JP2009504780A5 - - Google Patents

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Publication number
JP2009504780A5
JP2009504780A5 JP2008527189A JP2008527189A JP2009504780A5 JP 2009504780 A5 JP2009504780 A5 JP 2009504780A5 JP 2008527189 A JP2008527189 A JP 2008527189A JP 2008527189 A JP2008527189 A JP 2008527189A JP 2009504780 A5 JP2009504780 A5 JP 2009504780A5
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Japan
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aliphatic
carbonyl
aryl
alicyclic
oxy
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JP2008527189A
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English (en)
Japanese (ja)
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JP5203203B2 (ja
JP2009504780A (ja
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Priority claimed from PCT/US2006/032481 external-priority patent/WO2007022459A2/en
Publication of JP2009504780A publication Critical patent/JP2009504780A/ja
Publication of JP2009504780A5 publication Critical patent/JP2009504780A5/ja
Application granted granted Critical
Publication of JP5203203B2 publication Critical patent/JP5203203B2/ja
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Expired - Fee Related legal-status Critical Current

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JP2008527189A 2005-08-19 2006-08-18 製造工程および中間体 Expired - Fee Related JP5203203B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US70996405P 2005-08-19 2005-08-19
US60/709,964 2005-08-19
US81004206P 2006-06-01 2006-06-01
US60/810,042 2006-06-01
PCT/US2006/032481 WO2007022459A2 (en) 2005-08-19 2006-08-18 Processes and intermediates

Publications (3)

Publication Number Publication Date
JP2009504780A JP2009504780A (ja) 2009-02-05
JP2009504780A5 true JP2009504780A5 (enExample) 2009-10-01
JP5203203B2 JP5203203B2 (ja) 2013-06-05

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Family Applications (1)

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JP2008527189A Expired - Fee Related JP5203203B2 (ja) 2005-08-19 2006-08-18 製造工程および中間体

Country Status (24)

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US (3) US7776887B2 (enExample)
EP (4) EP2364970A1 (enExample)
JP (1) JP5203203B2 (enExample)
KR (4) KR20140069370A (enExample)
CN (2) CN101291909B (enExample)
AR (1) AR058025A1 (enExample)
AT (1) ATE463480T1 (enExample)
AU (1) AU2006279357B2 (enExample)
BR (1) BRPI0615029A2 (enExample)
CA (1) CA2619659A1 (enExample)
CY (2) CY1110214T1 (enExample)
DE (1) DE602006013492D1 (enExample)
DK (2) DK2194043T3 (enExample)
ES (2) ES2344156T3 (enExample)
IL (2) IL189585A (enExample)
NZ (3) NZ593214A (enExample)
PL (3) PL385229A1 (enExample)
PT (2) PT2194043E (enExample)
RU (2) RU2446171C2 (enExample)
SG (1) SG2014013338A (enExample)
SI (2) SI1934179T1 (enExample)
TW (2) TW201245149A (enExample)
WO (1) WO2007022459A2 (enExample)
ZA (1) ZA200801791B (enExample)

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ITMI20120800A1 (it) * 2012-05-10 2013-11-11 Dipharma Francis Srl Procedimento per la preparazione di un intermedio utile nella preparazione di un inibitore delle proteasi virali
CN103450066B (zh) * 2012-05-30 2017-03-15 博瑞生物医药（苏州）股份有限公司 特拉匹韦中间体的制备方法
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WO2014019179A1 (zh) * 2012-08-01 2014-02-06 上海迪赛诺药业有限公司 特拉匹韦及其中间体的制备方法
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CN102875648B (zh) * 2012-09-26 2014-02-19 深圳翰宇药业股份有限公司 一种制备特拉匹韦的方法
WO2014053533A1 (en) 2012-10-05 2014-04-10 Sanofi Use of substituted 3-heteroaroylamino-propionic acid derivatives as pharmaceuticals for prevention/treatment of atrial fibrillation
ITMI20122036A1 (it) * 2012-11-29 2014-05-30 Dipharma Francis Srl Sintesi di un intermedio di un composto antivirale
WO2014096343A1 (en) * 2012-12-21 2014-06-26 Sandoz Ag Novel forms of telaprevir
WO2014096374A1 (en) 2012-12-21 2014-06-26 Sandoz Ag Process for the synthesis of pyrrolidines and pyrroles
CN103936651B (zh) * 2013-01-18 2016-06-22 上海医药工业研究院 抗丙肝药物Boceprevir的中间体Ⅲ及其制备方法和应用
ITMI20130706A1 (it) * 2013-04-30 2014-10-31 Dipharma Francis Srl Procedimento per la preparazione di un inibitore delle proteasi virali e suoi intermedi
CN103288671B (zh) * 2013-06-20 2014-10-29 上海步越化工科技有限公司 一种(3s)-3-氨基-n-环丙基-2-羟基己酰胺盐酸盐的合成方法
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CN104292146B (zh) * 2013-06-24 2017-04-26 上海医药工业研究院 特拉匹韦中间体及其制备方法
CN103342656B (zh) * 2013-07-04 2015-04-08 苏州永健生物医药有限公司 特拉匹韦中间体的合成方法
CN103435532B (zh) * 2013-09-02 2015-07-08 苏州永健生物医药有限公司 波普瑞韦中间体的合成方法
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WO2016057931A1 (en) 2014-10-10 2016-04-14 The Research Foundation For The State University Of New York Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration
CN105646329A (zh) * 2014-11-28 2016-06-08 重庆圣华曦药业股份有限公司 一种制备特拉匹韦中间体的方法
CN105111129A (zh) * 2015-08-24 2015-12-02 上海合全药业股份有限公司 (1S,3aR,6aS)-八氢环戊烯并[C]吡咯-1-羧酸叔丁酯草酸盐的制备方法
CN105601556B (zh) * 2015-12-02 2018-11-13 镇江市高等专科学校 特拉匹韦双环吡咯烷中间体的制备方法
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