HRP20110882T1 - Ciklopenta [d] pirimidini kao inhibitori kinaze akt proteina - Google Patents

Ciklopenta [d] pirimidini kao inhibitori kinaze akt proteina Download PDF

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Publication number
HRP20110882T1
HRP20110882T1 HR20110882T HRP20110882T HRP20110882T1 HR P20110882 T1 HRP20110882 T1 HR P20110882T1 HR 20110882 T HR20110882 T HR 20110882T HR P20110882 T HRP20110882 T HR P20110882T HR P20110882 T1 HRP20110882 T1 HR P20110882T1
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HR
Croatia
Prior art keywords
methyl
cyclopenta
piperazin
dihydro
alkyl
Prior art date
Application number
HR20110882T
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English (en)
Croatian (hr)
Inventor
S. Mitchell Ian
F. Blake James
Xu Rui
C. Kallan Nicholas
Xiao Dengming
Lee Spencer Keith
R. Bencsik Josef
Liang Jun
Safina Brian
Li Jun
Chabot Christine
L. Banka Anna
M. Wallace Eli
T. Schlachter Stephen
Original Assignee
Array Biopharma
Genentech
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38686844&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20110882(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Array Biopharma, Genentech filed Critical Array Biopharma
Publication of HRP20110882T1 publication Critical patent/HRP20110882T1/hr

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/4965—Non-condensed pyrazines
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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HR20110882T 2006-07-06 2007-07-05 Ciklopenta [d] pirimidini kao inhibitori kinaze akt proteina HRP20110882T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81876206P 2006-07-06 2006-07-06
PCT/US2007/072876 WO2008006032A1 (en) 2006-07-06 2007-07-05 Cyclopenta [d] pyrimidines as akt protein kinase inhibitors

Publications (1)

Publication Number Publication Date
HRP20110882T1 true HRP20110882T1 (hr) 2012-01-31

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HR20110882T HRP20110882T1 (hr) 2006-07-06 2007-07-05 Ciklopenta [d] pirimidini kao inhibitori kinaze akt proteina

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US (3) US8003651B2 (enExample)
EP (1) EP2049500B1 (enExample)
JP (3) JP5268904B2 (enExample)
KR (2) KR101527232B1 (enExample)
CN (2) CN103288753A (enExample)
AR (1) AR061844A1 (enExample)
AT (1) ATE523499T1 (enExample)
AU (1) AU2007269052B2 (enExample)
BR (1) BRPI0713555A2 (enExample)
CA (1) CA2656618C (enExample)
CL (1) CL2007001992A1 (enExample)
CO (1) CO6160229A2 (enExample)
CR (2) CR10601A (enExample)
CY (1) CY1112142T1 (enExample)
DK (1) DK2049500T3 (enExample)
ES (1) ES2372955T3 (enExample)
HR (1) HRP20110882T1 (enExample)
IL (1) IL196051A (enExample)
MA (1) MA30952B1 (enExample)
MX (1) MX2008016203A (enExample)
MY (1) MY147628A (enExample)
NO (1) NO20090580L (enExample)
NZ (1) NZ573979A (enExample)
PL (1) PL2049500T3 (enExample)
PT (1) PT2049500E (enExample)
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SI (1) SI2049500T1 (enExample)
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Families Citing this family (52)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008006025A1 (en) 2006-07-06 2008-01-10 Array Biopharma Inc. Dihydrofuro pyrimidines as akt protein kinase inhibitors
WO2008006039A1 (en) * 2006-07-06 2008-01-10 Array Biopharma Inc. Dihydrothieno pyrimidines as akt protein kinase inhibitors
US8063050B2 (en) * 2006-07-06 2011-11-22 Array Biopharma Inc. Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors
PL2049500T3 (pl) 2006-07-06 2012-02-29 Array Biopharma Inc Cyklopenta[d]pirymidyny jako inhibitory kinaz białkowych AKT
UA95641C2 (xx) * 2006-07-06 2011-08-25 Эррей Биофарма Инк. Гідроксильовані піримідильні циклопентани як інгібітори акт протеїнкінази$гидроксилированные пиримидильные циклопентаны как ингибиторы акт протеинкиназы
AU2014201211B2 (en) * 2006-07-06 2016-04-14 Array Biopharma Inc. Hydroxylated and methoxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors
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