FI69301C - Foerfarande foer framstaellning av terapeutiskt verksamma substituerade 2-fenyl-imino-imidazolidiner - Google Patents
Foerfarande foer framstaellning av terapeutiskt verksamma substituerade 2-fenyl-imino-imidazolidiner Download PDFInfo
- Publication number
- FI69301C FI69301C FI790510A FI790510A FI69301C FI 69301 C FI69301 C FI 69301C FI 790510 A FI790510 A FI 790510A FI 790510 A FI790510 A FI 790510A FI 69301 C FI69301 C FI 69301C
- Authority
- FI
- Finland
- Prior art keywords
- acid
- formula
- preparation
- acid addition
- therapeutic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19782806775 DE2806775A1 (de) | 1978-02-17 | 1978-02-17 | Neue substituierte 2-phenylimino- imidazolidine deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zur herstellung derselben |
DE2806775 | 1978-02-17 |
Publications (3)
Publication Number | Publication Date |
---|---|
FI790510A FI790510A (fi) | 1979-08-18 |
FI69301B FI69301B (fi) | 1985-09-30 |
FI69301C true FI69301C (fi) | 1986-01-10 |
Family
ID=6032231
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI790510A FI69301C (fi) | 1978-02-17 | 1979-02-15 | Foerfarande foer framstaellning av terapeutiskt verksamma substituerade 2-fenyl-imino-imidazolidiner |
Country Status (32)
Country | Link |
---|---|
US (2) | US4250186A (fr) |
JP (1) | JPS54122273A (fr) |
AT (1) | AT370093B (fr) |
AU (1) | AU519356B2 (fr) |
BE (1) | BE874252A (fr) |
CA (1) | CA1115717A (fr) |
CH (1) | CH640230A5 (fr) |
CS (2) | CS207773B2 (fr) |
DD (1) | DD142048A5 (fr) |
DE (1) | DE2806775A1 (fr) |
DK (1) | DK69479A (fr) |
ES (2) | ES477784A1 (fr) |
FI (1) | FI69301C (fr) |
FR (1) | FR2417502A1 (fr) |
GB (1) | GB2014575B (fr) |
GR (2) | GR67626B (fr) |
HU (1) | HU180430B (fr) |
IE (1) | IE48073B1 (fr) |
IL (1) | IL56678A (fr) |
IT (1) | IT1113469B (fr) |
LU (1) | LU80924A1 (fr) |
NL (1) | NL7901241A (fr) |
NO (1) | NO151239C (fr) |
NZ (1) | NZ189684A (fr) |
PH (1) | PH16188A (fr) |
PL (2) | PL116527B1 (fr) |
PT (1) | PT69239A (fr) |
RO (2) | RO81504B (fr) |
SE (1) | SE7901405L (fr) |
SU (2) | SU812175A3 (fr) |
YU (1) | YU36779A (fr) |
ZA (1) | ZA79709B (fr) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2854659A1 (de) * | 1978-12-18 | 1980-07-10 | Boehringer Sohn Ingelheim | Neue 3,4-disubstituierte 2-phenylimino-imidazolidine, deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung |
DE3168754D1 (en) * | 1980-07-09 | 1985-03-21 | Beecham Group Plc | Clonidine derivatives useful in the treatment of diarrhoea |
EP0070084A3 (fr) * | 1981-04-24 | 1983-02-16 | Beecham Group Plc | Dérivés d'imidazoline |
US4517199A (en) * | 1981-11-20 | 1985-05-14 | Alcon Laboratories, Inc. | Method for lowering intraocular pressure using phenylimino-imidazoles |
CA1201066A (fr) * | 1981-11-20 | 1986-02-25 | Alcon Laboratories, Inc. | Solutions de n-¬3,5-dichloro-4-(2- imidazolidinylidene-amino)-phenyl|-acetamide pour diminuer la pression intra-oculaire |
US4515800A (en) * | 1981-11-20 | 1985-05-07 | Icilio Cavero | Method of lowering intraocular pressure using phenylimino-imidazoles |
US4644007A (en) * | 1981-11-20 | 1987-02-17 | Alcon Laboratories, Inc. | 3-chloro-4-(4,5-dihydro-1H-imidazo-2-yl)-amino-5-alkylbenzoic acids, esters, salts, compositions and methods |
US4461904A (en) * | 1981-11-20 | 1984-07-24 | Alcon Laboratories, Inc. | 2-(Trisubstituted phenylimino)-imidazolines |
FR2521140A1 (fr) * | 1982-02-05 | 1983-08-12 | Synthelabo | Derives d'imidazolidine, leur preparation et leur application en therapeutique |
GB2137191A (en) * | 1983-02-28 | 1984-10-03 | Sumitomo Chemical Co | Fungicidal N-phenylimidates |
DE19514579A1 (de) * | 1995-04-20 | 1996-10-24 | Boehringer Ingelheim Kg | Verwendung von alpha¶1¶¶L¶-Agonisten zur Behandlung der Harninkontinenz |
JP2003166617A (ja) | 2001-11-28 | 2003-06-13 | Honda Motor Co Ltd | トルクコンバータ付き内燃機関 |
JP2007308392A (ja) * | 2006-05-16 | 2007-11-29 | Bayer Cropscience Ag | 殺虫性ベンズアミジン類 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2938038A (en) * | 1960-05-24 | X-dihydroxyphenylamino | ||
US2899426A (en) * | 1959-08-11 | Synthesis of l | ||
FR1211341A (fr) * | 1955-12-19 | 1960-03-15 | A Wander Dr | Procédé pour la préparation de 2-amino-imidazolines |
US3595961A (en) * | 1965-10-01 | 1971-07-27 | Boehringer Sohn Ingelheim | Hypotensive compositions containing 2-(2' - halo-anilino) - 1,3 -diazacyclopentenes-(2) and methods of using the same |
DE1670274A1 (de) * | 1966-10-31 | 1970-07-16 | Boehringer Sohn Ingelheim | Neues Verfahren zur Herstellung von 2-Arylamino-1,3-diazacycloalkenen-(2) |
AT285599B (de) * | 1968-06-21 | 1970-11-10 | Boehringer Sohn Ingelheim | Verfahren zur Herstellung von neuen trisubstituierten 2-Arylaminoimidazolinen und ihren Salzen |
DE2446758C3 (de) * | 1974-10-01 | 1979-01-04 | C.H. Boehringer Sohn, 6507 Ingelheim | 2-(2-Fluor-6-trifluormethylphenylimino)-imidazolidin, dessen Säureadditionssalze, Verfahren zur Herstellung dieser Verbindungen und deren Verwendung bei der Bekämpfung der Hypertonie |
DE2523103C3 (de) * | 1975-05-24 | 1979-11-29 | C.H. Boehringer Sohn, 6507 Ingelheim | Substituierte 2-[N-Progargyl-N-(2-chlorphenyl)amino] -imidazoline-^), deren Säureadditionssalze, Verfahren zu ihrer Herstellung und deren Verwendung |
DE2630060C2 (de) * | 1976-07-03 | 1984-04-19 | C.H. Boehringer Sohn, 6507 Ingelheim | 2-(2-Brom-6-fluor-phenylimino)-imidazolidin, dessen Säureadditionssalze, diese enthaltende Arzneimittel und Verfahren zu deren Herstellung |
-
1978
- 1978-02-17 DE DE19782806775 patent/DE2806775A1/de not_active Withdrawn
-
1979
- 1979-02-09 SU SU792721602A patent/SU812175A3/ru active
- 1979-02-12 GR GR58340A patent/GR67626B/el unknown
- 1979-02-12 AT AT0101579A patent/AT370093B/de not_active IP Right Cessation
- 1979-02-13 RO RO103172A patent/RO81504B/ro unknown
- 1979-02-14 CH CH142879A patent/CH640230A5/de not_active IP Right Cessation
- 1979-02-15 FI FI790510A patent/FI69301C/fi not_active IP Right Cessation
- 1979-02-15 IL IL56678A patent/IL56678A/xx unknown
- 1979-02-15 YU YU00367/79A patent/YU36779A/xx unknown
- 1979-02-15 HU HU79BO1764A patent/HU180430B/hu unknown
- 1979-02-15 LU LU80924A patent/LU80924A1/de unknown
- 1979-02-15 PT PT7969239A patent/PT69239A/pt unknown
- 1979-02-15 IT IT48010/79A patent/IT1113469B/it active
- 1979-02-15 DD DD79211044A patent/DD142048A5/de unknown
- 1979-02-16 DK DK69479A patent/DK69479A/da not_active Application Discontinuation
- 1979-02-16 PL PL1979221508A patent/PL116527B1/pl unknown
- 1979-02-16 NZ NZ189684A patent/NZ189684A/xx unknown
- 1979-02-16 US US06/012,650 patent/US4250186A/en not_active Expired - Lifetime
- 1979-02-16 AU AU44325/79A patent/AU519356B2/en not_active Ceased
- 1979-02-16 FR FR7904052A patent/FR2417502A1/fr active Granted
- 1979-02-16 NL NL7901241A patent/NL7901241A/xx not_active Application Discontinuation
- 1979-02-16 IE IE311/79A patent/IE48073B1/en unknown
- 1979-02-16 ES ES477784A patent/ES477784A1/es not_active Expired
- 1979-02-16 NO NO790523A patent/NO151239C/no unknown
- 1979-02-16 BE BE0/193531A patent/BE874252A/fr not_active IP Right Cessation
- 1979-02-16 ZA ZA79709A patent/ZA79709B/xx unknown
- 1979-02-16 PL PL1979213475A patent/PL115759B1/pl unknown
- 1979-02-16 CA CA321,805A patent/CA1115717A/fr not_active Expired
- 1979-02-16 GB GB7905506A patent/GB2014575B/en not_active Expired
- 1979-02-16 JP JP1715679A patent/JPS54122273A/ja active Pending
- 1979-02-16 SE SE7901405A patent/SE7901405L/xx not_active Application Discontinuation
- 1979-02-17 RO RO7996602A patent/RO76799A/fr unknown
- 1979-02-19 CS CS791092A patent/CS207773B2/cs unknown
- 1979-02-19 CS CS798500A patent/CS207774B2/cs unknown
- 1979-06-18 GR GR59371A patent/GR69232B/el unknown
- 1979-10-16 ES ES485043A patent/ES485043A1/es not_active Expired
-
1980
- 1980-01-30 SU SU802874805A patent/SU828964A3/ru active
- 1980-08-20 US US06/179,839 patent/US4293564A/en not_active Expired - Lifetime
- 1980-09-08 PH PH24546A patent/PH16188A/en unknown
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM | Patent lapsed |
Owner name: C.H. BOEHRINGER SOHN |