BG105109A - Cell adhesion-inhibiting anti-inflammatory compounds - Google Patents

Cell adhesion-inhibiting anti-inflammatory compounds

Info

Publication number
BG105109A
BG105109A BG105109A BG10510901A BG105109A BG 105109 A BG105109 A BG 105109A BG 105109 A BG105109 A BG 105109A BG 10510901 A BG10510901 A BG 10510901A BG 105109 A BG105109 A BG 105109A
Authority
BG
Bulgaria
Prior art keywords
cell adhesion
inflammatory compounds
inhibiting anti
compounds
inhibiting
Prior art date
Application number
BG105109A
Other languages
Bulgarian (bg)
Inventor
Andrew Stewart
Steven Boyd
David ARENDSEN
Pramila Bhatia
Kevin CONDROSKI
Jennifer Freeman
Indrani Gunawardana
Gui-Dong Zhu
Kraig Lartey
Catherine MCCARTY
Nicholas MORT
Meena Patel
Michael Staeger
David STOUT
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of BG105109A publication Critical patent/BG105109A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Compounds having formula are useful for treating inflammation. Also disclosed are pharmaceutical compositions comprising said compounds, and methods of inhibiting/treating inflammatory diseases in a mammal. 23 claims, 1 figure
BG105109A 1998-06-04 2001-01-03 Cell adhesion-inhibiting anti-inflammatory compounds BG105109A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9070198A 1998-06-04 1998-06-04
PCT/US1999/012419 WO1999062908A2 (en) 1998-06-04 1999-06-03 Cell adhesion-inhibiting antinflammatory compounds

Publications (1)

Publication Number Publication Date
BG105109A true BG105109A (en) 2001-11-30

Family

ID=22223903

Family Applications (1)

Application Number Title Priority Date Filing Date
BG105109A BG105109A (en) 1998-06-04 2001-01-03 Cell adhesion-inhibiting anti-inflammatory compounds

Country Status (15)

Country Link
EP (1) EP1090009A2 (en)
JP (1) JP2002517396A (en)
KR (1) KR20010052570A (en)
CN (1) CN1332743A (en)
AU (1) AU4231299A (en)
BG (1) BG105109A (en)
BR (1) BR9910864A (en)
CA (1) CA2333770A1 (en)
HU (1) HUP0102366A2 (en)
IL (1) IL139811A0 (en)
NO (1) NO20006157L (en)
PL (1) PL345906A1 (en)
SK (1) SK18542000A3 (en)
TR (1) TR200100189T2 (en)
WO (1) WO1999062908A2 (en)

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