HRP20120758T1 - Antiviralni nukleozidni analozi - Google Patents

Antiviralni nukleozidni analozi Download PDF

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Publication number
HRP20120758T1
HRP20120758T1 HRP20120758AT HRP20120758T HRP20120758T1 HR P20120758 T1 HRP20120758 T1 HR P20120758T1 HR P20120758A T HRP20120758A T HR P20120758AT HR P20120758 T HRP20120758 T HR P20120758T HR P20120758 T1 HRP20120758 T1 HR P20120758T1
Authority
HR
Croatia
Prior art keywords
substituted
hydroxymethyl
alkyl
compound according
methyltetrahydrofuran
Prior art date
Application number
HRP20120758AT
Other languages
English (en)
Croatian (hr)
Inventor
Yarlagadda S. Babu
Pooran Chand
V. Satish Kumar
Pravin L. Kotian
Minwan Wu
Original Assignee
Biocryst Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biocryst Pharmaceuticals, Inc. filed Critical Biocryst Pharmaceuticals, Inc.
Publication of HRP20120758T1 publication Critical patent/HRP20120758T1/hr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/23Heterocyclic radicals containing two or more heterocyclic rings condensed among themselves or condensed with a common carbocyclic ring system, not provided for in groups C07H19/14 - C07H19/22
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HRP20120758AT 2007-01-12 2008-01-11 Antiviralni nukleozidni analozi HRP20120758T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88027807P 2007-01-12 2007-01-12
PCT/US2008/050929 WO2008089105A2 (en) 2007-01-12 2008-01-11 Antiviral nucleoside analogs

Publications (1)

Publication Number Publication Date
HRP20120758T1 true HRP20120758T1 (hr) 2012-10-31

Family

ID=39471795

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20120758AT HRP20120758T1 (hr) 2007-01-12 2008-01-11 Antiviralni nukleozidni analozi

Country Status (19)

Country Link
US (1) US8440813B2 (enExample)
EP (2) EP2114980B1 (enExample)
JP (1) JP2010515760A (enExample)
CN (1) CN101611046A (enExample)
AU (1) AU2008206406A1 (enExample)
CA (1) CA2674589A1 (enExample)
CY (1) CY1113282T1 (enExample)
DK (1) DK2114980T3 (enExample)
ES (1) ES2390188T3 (enExample)
HR (1) HRP20120758T1 (enExample)
IL (1) IL199664A0 (enExample)
MX (1) MX2009007333A (enExample)
NZ (2) NZ598927A (enExample)
PH (1) PH12012502284A1 (enExample)
PL (1) PL2114980T3 (enExample)
PT (1) PT2114980E (enExample)
SG (1) SG177974A1 (enExample)
SI (1) SI2114980T1 (enExample)
WO (1) WO2008089105A2 (enExample)

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AU2010295373B2 (en) * 2009-09-21 2016-09-29 Gilead Sciences, Inc. 2' -fluoro substituted carba-nucleoside analogs for antiviral treatment
US7973013B2 (en) 2009-09-21 2011-07-05 Gilead Sciences, Inc. 2'-fluoro substituted carba-nucleoside analogs for antiviral treatment
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Also Published As

Publication number Publication date
CN101611046A (zh) 2009-12-23
ES2390188T3 (es) 2012-11-07
JP2010515760A (ja) 2010-05-13
WO2008089105A3 (en) 2008-09-12
IL199664A0 (en) 2010-04-15
US8440813B2 (en) 2013-05-14
PH12012502284A1 (en) 2015-10-12
DK2114980T3 (da) 2012-09-24
CA2674589A1 (en) 2008-07-24
AU2008206406A1 (en) 2008-07-24
SI2114980T1 (sl) 2012-11-30
EP2535345A1 (en) 2012-12-19
PL2114980T3 (pl) 2012-11-30
NZ578556A (en) 2012-04-27
MX2009007333A (es) 2009-08-31
HK1138286A1 (en) 2010-08-20
WO2008089105A2 (en) 2008-07-24
PT2114980E (pt) 2012-09-25
NZ598927A (en) 2013-09-27
US20100015094A1 (en) 2010-01-21
EP2114980B1 (en) 2012-06-27
EP2114980A2 (en) 2009-11-11
SG177974A1 (en) 2012-02-28
CY1113282T1 (el) 2016-04-13

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