KR101698238B1 - 에스트로겐 수용체 조정제 및 이의 용도 - Google Patents
에스트로겐 수용체 조정제 및 이의 용도 Download PDFInfo
- Publication number
- KR101698238B1 KR101698238B1 KR1020137000592A KR20137000592A KR101698238B1 KR 101698238 B1 KR101698238 B1 KR 101698238B1 KR 1020137000592 A KR1020137000592 A KR 1020137000592A KR 20137000592 A KR20137000592 A KR 20137000592A KR 101698238 B1 KR101698238 B1 KR 101698238B1
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- South Korea
- Prior art keywords
- substituted
- unsubstituted
- chromen
- methyl
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 CC1C2=C(C(*)=C(C(*)(*3)C4C=CC(*CC(*)*5CC*(*)CC5)=CC4(C)C)C4=CC*(*)CC=C4)C3=CC(C)*C2C1COC Chemical compound CC1C2=C(C(*)=C(C(*)(*3)C4C=CC(*CC(*)*5CC*(*)CC5)=CC4(C)C)C4=CC*(*)CC=C4)C3=CC(C)*C2C1COC 0.000 description 17
- ONQBOTKLCMXPOF-UHFFFAOYSA-N CCN1CCCC1 Chemical compound CCN1CCCC1 ONQBOTKLCMXPOF-UHFFFAOYSA-N 0.000 description 4
- DQAIQTUGEVDNDQ-UHFFFAOYSA-N CC(COC(C)=O)N(C(CC1(C)C)=O)C1=O Chemical compound CC(COC(C)=O)N(C(CC1(C)C)=O)C1=O DQAIQTUGEVDNDQ-UHFFFAOYSA-N 0.000 description 1
- XBHXPWCJPBZNRP-UHFFFAOYSA-N CC(C[O]=C)N1CCCC1 Chemical compound CC(C[O]=C)N1CCCC1 XBHXPWCJPBZNRP-UHFFFAOYSA-N 0.000 description 1
Classifications
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- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
- A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35353110P | 2010-06-10 | 2010-06-10 | |
| US61/353,531 | 2010-06-10 | ||
| PCT/US2011/039669 WO2011156518A2 (en) | 2010-06-10 | 2011-06-08 | Estrogen receptor modulators and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20130082496A KR20130082496A (ko) | 2013-07-19 |
| KR101698238B1 true KR101698238B1 (ko) | 2017-01-19 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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