HK1016187A1 - Novel 5-o-deoaminyl 6-o-methyl erythronolide a derivatives, method for preraring the same - Google Patents

Novel 5-o-deoaminyl 6-o-methyl erythronolide a derivatives, method for preraring the same

Info

Publication number
HK1016187A1
HK1016187A1 HK99101038A HK99101038A HK1016187A1 HK 1016187 A1 HK1016187 A1 HK 1016187A1 HK 99101038 A HK99101038 A HK 99101038A HK 99101038 A HK99101038 A HK 99101038A HK 1016187 A1 HK1016187 A1 HK 1016187A1
Authority
HK
Hong Kong
Prior art keywords
preraring
deoaminyl
derivatives
novel
same
Prior art date
Application number
HK99101038A
Other languages
English (en)
Inventor
Alain Bonnet
Michael Delthil
Alain Mazurie
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9482423&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1016187(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of HK1016187A1 publication Critical patent/HK1016187A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HK99101038A 1995-09-11 1999-03-12 Novel 5-o-deoaminyl 6-o-methyl erythronolide a derivatives, method for preraring the same HK1016187A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9510601A FR2738571B1 (fr) 1995-09-11 1995-09-11 Nouveaux derives de la 5-0-desosaminyl 6-0-methyl- erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
PCT/FR1996/001384 WO1997010251A1 (fr) 1995-09-11 1996-09-10 Nouveaux derives de la 5-0-desosaminyl 6-0-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number Publication Date
HK1016187A1 true HK1016187A1 (en) 1999-10-29

Family

ID=9482423

Family Applications (2)

Application Number Title Priority Date Filing Date
HK99101038A HK1016187A1 (en) 1995-09-11 1999-03-12 Novel 5-o-deoaminyl 6-o-methyl erythronolide a derivatives, method for preraring the same
HK02103101.8A HK1041489B (zh) 1995-09-11 2002-04-19 5-0-德糖胺基-6-0-甲基-紅諾霉素a衍生物在製備生物活性產品方法的應用

Family Applications After (1)

Application Number Title Priority Date Filing Date
HK02103101.8A HK1041489B (zh) 1995-09-11 2002-04-19 5-0-德糖胺基-6-0-甲基-紅諾霉素a衍生物在製備生物活性產品方法的應用

Country Status (34)

Country Link
US (1) US5969161A (zh)
EP (1) EP0854880B1 (zh)
JP (1) JP4332218B2 (zh)
KR (1) KR100457755B1 (zh)
CN (2) CN1070498C (zh)
AP (1) AP887A (zh)
AR (1) AR004195A1 (zh)
AT (1) ATE266035T1 (zh)
AU (1) AU708811B2 (zh)
BG (1) BG63822B1 (zh)
BR (1) BR9610503A (zh)
CA (1) CA2228670C (zh)
CZ (3) CZ294865B6 (zh)
DE (1) DE69632405T2 (zh)
DK (1) DK0854880T3 (zh)
EA (1) EA000575B1 (zh)
EE (1) EE03774B1 (zh)
ES (1) ES2219698T3 (zh)
FR (1) FR2738571B1 (zh)
GE (1) GEP20022838B (zh)
HK (2) HK1016187A1 (zh)
HU (1) HU227565B1 (zh)
IL (1) IL123550A (zh)
MX (1) MX9801859A (zh)
NO (2) NO312678B1 (zh)
PL (1) PL183652B1 (zh)
PT (1) PT854880E (zh)
RO (1) RO120137B1 (zh)
SI (1) SI0854880T1 (zh)
SK (3) SK285853B6 (zh)
TR (1) TR199800438T1 (zh)
UA (1) UA53628C2 (zh)
WO (1) WO1997010251A1 (zh)
ZA (1) ZA966837B (zh)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL128681A0 (en) * 1996-09-04 2000-01-31 Abbott Lab 6-O substituted ketolides having antibacterial activity
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
US6034069A (en) * 1997-09-30 2000-03-07 Abbott Laboratories 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity
US6046171A (en) * 1997-10-29 2000-04-04 Abbott Laboratories 6,11-bridged erythromycin derivatives
US6124269A (en) * 1997-10-29 2000-09-26 Abbott Laboratories 2-Halo-6-O-substituted ketolide derivatives
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
US6420535B1 (en) 1999-06-07 2002-07-16 Abbott Laboratories 6-O-carbamate ketolide derivatives
CA2476423A1 (en) * 2002-02-15 2003-08-28 Sympore Gmbh Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
US6841664B2 (en) * 2002-07-25 2005-01-11 Enanra Pharmaceuticals, Inc. 6,11-4-carbon bridged ketolides
US6764998B1 (en) 2003-06-18 2004-07-20 Enanta Pharmaceuticals, Inc. 6,11-4C-bicyclic 9a-azalide derivatives
US6753318B1 (en) * 2002-07-25 2004-06-22 Enanta Pharmaceuticals, Inc. 6,11-4-carbon bridged erythromycin derivatives
KR100661973B1 (ko) * 2002-05-13 2006-12-28 이난타 파마슈티칼스, 인코포레이티드 6,11 바이사이클릭 에리스로마이신 유도체
WO2005070918A1 (en) * 2002-05-13 2005-08-04 Enanta Pharmaceuticals, Inc. Process for the preparation of t-11 bicyclic erythromycin derivatives
US6878691B2 (en) * 2002-05-13 2005-04-12 Enanta Pharmaceuticals, Inc. 6-11 bicyclic ketolide derivatives
US7273853B2 (en) * 2002-05-13 2007-09-25 Enanta Pharmaceuticals, Inc. 6-11 bicyclic ketolide derivatives
US7135573B2 (en) * 2002-05-13 2006-11-14 Enanta Pharmaceuticals, Inc. Processes for the preparation of O-(6-Pyrazol-1-yl-pyridin-3-ylmethyl)-hydroxylamine
US7910558B2 (en) * 2002-05-13 2011-03-22 Enanta Pharmaceuticals, Inc. Bridged macrocyclic compounds and processes for the preparation thereof
US7064110B2 (en) * 2002-05-13 2006-06-20 Enanta Pharmaceuticals, Inc. 6-11 bicycle ketolide derivatives
ITMI20021726A1 (it) * 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
US6645941B1 (en) 2003-03-26 2003-11-11 Enanta Pharmaceuticals, Inc. 6,11-3C-bicyclic 9a-azalide derivatives
US7276487B2 (en) * 2003-09-23 2007-10-02 Enanta Pharmaceuticals, Inc. 9a, 11-3C-bicyclic 9a-azalide derivatives
US7414030B2 (en) * 2004-01-07 2008-08-19 Enanta Pharmaceuticals, Inc. 6-11 Bicyclic erythromycin derivatives
US7265094B2 (en) * 2004-01-09 2007-09-04 Enanta Pharmaceuticals, Inc. 9N-substituted 6-11 bicyclic erythromycin derivatives
JP2008522978A (ja) 2004-12-07 2008-07-03 エナンタ ファーマシューティカルズ インコーポレイテッド ３，６−ビシクロライド
US7229972B2 (en) 2004-12-07 2007-06-12 Enanta Pharmaceuticals, Inc. 3,6-Bicyclolides
WO2006065721A2 (en) 2004-12-13 2006-06-22 Enanta Pharmaceuticals, Inc. 11, 12-lactone bicyclolides
TW200635600A (en) 2004-12-13 2006-10-16 Enanta Pharm Inc Tetracyclic bicyclolides
US7384922B2 (en) * 2005-05-04 2008-06-10 Enanta Pharmaceuticals, Inc. 6-11 bridged oxime erythromycin derivatives
WO2007012464A1 (en) * 2005-07-26 2007-02-01 Merckle Gmbh Macrolide conjugates of pyrrolizine and indolizine compounds as inhibitors of 5-lipooxygenase and cyclooxygenase
US8273720B2 (en) * 2007-09-17 2012-09-25 Enanta Pharmaceuticals, Inc. 6,11-bicyclolides: bridged biaryl macrolide derivatives
US8354383B2 (en) * 2007-09-17 2013-01-15 Enanta Pharmaceuticals, Inc. 6,11-bridged biaryl macrolides
EP2203435B1 (en) * 2007-09-17 2018-07-18 Enanta Pharmaceuticals, Inc. 6, 11-bridged biaryl macrolides
CN103232501A (zh) * 2013-04-11 2013-08-07 宜昌东阳光药业股份有限公司 阿奇霉素或阿奇霉素的中间体脱去克拉定糖化合物的制备工艺

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR960000434B1 (ko) * 1986-12-17 1996-01-06 다이쇼 세이야꾸 가부시끼가이샤 에리스로마이신 a유도체 및 그의 제조 방법
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives

Also Published As

Publication number Publication date
SI0854880T1 (en) 2004-12-31
BR9610503A (pt) 1999-07-06
CZ71798A3 (cs) 1998-07-15
ATE266035T1 (de) 2004-05-15
UA53628C2 (uk) 2003-02-17
JPH11512416A (ja) 1999-10-26
NO981053L (no) 1998-03-10
AP887A (en) 2000-11-10
CN1319602A (zh) 2001-10-31
NO981053D0 (no) 1998-03-10
CN1201462A (zh) 1998-12-09
AU708811B2 (en) 1999-08-12
SK283690B6 (sk) 2003-12-02
US5969161A (en) 1999-10-19
EA000575B1 (ru) 1999-12-29
NO20021111D0 (no) 2002-03-06
AU6991096A (en) 1997-04-01
FR2738571A1 (fr) 1997-03-14
CA2228670C (fr) 2005-04-12
HK1041489A1 (en) 2002-07-12
FR2738571B1 (fr) 1997-10-17
CZ294866B6 (cs) 2005-04-13
NO312678B1 (no) 2002-06-17
EE03774B1 (et) 2002-06-17
BG102312A (en) 1998-09-30
SK285853B6 (sk) 2007-09-06
KR100457755B1 (ko) 2005-02-28
NO315048B1 (no) 2003-06-30
EE9800065A (et) 1998-08-17
BG63822B1 (bg) 2003-02-28
PL326274A1 (en) 1998-08-31
SK29498A3 (en) 1998-12-02
ES2219698T3 (es) 2004-12-01
NO20021111L (no) 1998-03-10
CN1237069C (zh) 2006-01-18
RO120137B1 (ro) 2005-09-30
PL183652B1 (pl) 2002-06-28
DE69632405D1 (de) 2004-06-09
DK0854880T3 (da) 2004-08-16
EA199800288A1 (ru) 1998-08-27
ZA966837B (en) 1997-08-13
KR19990044543A (ko) 1999-06-25
HUP9802930A1 (hu) 1999-04-28
IL123550A (en) 2002-09-12
TR199800438T1 (xx) 1998-05-21
EP0854880B1 (fr) 2004-05-06
PT854880E (pt) 2004-09-30
EP0854880A1 (fr) 1998-07-29
SK285995B6 (sk) 2008-01-07
JP4332218B2 (ja) 2009-09-16
MX9801859A (es) 1998-11-30
CN1070498C (zh) 2001-09-05
CZ289945B6 (cs) 2002-04-17
GEP20022838B (en) 2002-11-25
DE69632405T2 (de) 2005-05-19
CZ294865B6 (cs) 2005-04-13
AR004195A1 (es) 1998-11-04
WO1997010251A1 (fr) 1997-03-20
HU227565B1 (en) 2011-08-29
HUP9802930A3 (en) 1999-12-28
CA2228670A1 (fr) 1997-03-20
HK1041489B (zh) 2006-09-08
AP9801210A0 (en) 1998-03-31
IL123550A0 (en) 1998-10-30

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Legal Events

Date Code Title Description
PF Patent in force
AS Change of ownership

Owner name: AVENTIS PHARMA S.A.

Free format text: FORMER OWNER(S): HOECHST MARION ROUSSEL

Owner name: HOECHST MARION ROUSSEL

Free format text: FORMER OWNER(S): ROUSSEL UCLAF

CHPA Change of a particular in the register (except of change of ownership)
PE Patent expired

Effective date: 20160909