IL163691A0 - 5-Pphenylthiazole derivatives and use as pi3 kinase - Google Patents

5-Pphenylthiazole derivatives and use as pi3 kinase

Info

Publication number
IL163691A0
IL163691A0 IL16369103A IL16369103A IL163691A0 IL 163691 A0 IL163691 A0 IL 163691A0 IL 16369103 A IL16369103 A IL 16369103A IL 16369103 A IL16369103 A IL 16369103A IL 163691 A0 IL163691 A0 IL 163691A0
Authority
IL
Israel
Prior art keywords
pphenylthiazole
kinase
derivatives
pphenylthiazole derivatives
Prior art date
Application number
IL16369103A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27767104&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL163691(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0204765A external-priority patent/GB0204765D0/en
Priority claimed from GB0229626A external-priority patent/GB0229626D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of IL163691A0 publication Critical patent/IL163691A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
IL16369103A 2002-02-28 2003-02-27 5-Pphenylthiazole derivatives and use as pi3 kinase IL163691A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0204765A GB0204765D0 (en) 2002-02-28 2002-02-28 Organic compounds
GB0229626A GB0229626D0 (en) 2002-12-19 2002-12-19 Organic compounds
PCT/EP2003/002036 WO2003072557A1 (en) 2002-02-28 2003-02-27 5-phenylthiazole derivatives and use as pi3 kinase inhibitors

Publications (1)

Publication Number Publication Date
IL163691A0 true IL163691A0 (en) 2005-12-18

Family

ID=27767104

Family Applications (2)

Application Number Title Priority Date Filing Date
IL16369103A IL163691A0 (en) 2002-02-28 2003-02-27 5-Pphenylthiazole derivatives and use as pi3 kinase
IL163691A IL163691A (en) 2002-02-28 2004-08-23 5-phenylthiazole derivatives, process for their preparation, compositions comprising them and use thereof in the preparation of medicaments for the treatment of diseases mediated by pi3 kinase

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL163691A IL163691A (en) 2002-02-28 2004-08-23 5-phenylthiazole derivatives, process for their preparation, compositions comprising them and use thereof in the preparation of medicaments for the treatment of diseases mediated by pi3 kinase

Country Status (28)

Country Link
US (2) US7687637B2 (es)
EP (1) EP1480962B1 (es)
JP (2) JP4408701B2 (es)
KR (1) KR100688370B1 (es)
CN (1) CN100548996C (es)
AR (1) AR038703A1 (es)
AT (1) ATE521598T1 (es)
AU (1) AU2003214080A1 (es)
BR (1) BR0308030A (es)
CA (1) CA2477601C (es)
CO (1) CO5611131A2 (es)
CY (2) CY1112084T1 (es)
DK (2) DK1480962T3 (es)
EC (2) ECSP045253A (es)
ES (2) ES2405816T3 (es)
HK (1) HK1071363A1 (es)
IL (2) IL163691A0 (es)
MX (1) MXPA04008362A (es)
MY (1) MY156407A (es)
NO (1) NO329175B1 (es)
NZ (1) NZ534657A (es)
PE (1) PE20030968A1 (es)
PL (2) PL215581B1 (es)
PT (2) PT2311818E (es)
RU (2) RU2436780C2 (es)
SI (1) SI1480962T1 (es)
TW (1) TWI314928B (es)
WO (1) WO2003072557A1 (es)

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