/en
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Claims (6)

  1. Figure 2009535352
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    :からなる群から選択される化合物。
  2. 請求項1に記載の化合物、またはその医薬的に許容される塩の抗ウイルス有効量、および一つ以上の医薬的に許容される担体、賦形剤または希釈剤を含む、医薬組成物。
  3. 抗HIV活性を有する第2の化合物をさらに含む、請求項2に記載の組成物。
  4. (a)抗AIDSウイルス薬;
    (b)抗感染症薬;
    (c)免疫調節剤; および
    (d)HIV侵入阻害剤
    :からなる群から選択されるAIDS治療薬の抗ウイルス有効量をさらに含む、HIVによる感染を治療するための請求項2に記載の医薬組成物。
  5. HIVを治療するための医薬の製造における、請求項1に記載の化合物、またはその医薬的に許容される塩の使用。
  6. HIVを治療するための医薬の製造における、請求項1に記載の化合物、またはその医薬的に許容される塩、ならびに、抗AIDSウイルス薬; 抗感染症薬; 免疫調節剤; およびHIV侵入阻害剤からなる群から選択されるAIDS治療薬の使用。
JP2009507893A 2006-04-25 2007-04-16 抗ウイルス薬としてのジケト−ピペラジンおよびピペリジン誘導体 Active JP5214590B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US79470306P 2006-04-25 2006-04-25
US79470006P 2006-04-25 2006-04-25
US60/794,703 2006-04-25
US60/794,700 2006-04-25
US11/733,283 US7807671B2 (en) 2006-04-25 2007-04-10 Diketo-piperazine and piperidine derivatives as antiviral agents
US11/733,283 2007-04-10
PCT/US2007/066700 WO2007127635A2 (en) 2006-04-25 2007-04-16 Diketo-piperazine and piperidine derivatives as antiviral agents

Publications (3)

Publication Number Publication Date
JP2009535352A JP2009535352A (ja) 2009-10-01
JP2009535352A5 true JP2009535352A5 (ja) 2010-06-03
JP5214590B2 JP5214590B2 (ja) 2013-06-19

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JP2009507893A Active JP5214590B2 (ja) 2006-04-25 2007-04-16 抗ウイルス薬としてのジケト−ピペラジンおよびピペリジン誘導体

Country Status (17)

Country Link
US (2) US7807671B2 (ja)
EP (1) EP2010525B1 (ja)
JP (1) JP5214590B2 (ja)
KR (1) KR101450349B1 (ja)
AR (1) AR060658A1 (ja)
AU (1) AU2007242989B2 (ja)
BR (1) BRPI0710919A2 (ja)
CA (1) CA2650382C (ja)
EA (1) EA014957B1 (ja)
ES (1) ES2432758T3 (ja)
IL (1) IL194540A (ja)
MX (1) MX2008013265A (ja)
NO (1) NO341412B1 (ja)
NZ (1) NZ571995A (ja)
PE (1) PE20080318A1 (ja)
TW (1) TWI394754B (ja)
WO (1) WO2007127635A2 (ja)

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