HK1141806A1 - Process for preparing 5-fluoro-1h-pyrazolo[3,4-b]pyridin-3-amine and derivatives thereof 5--1h-[34-b]-3- - Google Patents
Process for preparing 5-fluoro-1h-pyrazolo[3,4-b]pyridin-3-amine and derivatives thereof 5--1h-[34-b]-3-Info
- Publication number
- HK1141806A1 HK1141806A1 HK10108334.6A HK10108334A HK1141806A1 HK 1141806 A1 HK1141806 A1 HK 1141806A1 HK 10108334 A HK10108334 A HK 10108334A HK 1141806 A1 HK1141806 A1 HK 1141806A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- pyrazolo
- pyridin
- fluoro
- amine
- derivatives
- Prior art date
Links
- UFONWAPOQPJJLL-UHFFFAOYSA-N 5-fluoro-2h-pyrazolo[3,4-b]pyridin-3-amine Chemical compound C1=C(F)C=C2C(N)=NNC2=N1 UFONWAPOQPJJLL-UHFFFAOYSA-N 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Transplantation (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US95301907P | 2007-07-31 | 2007-07-31 | |
PCT/US2008/071714 WO2009018415A1 (en) | 2007-07-31 | 2008-07-31 | Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1141806A1 true HK1141806A1 (en) | 2010-11-19 |
Family
ID=39884162
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK10108334.6A HK1141806A1 (en) | 2007-07-31 | 2010-09-02 | Process for preparing 5-fluoro-1h-pyrazolo[3,4-b]pyridin-3-amine and derivatives thereof 5--1h-[34-b]-3- |
Country Status (13)
Country | Link |
---|---|
US (2) | US8242272B2 (de) |
EP (1) | EP2176261B1 (de) |
JP (2) | JP5553751B2 (de) |
CN (1) | CN101790532B (de) |
AR (1) | AR067762A1 (de) |
AU (1) | AU2008282156B2 (de) |
CA (1) | CA2694499A1 (de) |
ES (1) | ES2400104T3 (de) |
HK (1) | HK1141806A1 (de) |
MX (1) | MX2010001137A (de) |
NZ (1) | NZ582879A (de) |
TW (1) | TW200916468A (de) |
WO (1) | WO2009018415A1 (de) |
Families Citing this family (44)
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DE102010040233A1 (de) | 2010-09-03 | 2012-03-08 | Bayer Schering Pharma Aktiengesellschaft | Bicyclische Aza-Heterocyclen und ihre Verwendung |
DE102010040234A1 (de) | 2010-09-03 | 2012-03-08 | Bayer Schering Pharma Aktiengesellschaft | Verfahren zur Herstellung von 5-Flour-1H-pyrazolo[3,4-b]pyridin-3-carbonitril |
DE102010043380A1 (de) | 2010-11-04 | 2012-05-10 | Bayer Schering Pharma Aktiengesellschaft | Benzyl-substituierte Carbamate und ihre Verwendung |
DE102010043379A1 (de) | 2010-11-04 | 2012-05-10 | Bayer Schering Pharma Aktiengesellschaft | Substituierte 6-Fluor-1H-Pyrazolo[4,3-b]pyridine und ihre Verwendung |
DE102011007890A1 (de) | 2011-04-21 | 2012-10-25 | Bayer Pharma Aktiengesellschaft | Fluoralkyl-substituierte Pyrazolopyridine und ihre Verwendung |
DE102012200357A1 (de) | 2012-01-11 | 2013-07-11 | Bayer Intellectual Property Gmbh | Fluoralkyl-substituierte Pyrazolopyridine und ihre Verwendung |
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DE102012200360A1 (de) | 2012-01-11 | 2013-07-11 | Bayer Intellectual Property Gmbh | Substituierte Triazine und ihre Verwendung |
DE102012200349A1 (de) | 2012-01-11 | 2013-07-11 | Bayer Intellectual Property Gmbh | Substituierte annellierte Pyrimidine und Triazine und ihre Verwendung |
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EP3068776B1 (de) | 2013-11-13 | 2019-05-29 | Vertex Pharmaceuticals Incorporated | Hemmer der influenzavirenreplikation |
JP6704416B2 (ja) | 2015-05-13 | 2020-06-03 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | インフルエンザウイルスの複製の阻害剤を調製する方法 |
JP6857617B2 (ja) | 2015-05-13 | 2021-04-14 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | インフルエンザウイルスの複製の阻害剤 |
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-
2008
- 2008-07-31 EP EP08796922A patent/EP2176261B1/de not_active Not-in-force
- 2008-07-31 AR ARP080103330A patent/AR067762A1/es unknown
- 2008-07-31 NZ NZ582879A patent/NZ582879A/en not_active IP Right Cessation
- 2008-07-31 WO PCT/US2008/071714 patent/WO2009018415A1/en active Application Filing
- 2008-07-31 AU AU2008282156A patent/AU2008282156B2/en not_active Ceased
- 2008-07-31 CN CN2008801048142A patent/CN101790532B/zh not_active Expired - Fee Related
- 2008-07-31 TW TW097129121A patent/TW200916468A/zh unknown
- 2008-07-31 ES ES08796922T patent/ES2400104T3/es active Active
- 2008-07-31 MX MX2010001137A patent/MX2010001137A/es not_active Application Discontinuation
- 2008-07-31 CA CA2694499A patent/CA2694499A1/en not_active Abandoned
- 2008-07-31 JP JP2010520181A patent/JP5553751B2/ja not_active Expired - Fee Related
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2010
- 2010-01-28 US US12/695,292 patent/US8242272B2/en not_active Expired - Fee Related
- 2010-09-02 HK HK10108334.6A patent/HK1141806A1/xx not_active IP Right Cessation
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2012
- 2012-01-11 US US13/347,926 patent/US8598361B2/en not_active Expired - Fee Related
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Also Published As
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---|---|
CA2694499A1 (en) | 2009-02-05 |
JP5553751B2 (ja) | 2014-07-16 |
TW200916468A (en) | 2009-04-16 |
AR067762A1 (es) | 2009-10-21 |
US20120232275A1 (en) | 2012-09-13 |
CN101790532B (zh) | 2013-11-20 |
US20100184980A1 (en) | 2010-07-22 |
JP2010535241A (ja) | 2010-11-18 |
EP2176261A1 (de) | 2010-04-21 |
AU2008282156B2 (en) | 2014-07-17 |
JP2014055160A (ja) | 2014-03-27 |
US8598361B2 (en) | 2013-12-03 |
CN101790532A (zh) | 2010-07-28 |
EP2176261B1 (de) | 2012-12-19 |
MX2010001137A (es) | 2010-03-31 |
AU2008282156A1 (en) | 2009-02-05 |
NZ582879A (en) | 2012-03-30 |
ES2400104T3 (es) | 2013-04-05 |
WO2009018415A1 (en) | 2009-02-05 |
US8242272B2 (en) | 2012-08-14 |
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