IL164162A0 - 5Ht2c receptor modulators - Google Patents

5Ht2c receptor modulators

Info

Publication number
IL164162A0
IL164162A0 IL16416203A IL16416203A IL164162A0 IL 164162 A0 IL164162 A0 IL 164162A0 IL 16416203 A IL16416203 A IL 16416203A IL 16416203 A IL16416203 A IL 16416203A IL 164162 A0 IL164162 A0 IL 164162A0
Authority
IL
Israel
Prior art keywords
disorder
age
mental
pain
depression
Prior art date
Application number
IL16416203A
Other languages
English (en)
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29255581&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL164162(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of IL164162A0 publication Critical patent/IL164162A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A—HUMAN NECESSITIES
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Emergency Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Vascular Medicine (AREA)
  • Pregnancy & Childbirth (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
IL16416203A 2002-04-12 2003-04-11 5Ht2c receptor modulators IL164162A0 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US37205802P 2002-04-12 2002-04-12
US40549502P 2002-08-23 2002-08-23
US43460702P 2002-12-18 2002-12-18
US10/410,991 US6953787B2 (en) 2002-04-12 2003-04-10 5HT2C receptor modulators
PCT/US2003/011076 WO2003086306A2 (en) 2002-04-12 2003-04-11 5ht2c receptor modulators

Publications (1)

Publication Number Publication Date
IL164162A0 true IL164162A0 (en) 2005-12-18

Family

ID=29255581

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16416203A IL164162A0 (en) 2002-04-12 2003-04-11 5Ht2c receptor modulators

Country Status (28)

Country Link
US (11) US6953787B2 (cg-RX-API-DMAC7.html)
EP (4) EP1557409A1 (cg-RX-API-DMAC7.html)
JP (5) JP4155926B2 (cg-RX-API-DMAC7.html)
KR (3) KR100908167B1 (cg-RX-API-DMAC7.html)
CN (5) CN101486679A (cg-RX-API-DMAC7.html)
AT (1) ATE294781T1 (cg-RX-API-DMAC7.html)
AU (1) AU2003221866B2 (cg-RX-API-DMAC7.html)
BR (2) BR122017023795B8 (cg-RX-API-DMAC7.html)
CA (1) CA2481723C (cg-RX-API-DMAC7.html)
CR (2) CR7503A (cg-RX-API-DMAC7.html)
DE (1) DE60300610T2 (cg-RX-API-DMAC7.html)
DK (1) DK1411881T3 (cg-RX-API-DMAC7.html)
ES (2) ES2670568T3 (cg-RX-API-DMAC7.html)
GE (1) GEP20074197B (cg-RX-API-DMAC7.html)
IL (1) IL164162A0 (cg-RX-API-DMAC7.html)
IS (1) IS2134B (cg-RX-API-DMAC7.html)
MX (1) MXPA04009965A (cg-RX-API-DMAC7.html)
MY (1) MY141476A (cg-RX-API-DMAC7.html)
NO (1) NO323528B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ535381A (cg-RX-API-DMAC7.html)
PL (4) PL219017B1 (cg-RX-API-DMAC7.html)
PT (1) PT1411881E (cg-RX-API-DMAC7.html)
RU (1) RU2317982C2 (cg-RX-API-DMAC7.html)
SI (1) SI1411881T1 (cg-RX-API-DMAC7.html)
TW (1) TWI252105B (cg-RX-API-DMAC7.html)
UA (1) UA77788C2 (cg-RX-API-DMAC7.html)
WO (1) WO2003086306A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA200408506B (cg-RX-API-DMAC7.html)

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US8478824B2 (en) * 2002-02-05 2013-07-02 Portauthority Technologies Inc. Apparatus and method for controlling unauthorized dissemination of electronic mail
SE0200968D0 (sv) * 2002-03-26 2002-03-26 Lars Baltzer Novel polypeptide scaffolds and use thereof
US6953787B2 (en) * 2002-04-12 2005-10-11 Arena Pharmaceuticals, Inc. 5HT2C receptor modulators
US7595311B2 (en) 2002-05-24 2009-09-29 Exelixis, Inc. Azepinoindole derivatives as pharmaceutical agents
TWI329111B (en) 2002-05-24 2010-08-21 X Ceptor Therapeutics Inc Azepinoindole and pyridoindole derivatives as pharmaceutical agents
TWI323256B (en) 2002-12-20 2010-04-11 Glaxo Group Ltd Novel benzazepine derivatives and pharmaceutical compositions comprising said compounds
EA016558B1 (ru) * 2003-06-17 2012-05-30 Арена Фармасьютикалз, Инк. Производные бензазепина, используемые для лечения заболеваний, ассоциированных с 5-ht-рецептором
SI2332921T1 (sl) 2003-06-17 2016-06-30 Arena Pharmaceuticals, Inc. 8-kloro-1-metil-2,3,4,5-tetrahidro-1H-3-benzazapin hidroklorid
TW200510324A (en) * 2003-08-11 2005-03-16 Lilly Co Eli 6-(2,2,2-trifluoroethylamino)-7-chiloro-2, 3, 4, 5-tetrahydro-1h-benzo[d]azepine as a 5-ht2c receptor agonist
US20080009478A1 (en) * 2003-10-22 2008-01-10 Arena Pharmaceuticals, Inc. Benzazepine Derivatives and Methods of Prophylaxis or Treatment of 5Ht2c Receptor Associated Diseases
US20070275949A1 (en) * 2003-10-22 2007-11-29 Arena Pharmaceuticals, Inc. Benzazepine Derivatives and Methods of Prophylaxis or Treatment of 5Ht2C Receptor Associated Diseases
RU2006117366A (ru) * 2003-10-23 2007-12-10 Ф.Хоффманн-Ля Рош Аг (Ch) Производные бензазепина в качестве ингибиторов мао-в
JP4796047B2 (ja) 2004-02-25 2011-10-19 イーライ リリー アンド カンパニー ５−ＨＴ２Ｃ受容体作用薬としての６−置換２，３，４，５−テトラヒドロ−１Ｈ−ベンゾ［ｄ］アゼピン
WO2006022420A1 (ja) 2004-08-25 2006-03-02 Takeda Pharmaceutical Company Limited 腹圧性尿失禁の予防・治療剤及びそのスクリーニング方法
DK1796663T3 (da) * 2004-09-03 2011-08-15 Athersys Inc Tricykliske heteroaryl-piperaziner, pyrrolidiner og azetidiner som serotonin-receptor-modulatorer
US7528175B2 (en) * 2004-10-08 2009-05-05 Inverseon, Inc. Method of treating airway diseases with beta-adrenergic inverse agonists
WO2006044762A2 (en) * 2004-10-15 2006-04-27 Bayer Pharmaceuticals Corporation Tetrahydro-5h-pyrimido[4,5-d]azepine derivatives useful for the treatment of diseases associated with the 5-ht2c receptor
MX2007007103A (es) * 2004-12-13 2008-03-10 Lilly Co Eli Derivados espiro como inhibidores de lipoxigenasa.
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JP2009001584A (ja) 2009-01-08
CN101486678A (zh) 2009-07-22
HK1064095A1 (en) 2005-01-21
ES2670568T3 (es) 2018-05-31
US20160024014A1 (en) 2016-01-28
JP2006143751A (ja) 2006-06-08
CN101485664A (zh) 2009-07-22
IS2134B (is) 2006-08-15
BRPI0309303B8 (pt) 2021-05-25
PT1411881E (pt) 2005-09-30
US20130217676A1 (en) 2013-08-22
US6953787B2 (en) 2005-10-11
MY141476A (en) 2010-04-30
PL231405B1 (pl) 2019-02-28
US20130012495A1 (en) 2013-01-10
JP2005527579A (ja) 2005-09-15
CR10393A (es) 2008-11-11
CN101486677A (zh) 2009-07-22
ES2242165T3 (es) 2005-11-01
BR0309303A (pt) 2005-04-26
CN101486679A (zh) 2009-07-22
PL396873A1 (pl) 2012-01-30
JP4155926B2 (ja) 2008-09-24
MXPA04009965A (es) 2005-09-30
JP2012006970A (ja) 2012-01-12
US8273734B1 (en) 2012-09-25
CN101486677B (zh) 2012-12-12
ATE294781T1 (de) 2005-05-15
BRPI0309303B1 (pt) 2018-05-29
WO2003086306A3 (en) 2004-02-19
WO2003086306A2 (en) 2003-10-23
CN1646493A (zh) 2005-07-27
US20070060568A1 (en) 2007-03-15
EP1411881A4 (en) 2004-07-07
RU2317982C2 (ru) 2008-02-27
US8207158B2 (en) 2012-06-26
CA2481723A1 (en) 2003-10-23
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JP4966929B2 (ja) 2012-07-04
TWI252105B (en) 2006-04-01
US20150045552A1 (en) 2015-02-12
KR100908166B1 (ko) 2009-07-16
US7977329B2 (en) 2011-07-12
US20120135982A1 (en) 2012-05-31
NO323528B1 (no) 2007-06-04
IS7490A (is) 2004-10-06
EP1557409A1 (en) 2005-07-27
PL211314B1 (pl) 2012-05-31
SI1411881T1 (en) 2005-10-31
RU2004133068A (ru) 2005-04-20
JP4191741B2 (ja) 2008-12-03
DE60300610D1 (de) 2005-06-09
CA2481723C (en) 2008-02-19
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US20120252788A1 (en) 2012-10-04
KR100812925B1 (ko) 2008-03-11
US8575149B2 (en) 2013-11-05
BR122017023795B1 (pt) 2020-11-24
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CR7503A (es) 2005-04-27

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