JP2005525324A5 - - Google Patents

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Publication number
JP2005525324A5
JP2005525324A5 JP2003564044A JP2003564044A JP2005525324A5 JP 2005525324 A5 JP2005525324 A5 JP 2005525324A5 JP 2003564044 A JP2003564044 A JP 2003564044A JP 2003564044 A JP2003564044 A JP 2003564044A JP 2005525324 A5 JP2005525324 A5 JP 2005525324A5
Authority
JP
Japan
Prior art keywords
hydroxy
fluoro
ylamino
ethyl
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2003564044A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005525324A (ja
JP4445753B2 (ja
Filing date
Publication date
Priority claimed from GB0202026A external-priority patent/GB0202026D0/en
Priority claimed from GB0229824A external-priority patent/GB0229824D0/en
Application filed filed Critical
Priority claimed from PCT/EP2003/000823 external-priority patent/WO2003064421A1/en
Publication of JP2005525324A publication Critical patent/JP2005525324A/ja
Publication of JP2005525324A5 publication Critical patent/JP2005525324A5/ja
Application granted granted Critical
Publication of JP4445753B2 publication Critical patent/JP4445753B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2003564044A 2002-01-29 2003-01-27 アミノピペリジン誘導体 Expired - Fee Related JP4445753B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0202026A GB0202026D0 (en) 2002-01-29 2002-01-29 Compounds
GB0229824A GB0229824D0 (en) 2002-12-20 2002-12-20 Compounds
PCT/EP2003/000823 WO2003064421A1 (en) 2002-01-29 2003-01-27 Aminopiperidine derivatives

Publications (3)

Publication Number Publication Date
JP2005525324A JP2005525324A (ja) 2005-08-25
JP2005525324A5 true JP2005525324A5 (https=) 2006-01-12
JP4445753B2 JP4445753B2 (ja) 2010-04-07

Family

ID=27665357

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003564044A Expired - Fee Related JP4445753B2 (ja) 2002-01-29 2003-01-27 アミノピペリジン誘導体

Country Status (6)

Country Link
US (1) US7312212B2 (https=)
EP (2) EP1470125A1 (https=)
JP (1) JP4445753B2 (https=)
AR (1) AR038240A1 (https=)
TW (1) TW200406410A (https=)
WO (1) WO2003064421A1 (https=)

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CN102232078B (zh) * 2008-12-12 2014-07-16 埃科特莱茵药品有限公司 5-氨基-2-(1-羟基-乙基)-四氢吡喃衍生物
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UA108618C2 (uk) 2009-08-07 2015-05-25 Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку
US9059778B2 (en) * 2011-01-07 2015-06-16 Integrated Device Technology Inc. Frequency domain compression in a base transceiver system
JP5918624B2 (ja) * 2012-05-18 2016-05-18 東ソ−・エフテック株式会社 光学活性含フッ素５，６−ジヒドロピリドン誘導体及びその製造方法
CN102702080B (zh) * 2012-06-21 2014-02-19 扬州氟药科技有限公司 一种3-三氟甲基哌啶衍生物的制备方法
WO2016004297A1 (en) * 2014-07-02 2016-01-07 Board Of Regents, The University Of Texas System Novel inhibitors of trypanosoma brucei methionyl t-rna synthetase (tb metrs) for the treatment of african trypanosomiasis
JP6546654B2 (ja) 2014-08-22 2019-07-17 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ 淋菌感染を治療するための三環式含窒素化合物
UY36851A (es) 2015-08-16 2017-03-31 Glaxosmithkline Ip Dev Ltd Compuestos para uso en aplicaciones antibacterianas
CN114957114A (zh) * 2021-02-26 2022-08-30 冷志 一种4-溴-3-氯-7-甲氧基喹啉的合成方法

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WO2004035569A2 (de) 2002-10-10 2004-04-29 Morphochem Aktiengesellschaft für kombinatorische Chemie Neue verbindungen mit antibakterieller aktivität
DE60331849D1 (de) 2002-11-05 2010-05-06 Glaxosmithkline Llc Antibakterielle wirkstoffe
ATE479683T1 (de) 2002-11-05 2010-09-15 Glaxo Group Ltd Antibakterielle mittel
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TW200427688A (en) 2002-12-18 2004-12-16 Glaxo Group Ltd Antibacterial agents

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