JP2013528223A - エストロゲン受容体モジュレーターおよびその用途 - Google Patents
エストロゲン受容体モジュレーターおよびその用途 Download PDFInfo
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- JP2013528223A JP2013528223A JP2013514346A JP2013514346A JP2013528223A JP 2013528223 A JP2013528223 A JP 2013528223A JP 2013514346 A JP2013514346 A JP 2013514346A JP 2013514346 A JP2013514346 A JP 2013514346A JP 2013528223 A JP2013528223 A JP 2013528223A
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- substituted
- unsubstituted
- phenyl
- chromene
- methyl
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
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- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
- A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35353110P | 2010-06-10 | 2010-06-10 | |
| US61/353,531 | 2010-06-10 | ||
| PCT/US2011/039669 WO2011156518A2 (en) | 2010-06-10 | 2011-06-08 | Estrogen receptor modulators and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016149008A Division JP6465840B2 (ja) | 2010-06-10 | 2016-07-28 | エストロゲン受容体モジュレーターおよびその用途 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013528223A true JP2013528223A (ja) | 2013-07-08 |
| JP2013528223A5 JP2013528223A5 (enExample) | 2015-12-03 |
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Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
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| JP2013514346A Pending JP2013528223A (ja) | 2010-06-10 | 2011-06-08 | エストロゲン受容体モジュレーターおよびその用途 |
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| JP2017509631A (ja) * | 2014-03-13 | 2017-04-06 | エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト | エストロゲン受容体突然変異体を調節する方法及び組成物 |
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