JP2009530281A - 代謝障害の治療に有用である二環式カルボン酸誘導体 - Google Patents

代謝障害の治療に有用である二環式カルボン酸誘導体 Download PDF

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JP2009530281A
JP2009530281A JP2009500426A JP2009500426A JP2009530281A JP 2009530281 A JP2009530281 A JP 2009530281A JP 2009500426 A JP2009500426 A JP 2009500426A JP 2009500426 A JP2009500426 A JP 2009500426A JP 2009530281 A JP2009530281 A JP 2009530281A
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JP2009530281A5 (enExample
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シヤルマ，ラジブ
アケルマン，ミツシエル
カルドソ，マリオ・ヘ
ハウズ，ジヨナサン・ビー
リー，アン−ロン
リウ，チンチアン
リウ，ジウエン
マ，チーホワ
メデイナ，ジユリオ・シー
シユミツト，マイケル・ジエイ
スン，イン
ワン，インツアイ
ワン，ジヨンユイ
チユー，リウシヨン
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アムジエン・インコーポレーテツド
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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  • Indole Compounds (AREA)
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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
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JP2009500426A 2006-03-14 2007-03-12 代謝障害の治療に有用である二環式カルボン酸誘導体 Withdrawn JP2009530281A (ja)

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US78270606P 2006-03-14 2006-03-14
US90520707P 2007-03-05 2007-03-05
PCT/US2007/006279 WO2007106469A2 (en) 2006-03-14 2007-03-12 Bicyclic carboxylic acid derivatives useful for treating metabolic disorders

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JP2009530281A true JP2009530281A (ja) 2009-08-27
JP2009530281A5 JP2009530281A5 (enExample) 2010-04-22

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US (1) US20070244155A1 (enExample)
EP (1) EP2001844A2 (enExample)
JP (1) JP2009530281A (enExample)
AR (1) AR059895A1 (enExample)
AU (1) AU2007225208A1 (enExample)
CA (1) CA2646430A1 (enExample)
MX (1) MX2008011615A (enExample)
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Cited By (6)

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JP2013528647A (ja) * 2010-06-16 2013-07-11 メタボレックス， インコーポレイテッド Ｇｐｒ１２０受容体作動薬及びその使用
JP2015503595A (ja) * 2012-01-12 2015-02-02 ジエンス ヘンルイ メデイシンカンパニー リミテッドＪｉａｎｇｓｕ Ｈｅｎｇｒｕｉ Ｍｅｄｉｃｉｎｅ Ｃｏ．，Ｌｔｄ． 多環式化合物誘導体、それらの製造方法および医薬用途
JP2016508506A (ja) * 2013-02-06 2016-03-22 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新しいインダニルオキシジヒドロベンゾフラニル酢酸
JP2016513135A (ja) * 2013-02-28 2016-05-12 エスケー ケミカルズ カンパニー リミテッド 三環式化合物およびその使用
JP2019522043A (ja) * 2016-05-23 2019-08-08 中国医学科学院薬物研究所Ｉｎｓｔｉｔｕｔｅ Ｏｆ Ｍａｔｅｒｉａ Ｍｅｄｉｃａ， Ｃｈｉｎｅｓｅ Ａｃａｄｅｍｙ Ｏｆ Ｍｅｄｉｃａｌ Ｓｃｉｅｎｃｅｓ フェニレート誘導体、調製及び医薬組成物及び使用
JP2020512387A (ja) * 2017-03-31 2020-04-23 武田薬品工業株式会社 代謝性障害の治療の為の置換シクリル酢酸誘導体

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WO2008030618A1 (en) * 2006-09-07 2008-03-13 Amgen Inc. Benzo-fused compounds for use in treating metabolic disorders
EP2064193A1 (en) * 2006-09-07 2009-06-03 Amgen, Inc Heterocyclic gpr40 modulators
WO2008130514A1 (en) * 2007-04-16 2008-10-30 Amgen Inc. Substituted biphenyl phenoxy-, thiophenyl- and aminophenylpropanoic acid gpr40 modulators
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
KR20100090249A (ko) 2007-10-10 2010-08-13 암젠 인크 치환된 비페닐 ｇｒｐ４０ 조절제
EP2215068B1 (en) * 2007-10-29 2012-06-13 Merck Sharp & Dohme Corp. Antidiabetic tricyclic compounds
EP2260017A1 (en) * 2008-03-06 2010-12-15 Amgen, Inc Conformationally constrained carboxylic acid derivatives useful for treating metabolic disorders
KR20220084423A (ko) 2008-07-23 2022-06-21 아레나 파마슈티칼스, 인크. 자가면역성 및 염증성의 장애의 치료에 유용한 치환된 1,2,3,4-테트라히드로시클로펜타[ｂ]인돌-3-일)아세트산 유도체
JP2012503595A (ja) * 2008-07-28 2012-02-09 シダンスク ユニバーシティ 代謝病の治療用の化合物
BRPI0917923B1 (pt) * 2008-08-27 2022-04-05 Arena Pharmaceuticals Inc Derivado de ácido tricíclico substituído, sua composição, seu uso e processo para preparar a referida composição
CA2739888C (en) * 2008-10-15 2013-11-19 Amgen Inc. Spirocyclic gpr40 modulators
EP2690095A1 (en) * 2008-10-21 2014-01-29 Camabay Therapeutics, Inc. Aryl gpr120 receptor agonists and uses thereof
AR074760A1 (es) * 2008-12-18 2011-02-09 Metabolex Inc Agonistas del receptor gpr120 y usos de los mismos en medicamentos para el tratamiento de diabetes y el sindrome metabolico.
EP2389226B1 (en) * 2009-01-23 2013-11-20 Merck Sharp & Dohme Corp. Bridged and fused heterocyclic antidiabetic compounds
AU2010240142A1 (en) * 2009-04-22 2011-11-10 Astellas Pharma Inc. Carboxylic acid compound
JP5856980B2 (ja) 2010-01-27 2016-02-10 アリーナ ファーマシューティカルズ， インコーポレイテッド （Ｒ）−２−（７−（４−シクロペンチル−３−（トリフルオロメチル）ベンジルオキシ）−１，２，３，４−テトラヒドロシクロペンタ［ｂ］インドール−３−イル）酢酸およびその塩の調製のためのプロセス
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
CA2789480A1 (en) 2010-03-03 2011-09-09 Arena Pharmaceuticals, Inc. Processes for the preparation of s1p1 receptor modulators and crystalline forms thereof
US8933024B2 (en) 2010-06-18 2015-01-13 Sanofi Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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