JP2002517396A - 細胞接着阻害抗炎症性化合物 - Google Patents

細胞接着阻害抗炎症性化合物

Info

Publication number
JP2002517396A
JP2002517396A JP2000552119A JP2000552119A JP2002517396A JP 2002517396 A JP2002517396 A JP 2002517396A JP 2000552119 A JP2000552119 A JP 2000552119A JP 2000552119 A JP2000552119 A JP 2000552119A JP 2002517396 A JP2002517396 A JP 2002517396A
Authority
JP
Japan
Prior art keywords
thieno
pyridine
carboxamide
chlorophenoxy
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2000552119A
Other languages
English (en)
Japanese (ja)
Inventor
スチユアート,アンドリユー・オー
ボイド,ステイーブン・エイ
アレンドセン,デイビツド・エル
バーテイア,プラミラ
コンドロスキー,ケビン・アール
フリーマン,ジエニフアー・シー
グナワーダナ,インダラニ・ダブリユ
チユー,コイ−トン
ラーテイ,クレイグ
マツカーテイ,キヤサリン・エム
モート,ニコラス・エイ
パテル,ミーナ・ブイ
ステイガー,マイケル・エイ
スタウト,デイビツド・エム
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of JP2002517396A publication Critical patent/JP2002517396A/ja
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP2000552119A 1998-06-04 1999-06-03 細胞接着阻害抗炎症性化合物 Withdrawn JP2002517396A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9070198A 1998-06-04 1998-06-04
US09/090,701 1998-06-04
PCT/US1999/012419 WO1999062908A2 (fr) 1998-06-04 1999-06-03 Composes anti-inflammatoires inhibant l'adhesion cellulaire

Publications (1)

Publication Number Publication Date
JP2002517396A true JP2002517396A (ja) 2002-06-18

Family

ID=22223903

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000552119A Withdrawn JP2002517396A (ja) 1998-06-04 1999-06-03 細胞接着阻害抗炎症性化合物

Country Status (15)

Country Link
EP (1) EP1090009A2 (fr)
JP (1) JP2002517396A (fr)
KR (1) KR20010052570A (fr)
CN (1) CN1332743A (fr)
AU (1) AU4231299A (fr)
BG (1) BG105109A (fr)
BR (1) BR9910864A (fr)
CA (1) CA2333770A1 (fr)
HU (1) HUP0102366A2 (fr)
IL (1) IL139811A0 (fr)
NO (1) NO20006157L (fr)
PL (1) PL345906A1 (fr)
SK (1) SK18542000A3 (fr)
TR (1) TR200100189T2 (fr)
WO (1) WO1999062908A2 (fr)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006516610A (ja) * 2003-02-05 2006-07-06 リモニクス ファーマシューティカルズ リミテッド チエノ[2,3−c]ピリジン誘導体を含む薬剤組成物、及びその使用
JP2007536301A (ja) * 2004-05-04 2007-12-13 エフ.ホフマン−ラ ロシュ アーゲー Ikk阻害剤としてのチエノピリダジン
JP2007536303A (ja) * 2004-05-04 2007-12-13 エフ.ホフマン−ラ ロシュ アーゲー Ikk阻害剤としてのチエノピリジン
JP2008517936A (ja) * 2004-10-21 2008-05-29 ダウ アグロサイエンシィズ エルエルシー 殺真菌活性を有するチエノ−ピリミジン化合物

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AU4231299A (en) 1999-12-20
HUP0102366A2 (hu) 2001-11-28
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BR9910864A (pt) 2002-02-05
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EP1090009A2 (fr) 2001-04-11
CA2333770A1 (fr) 1999-12-09
PL345906A1 (en) 2002-01-14
NO20006157L (no) 2001-02-02
WO1999062908A3 (fr) 2000-03-30
CN1332743A (zh) 2002-01-23
BG105109A (en) 2001-11-30

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