SG185637A1 - Estrogen receptor modulators and uses thereof - Google Patents

Estrogen receptor modulators and uses thereof Download PDF

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Publication number
SG185637A1
SG185637A1 SG2012084737A SG2012084737A SG185637A1 SG 185637 A1 SG185637 A1 SG 185637A1 SG 2012084737 A SG2012084737 A SG 2012084737A SG 2012084737 A SG2012084737 A SG 2012084737A SG 185637 A1 SG185637 A1 SG 185637A1
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Singapore
Prior art keywords
substituted
unsubstituted
phenyl
methyl
chromen
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SG2012084737A
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English (en)
Inventor
Mehmet Kahraman
Steven P Govek
Johnny Y Nagasawa
Nicholas D Smith
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Aragon Pharmaceuticals Inc
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Publication of SG185637A1 publication Critical patent/SG185637A1/en

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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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SG2012084737A 2010-06-10 2011-06-08 Estrogen receptor modulators and uses thereof SG185637A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35353110P 2010-06-10 2010-06-10
PCT/US2011/039669 WO2011156518A2 (en) 2010-06-10 2011-06-08 Estrogen receptor modulators and uses thereof

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