IN2013MN02170A - - Google Patents

Info

Publication number
IN2013MN02170A
IN2013MN02170A IN2170MUN2013A IN2013MN02170A IN 2013MN02170 A IN2013MN02170 A IN 2013MN02170A IN 2170MUN2013 A IN2170MUN2013 A IN 2170MUN2013A IN 2013MN02170 A IN2013MN02170 A IN 2013MN02170A
Authority
IN
India
Prior art keywords
compounds
formula
preparation
relates
present
Prior art date
Application number
Other languages
English (en)
Inventor
Malcolm Mascarenhas
Shashikant Patil
Ravindra Ashok Janrao
Abhijit Roychowdhury
Original Assignee
Piramal Entpr Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Piramal Entpr Ltd filed Critical Piramal Entpr Ltd
Publication of IN2013MN02170A publication Critical patent/IN2013MN02170A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IN2170MUN2013 2011-04-21 2012-04-19 IN2013MN02170A (enExample)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161477937P 2011-04-21 2011-04-21
PCT/IB2012/051958 WO2012143874A1 (en) 2011-04-21 2012-04-19 A process for the preparation of morpholino sulfonyl indole derivatives

Publications (1)

Publication Number Publication Date
IN2013MN02170A true IN2013MN02170A (enExample) 2015-06-12

Family

ID=46026953

Family Applications (1)

Application Number Title Priority Date Filing Date
IN2170MUN2013 IN2013MN02170A (enExample) 2011-04-21 2012-04-19

Country Status (9)

Country Link
US (3) US20140046059A1 (enExample)
EP (2) EP2699567A1 (enExample)
JP (1) JP2014514321A (enExample)
CN (1) CN103732592A (enExample)
AU (2) AU2012245455A1 (enExample)
CA (2) CA2831730A1 (enExample)
IL (1) IL228810A0 (enExample)
IN (1) IN2013MN02170A (enExample)
WO (3) WO2012145471A1 (enExample)

Families Citing this family (11)

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Publication number Priority date Publication date Assignee Title
WO2012145471A1 (en) * 2011-04-21 2012-10-26 Merck Sharp & Dohme Corp. Insulin-like growth factor-1 receptor inhibitors
WO2014002007A1 (en) * 2012-06-26 2014-01-03 Piramal Enterprises Limited Method of predicting or monitoring response to igf-1r and ir inhibitors using biomarkers
KR102196374B1 (ko) 2012-11-29 2020-12-31 케모센트릭스, 인크. Cxcr7 길항제
WO2014177915A1 (en) 2013-05-01 2014-11-06 Piramal Enterprises Limited Cancer combination therapy using imidazo[4,5-c]quinoline derivatives
CN104098498A (zh) * 2014-07-30 2014-10-15 天津市斯芬克司药物研发有限公司 一种吲唑类化合物及其制备方法
CN107003600A (zh) 2014-09-15 2017-08-01 德米特里·戈里洛夫斯基 包括观察大场景的多个数字照相机的系统
CN105218475A (zh) * 2015-10-15 2016-01-06 湖南华腾制药有限公司 1,2-吗啉盐酸盐的合成方法
MX2020006219A (es) * 2017-12-15 2020-12-03 Inthera Bioscience AG Derivados de 1-piperidinocarbonilmetil)-2-oxopiperazina para tratar cancer.
CN113194956A (zh) 2018-12-12 2021-07-30 凯莫森特里克斯股份有限公司 用于癌症治疗的cxcr7抑制剂
CN113149941A (zh) * 2020-01-22 2021-07-23 中国科学院上海药物研究所 醚类化合物及其在防治糖尿病及代谢综合征中的药学用途
TW202509078A (zh) 2023-07-07 2025-03-01 美商維里迪恩醫療股份有限公司 治療慢性甲狀腺眼病之方法

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US20140046059A1 (en) 2014-02-13
WO2012143874A1 (en) 2012-10-26
JP2014514321A (ja) 2014-06-19
AU2012245455A8 (en) 2013-11-07
US20140045847A1 (en) 2014-02-13
AU2012245455A1 (en) 2013-10-31
AU2012245971A1 (en) 2013-10-17
EP2699567A1 (en) 2014-02-26
EP2699568A1 (en) 2014-02-26
CA2831730A1 (en) 2012-10-26
IL228810A0 (en) 2013-12-31

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