IN2014MN00258A - - Google Patents

Info

Publication number
IN2014MN00258A
IN2014MN00258A IN258MUN2014A IN2014MN00258A IN 2014MN00258 A IN2014MN00258 A IN 2014MN00258A IN 258MUN2014 A IN258MUN2014 A IN 258MUN2014A IN 2014MN00258 A IN2014MN00258 A IN 2014MN00258A
Authority
IN
India
Prior art keywords
compounds
present
novel
medicament
concerned
Prior art date
Application number
Other languages
English (en)
Inventor
Garrett Berlond Minne
François Paul Bischoff
Henricus Jacobus Maria Gijsen
Adriana Ingrid Velter
Serge Maria Aloysius Pieters
Didier Jean Claude Berthelot
Original Assignee
Janssen Pharmaceuticals Inc
Cellzome Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceuticals Inc, Cellzome Ltd filed Critical Janssen Pharmaceuticals Inc
Publication of IN2014MN00258A publication Critical patent/IN2014MN00258A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Indole Compounds (AREA)
IN258MUN2014 2011-07-15 2012-07-12 IN2014MN00258A (OSRAM)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP11174120 2011-07-15
PCT/EP2012/063667 WO2013010904A1 (en) 2011-07-15 2012-07-12 Novel substituted indole derivatives as gamma secretase modulators

Publications (1)

Publication Number Publication Date
IN2014MN00258A true IN2014MN00258A (OSRAM) 2015-09-25

Family

ID=46506432

Family Applications (1)

Application Number Title Priority Date Filing Date
IN258MUN2014 IN2014MN00258A (OSRAM) 2011-07-15 2012-07-12

Country Status (16)

Country Link
US (1) US9115143B2 (OSRAM)
EP (1) EP2731948B1 (OSRAM)
JP (1) JP6068464B2 (OSRAM)
KR (1) KR101913135B1 (OSRAM)
CN (1) CN103874702B (OSRAM)
AR (1) AR087182A1 (OSRAM)
AU (1) AU2012285931B2 (OSRAM)
BR (1) BR112014000713A2 (OSRAM)
CA (1) CA2841102C (OSRAM)
EA (1) EA023045B1 (OSRAM)
ES (1) ES2555167T3 (OSRAM)
IL (1) IL230422B (OSRAM)
IN (1) IN2014MN00258A (OSRAM)
MX (1) MX2014000626A (OSRAM)
TW (1) TWI567079B (OSRAM)
WO (1) WO2013010904A1 (OSRAM)

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AU2018390610A1 (en) 2017-12-20 2020-08-06 Bristol-Myers Squibb Company Amino indole compounds useful as TLR inhibitors
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ES2987832T3 (es) 2019-05-09 2024-11-18 Bristol Myers Squibb Co Compuestos de benzimidazolona sustituidos
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Also Published As

Publication number Publication date
NZ619683A (en) 2015-01-30
TW201315736A (zh) 2013-04-16
CN103874702A (zh) 2014-06-18
CA2841102A1 (en) 2013-01-24
BR112014000713A2 (pt) 2017-01-10
EA023045B1 (ru) 2016-04-29
WO2013010904A1 (en) 2013-01-24
KR101913135B1 (ko) 2018-10-30
US9115143B2 (en) 2015-08-25
JP2014518286A (ja) 2014-07-28
JP6068464B2 (ja) 2017-01-25
ES2555167T3 (es) 2015-12-29
MX2014000626A (es) 2014-04-30
AU2012285931B2 (en) 2017-01-12
EP2731948B1 (en) 2015-09-09
TWI567079B (zh) 2017-01-21
EP2731948A1 (en) 2014-05-21
CN103874702B (zh) 2015-12-09
US20140148450A1 (en) 2014-05-29
KR20140063595A (ko) 2014-05-27
EA201490287A1 (ru) 2014-05-30
IL230422B (en) 2018-03-29
CA2841102C (en) 2019-08-13
AR087182A1 (es) 2014-02-26

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