HK1169998A1 - 胃抑勝肽受體活化的胰高血糖素化合物 - Google Patents
胃抑勝肽受體活化的胰高血糖素化合物Info
- Publication number
- HK1169998A1 HK1169998A1 HK12110717.7A HK12110717A HK1169998A1 HK 1169998 A1 HK1169998 A1 HK 1169998A1 HK 12110717 A HK12110717 A HK 12110717A HK 1169998 A1 HK1169998 A1 HK 1169998A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- gip receptor
- active glucagon
- glucagon compounds
- compounds
- active
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US18757809P | 2009-06-16 | 2009-06-16 | |
PCT/US2010/038825 WO2010148089A1 (en) | 2009-06-16 | 2010-06-16 | Gip receptor-active glucagon compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1169998A1 true HK1169998A1 (zh) | 2013-02-15 |
Family
ID=43356738
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK12110717.7A HK1169998A1 (zh) | 2009-06-16 | 2012-10-25 | 胃抑勝肽受體活化的胰高血糖素化合物 |
Country Status (18)
Country | Link |
---|---|
US (2) | US9150632B2 (zh) |
EP (1) | EP2443146B1 (zh) |
JP (1) | JP5887265B2 (zh) |
KR (1) | KR20120087875A (zh) |
CN (1) | CN102459325B (zh) |
AU (1) | AU2010260058B2 (zh) |
BR (1) | BRPI1014508A2 (zh) |
CA (1) | CA2765026A1 (zh) |
CL (1) | CL2011003173A1 (zh) |
HK (1) | HK1169998A1 (zh) |
IL (1) | IL216881A (zh) |
IN (1) | IN2012DN00377A (zh) |
MX (1) | MX2011013625A (zh) |
PE (1) | PE20120914A1 (zh) |
RU (1) | RU2012101274A (zh) |
SG (1) | SG176858A1 (zh) |
TW (1) | TWI549687B (zh) |
WO (1) | WO2010148089A1 (zh) |
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US8669228B2 (en) | 2007-01-05 | 2014-03-11 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting enhanced solubility in physiological pH buffers |
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CA2707861A1 (en) | 2007-10-30 | 2009-05-07 | Indiana University Research And Technology Corporation | Glucagon antagonists |
JP5771005B2 (ja) | 2007-10-30 | 2015-08-26 | インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションIndiana University Research And Technology Corporation | グルカゴンアンタゴニスト及びglp−1アゴニスト活性を示す化合物 |
PE20100255A1 (es) | 2008-06-17 | 2010-04-25 | Univ Indiana Res & Tech Corp | Co-agonistas del receptor de glucagon/glp-1 |
TWI474835B (zh) | 2008-06-17 | 2015-03-01 | Univ Indiana Res & Tech Corp | 用於治療代謝病症及肥胖症之基於gip之混合激動劑 |
CN102088989B (zh) | 2008-06-17 | 2014-11-26 | 印第安纳大学研究及科技有限公司 | 在生理pH缓冲液中具有增强的溶解性和稳定性的胰高血糖素类似物 |
JP2012512903A (ja) | 2008-12-19 | 2012-06-07 | インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーション | アミド系グルカゴンスーパーファミリーペプチドプロドラッグ |
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WO2011143208A1 (en) | 2010-05-13 | 2011-11-17 | Indiana University Research And Technology Corporation | Glucagon superfamily peptides exhibiting g protein-coupled receptor activity |
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-
2010
- 2010-06-16 AU AU2010260058A patent/AU2010260058B2/en not_active Ceased
- 2010-06-16 KR KR20127000871A patent/KR20120087875A/ko not_active Application Discontinuation
- 2010-06-16 RU RU2012101274/10A patent/RU2012101274A/ru not_active Application Discontinuation
- 2010-06-16 EP EP10790117.5A patent/EP2443146B1/en not_active Not-in-force
- 2010-06-16 WO PCT/US2010/038825 patent/WO2010148089A1/en active Application Filing
- 2010-06-16 BR BRPI1014508A patent/BRPI1014508A2/pt not_active IP Right Cessation
- 2010-06-16 US US13/378,001 patent/US9150632B2/en not_active Expired - Fee Related
- 2010-06-16 IN IN377DEN2012 patent/IN2012DN00377A/en unknown
- 2010-06-16 SG SG2011092772A patent/SG176858A1/en unknown
- 2010-06-16 MX MX2011013625A patent/MX2011013625A/es not_active Application Discontinuation
- 2010-06-16 CN CN201080027026.5A patent/CN102459325B/zh not_active Expired - Fee Related
- 2010-06-16 JP JP2012516264A patent/JP5887265B2/ja not_active Expired - Fee Related
- 2010-06-16 CA CA2765026A patent/CA2765026A1/en not_active Abandoned
- 2010-06-16 PE PE2011002102A patent/PE20120914A1/es not_active Application Discontinuation
- 2010-06-17 TW TW099119633A patent/TWI549687B/zh not_active IP Right Cessation
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- 2011-12-15 CL CL2011003173A patent/CL2011003173A1/es unknown
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CN102459325B (zh) | 2015-03-25 |
TWI549687B (zh) | 2016-09-21 |
US9790263B2 (en) | 2017-10-17 |
EP2443146B1 (en) | 2016-10-05 |
AU2010260058A1 (en) | 2012-02-02 |
AU2010260058B2 (en) | 2015-09-24 |
SG176858A1 (en) | 2012-02-28 |
TW201103556A (en) | 2011-02-01 |
BRPI1014508A2 (pt) | 2016-04-05 |
WO2010148089A1 (en) | 2010-12-23 |
CN102459325A (zh) | 2012-05-16 |
US9150632B2 (en) | 2015-10-06 |
MX2011013625A (es) | 2012-01-20 |
KR20120087875A (ko) | 2012-08-07 |
IL216881A0 (en) | 2012-02-29 |
US20160052989A1 (en) | 2016-02-25 |
CA2765026A1 (en) | 2010-12-23 |
JP5887265B2 (ja) | 2016-03-16 |
RU2012101274A (ru) | 2013-07-27 |
IN2012DN00377A (zh) | 2015-08-21 |
EP2443146A1 (en) | 2012-04-25 |
CL2011003173A1 (es) | 2012-05-25 |
PE20120914A1 (es) | 2012-08-22 |
US20120172295A1 (en) | 2012-07-05 |
JP2012530145A (ja) | 2012-11-29 |
EP2443146A4 (en) | 2012-11-21 |
IL216881A (en) | 2016-08-31 |
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