JP2005539087A5 - - Google Patents

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Publication number
JP2005539087A5
JP2005539087A5 JP2004548887A JP2004548887A JP2005539087A5 JP 2005539087 A5 JP2005539087 A5 JP 2005539087A5 JP 2004548887 A JP2004548887 A JP 2004548887A JP 2004548887 A JP2004548887 A JP 2004548887A JP 2005539087 A5 JP2005539087 A5 JP 2005539087A5
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JP
Japan
Prior art keywords
alkyl
hydroxy
amino
dihydro
oxo
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
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JP2004548887A
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English (en)
Japanese (ja)
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JP4522262B2 (ja
JP2005539087A (ja
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Priority claimed from PCT/EP2003/006756 external-priority patent/WO2004002992A1/en
Publication of JP2005539087A publication Critical patent/JP2005539087A/ja
Publication of JP2005539087A5 publication Critical patent/JP2005539087A5/ja
Application granted granted Critical
Publication of JP4522262B2 publication Critical patent/JP4522262B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2004548887A 2002-06-26 2003-06-25 化合物 Expired - Fee Related JP4522262B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US39170002P 2002-06-26 2002-06-26
US46096103P 2003-04-07 2003-04-07
PCT/EP2003/006756 WO2004002992A1 (en) 2002-06-26 2003-06-25 Compounds

Publications (3)

Publication Number Publication Date
JP2005539087A JP2005539087A (ja) 2005-12-22
JP2005539087A5 true JP2005539087A5 (https=) 2006-06-15
JP4522262B2 JP4522262B2 (ja) 2010-08-11

Family

ID=30003201

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004548887A Expired - Fee Related JP4522262B2 (ja) 2002-06-26 2003-06-25 化合物

Country Status (10)

Country Link
US (2) US7622481B2 (https=)
EP (1) EP1537123B1 (https=)
JP (1) JP4522262B2 (https=)
AR (1) AR040335A1 (https=)
AT (1) ATE430154T1 (https=)
AU (1) AU2003266949A1 (https=)
DE (1) DE60327438D1 (https=)
ES (1) ES2325831T3 (https=)
TW (1) TW200406413A (https=)
WO (1) WO2004002992A1 (https=)

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US8394858B2 (en) 2009-12-03 2013-03-12 Novartis Ag Cyclohexane derivatives and uses thereof
HRP20140005T1 (hr) 2009-12-18 2014-01-31 Basilea Pharmaceutica Ag Tricikliäśki antibiotici
TW201309689A (zh) 2011-02-07 2013-03-01 Daiichi Sankyo Co Ltd 含胺基之吡咯啶酮衍生物
ES2596369T3 (es) 2011-06-17 2017-01-09 Basilea Pharmaceutica Ag Antibióticos N-heterotricíclicos
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US9359275B2 (en) * 2012-02-23 2016-06-07 Children's Medical Center Corporation Natural product antibiotics and analogs thereof
KR20150138214A (ko) * 2013-03-29 2015-12-09 다이이찌 산쿄 가부시키가이샤 (1s,4s,5s)-4-브로모-6-옥사비시클로[3.2.1]옥탄-7-온의 제조 방법
CN103145709A (zh) * 2013-04-12 2013-06-12 苏州科捷生物医药有限公司 一种4-氯-1,6-萘啶的合成工艺
PL2986607T3 (pl) 2013-04-16 2017-11-30 Idorsia Pharmaceuticals Ltd Przeciwbakteryjne pochodne biaromatyczne
WO2015193506A1 (en) * 2014-06-20 2015-12-23 Institut Pasteur Korea Anti-infective compounds
JP6546654B2 (ja) 2014-08-22 2019-07-17 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ 淋菌感染を治療するための三環式含窒素化合物
AR102256A1 (es) 2014-10-15 2017-02-15 Actelion Pharmaceuticals Ltd Derivados biaromáticos básicos antibacterianos con sustitución de aminoalcoxi
KR20200087273A (ko) 2014-10-24 2020-07-20 란도스 바이오파마, 인크. 란티오닌 합성효소 c-유사 2-계 치료제
UY36851A (es) 2015-08-16 2017-03-31 Glaxosmithkline Ip Dev Ltd Compuestos para uso en aplicaciones antibacterianas
WO2019032956A1 (en) 2017-08-10 2019-02-14 President And Fellows Of Harvard College LINCONSAMIDE ANTIBIOTICS AND USES THEREOF
EP3664799B1 (en) * 2017-08-10 2025-10-01 President And Fellows Of Harvard College Lincosamide antibiotics and uses thereof
BR112020010983A2 (pt) 2017-11-30 2020-11-17 Landos Biopharma, Inc método in vitro para gerar células preparadas a partir de células precursoras, células isoladas e método para tratar uma afecção em um animal com as células isoladas
CN108003100A (zh) * 2017-12-20 2018-05-08 北京六合宁远科技有限公司 一种药物中间体含氮杂环的胺类化合物的合成方法
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WO2023125877A1 (zh) 2021-12-30 2023-07-06 上海翰森生物医药科技有限公司 三并环类衍生物抑制剂、其制备方法和应用

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