HK1141806A1 - Process for preparing 5-fluoro-1h-pyrazolo[3,4-b]pyridin-3-amine and derivatives thereof 5--1h-[34-b]-3- - Google Patents

Process for preparing 5-fluoro-1h-pyrazolo[3,4-b]pyridin-3-amine and derivatives thereof 5--1h-[34-b]-3-

Info

Publication number
HK1141806A1
HK1141806A1 HK10108334.6A HK10108334A HK1141806A1 HK 1141806 A1 HK1141806 A1 HK 1141806A1 HK 10108334 A HK10108334 A HK 10108334A HK 1141806 A1 HK1141806 A1 HK 1141806A1
Authority
HK
Hong Kong
Prior art keywords
pyrazolo
pyridin
fluoro
amine
derivatives
Prior art date
Application number
HK10108334.6A
Other languages
English (en)
Chinese (zh)
Inventor
‧吉米內斯
‧克裡爾
‧米勒
‧格林
高淮
‧哈蒙
‧德洛斯
Original Assignee
沃泰克斯藥物股份有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 沃泰克斯藥物股份有限公司 filed Critical 沃泰克斯藥物股份有限公司
Publication of HK1141806A1 publication Critical patent/HK1141806A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Transplantation (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK10108334.6A 2007-07-31 2010-09-02 Process for preparing 5-fluoro-1h-pyrazolo[3,4-b]pyridin-3-amine and derivatives thereof 5--1h-[34-b]-3- HK1141806A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US95301907P 2007-07-31 2007-07-31
PCT/US2008/071714 WO2009018415A1 (en) 2007-07-31 2008-07-31 Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof

Publications (1)

Publication Number Publication Date
HK1141806A1 true HK1141806A1 (en) 2010-11-19

Family

ID=39884162

Family Applications (1)

Application Number Title Priority Date Filing Date
HK10108334.6A HK1141806A1 (en) 2007-07-31 2010-09-02 Process for preparing 5-fluoro-1h-pyrazolo[3,4-b]pyridin-3-amine and derivatives thereof 5--1h-[34-b]-3-

Country Status (13)

Country Link
US (2) US8242272B2 (de)
EP (1) EP2176261B1 (de)
JP (2) JP5553751B2 (de)
CN (1) CN101790532B (de)
AR (1) AR067762A1 (de)
AU (1) AU2008282156B2 (de)
CA (1) CA2694499A1 (de)
ES (1) ES2400104T3 (de)
HK (1) HK1141806A1 (de)
MX (1) MX2010001137A (de)
NZ (1) NZ582879A (de)
TW (1) TW200916468A (de)
WO (1) WO2009018415A1 (de)

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PT3068782T (pt) 2013-11-13 2018-10-08 Vertex Pharma Métodos de preparação de inibidores da replicação de vírus da gripe
EP3068776B1 (de) 2013-11-13 2019-05-29 Vertex Pharmaceuticals Incorporated Hemmer der influenzavirenreplikation
JP6704416B2 (ja) 2015-05-13 2020-06-03 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ インフルエンザウイルスの複製の阻害剤を調製する方法
JP6857617B2 (ja) 2015-05-13 2021-04-14 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ インフルエンザウイルスの複製の阻害剤
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AR067762A1 (es) 2009-10-21
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CN101790532B (zh) 2013-11-20
US20100184980A1 (en) 2010-07-22
JP2010535241A (ja) 2010-11-18
EP2176261A1 (de) 2010-04-21
AU2008282156B2 (en) 2014-07-17
JP2014055160A (ja) 2014-03-27
US8598361B2 (en) 2013-12-03
CN101790532A (zh) 2010-07-28
EP2176261B1 (de) 2012-12-19
MX2010001137A (es) 2010-03-31
AU2008282156A1 (en) 2009-02-05
NZ582879A (en) 2012-03-30
ES2400104T3 (es) 2013-04-05
WO2009018415A1 (en) 2009-02-05
US8242272B2 (en) 2012-08-14

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