HRP20170786T1 - Modulatori estrogenskog receptora i njihove uporabe - Google Patents

Modulatori estrogenskog receptora i njihove uporabe Download PDF

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Publication number
HRP20170786T1
HRP20170786T1 HRP20170786TT HRP20170786T HRP20170786T1 HR P20170786 T1 HRP20170786 T1 HR P20170786T1 HR P20170786T T HRP20170786T T HR P20170786TT HR P20170786 T HRP20170786 T HR P20170786T HR P20170786 T1 HRP20170786 T1 HR P20170786T1
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HR
Croatia
Prior art keywords
phenyl
methyl
methylpyrrolidin
propoxy
substituted
Prior art date
Application number
HRP20170786TT
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English (en)
Croatian (hr)
Inventor
Mehmet Kahraman
Steven P. Govek
Johnny Y. Nagasawa
Nicholas D. Smith
Original Assignee
Seragon Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Seragon Pharmaceuticals, Inc. filed Critical Seragon Pharmaceuticals, Inc.
Publication of HRP20170786T1 publication Critical patent/HRP20170786T1/hr

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • AHUMAN NECESSITIES
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    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/3533,4-Dihydrobenzopyrans, e.g. chroman, catechin
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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HRP20170786TT 2010-06-10 2011-06-08 Modulatori estrogenskog receptora i njihove uporabe HRP20170786T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35353110P 2010-06-10 2010-06-10
PCT/US2011/039669 WO2011156518A2 (en) 2010-06-10 2011-06-08 Estrogen receptor modulators and uses thereof
EP11793115.4A EP2580210B1 (en) 2010-06-10 2011-06-08 Estrogen receptor modulators and uses thereof

Publications (1)

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HRP20170786T1 true HRP20170786T1 (hr) 2017-08-11

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HRP20170786TT HRP20170786T1 (hr) 2010-06-10 2011-06-08 Modulatori estrogenskog receptora i njihove uporabe

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US (2) US8703810B2 (enExample)
EP (2) EP2580210B1 (enExample)
JP (3) JP2013528223A (enExample)
KR (1) KR101698238B1 (enExample)
CN (1) CN102939287B (enExample)
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