FI109453B - Farmaseuttinen koostumus - Google Patents

Farmaseuttinen koostumus Download PDF

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Publication number
FI109453B
FI109453B FI991485A FI991485A FI109453B FI 109453 B FI109453 B FI 109453B FI 991485 A FI991485 A FI 991485A FI 991485 A FI991485 A FI 991485A FI 109453 B FI109453 B FI 109453B
Authority
FI
Finland
Prior art keywords
pharmaceutically acceptable
carbidopa
entacapone
levodopa
mixture
Prior art date
Application number
FI991485A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI991485A0 (fi
FI991485L (fi
Inventor
Kari Vahervuo
Sari Kallioinen
Lasse Kervinen
Marja Laaksonen
Jarmo Lintulaakso
Mervi Niskanen
Marja Partanen
Marja Ritala
Matti Virkki
Original Assignee
Orion Yhtymae Oyj
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8554988&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI109453(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Orion Yhtymae Oyj filed Critical Orion Yhtymae Oyj
Priority to FI991485A priority Critical patent/FI109453B/fi
Publication of FI991485A0 publication Critical patent/FI991485A0/fi
Priority to TW089110218A priority patent/TWI241187B/zh
Priority to PE2000000641A priority patent/PE20010399A1/es
Priority to IT2000MI001450A priority patent/ITMI20001450A1/it
Priority to EEP200100716A priority patent/EE05473B1/xx
Priority to AU58306/00A priority patent/AU765932B2/en
Priority to ES00944070T priority patent/ES2203495T3/es
Priority to CZ20014636A priority patent/CZ303010B6/cs
Priority to PL352775A priority patent/PL197818B1/pl
Priority to TR2001/03763T priority patent/TR200103763T2/xx
Priority to YUP-925/01A priority patent/RS50368B/sr
Priority to ARP000103325A priority patent/AR033796A1/es
Priority to CA002378469A priority patent/CA2378469C/en
Priority to CZ2011-885A priority patent/CZ304416B6/cs
Priority to CO00048944A priority patent/CO5180579A1/es
Priority to MEP-2008-863A priority patent/ME00520B/me
Priority to EP00944070A priority patent/EP1189608B1/en
Priority to KR1020017015737A priority patent/KR100905428B1/ko
Priority to HR20020088A priority patent/HRP20020088B1/xx
Priority to PCT/FI2000/000593 priority patent/WO2001001984A1/en
Priority to HU0202273A priority patent/HU230395B1/hu
Priority to UA2002010771A priority patent/UA75047C2/uk
Priority to BRPI0011867A priority patent/BRPI0011867B8/pt
Priority to SK1923-2001A priority patent/SK286451B6/sk
Priority to JP2001507476A priority patent/JP4204783B2/ja
Priority to CNB008095868A priority patent/CN1168440C/zh
Priority to NZ515780A priority patent/NZ515780A/en
Priority to SI200030190T priority patent/SI1189608T1/xx
Priority to MYPI20002972A priority patent/MY127685A/en
Priority to US09/605,529 priority patent/US6500867B1/en
Priority to BR0011867-2A priority patent/BR0011867A/pt
Priority to DK00944070T priority patent/DK1189608T3/da
Priority to MXPA01013167A priority patent/MXPA01013167A/es
Priority to EA200200106A priority patent/EA004503B1/ru
Priority to DE60004052T priority patent/DE60004052T2/de
Priority to HK02108609.4A priority patent/HK1047040B/zh
Priority to PT00944070T priority patent/PT1189608E/pt
Priority to GE4619A priority patent/GEP20043314B/en
Priority to AT00944070T priority patent/ATE245417T1/de
Priority to FR0008472A priority patent/FR2797587A1/fr
Publication of FI991485L publication Critical patent/FI991485L/fi
Priority to IL146807A priority patent/IL146807A/en
Priority to ZA200109868A priority patent/ZA200109868B/xx
Priority to NO20016203A priority patent/NO330260B1/no
Priority to BG106251A priority patent/BG65364B1/bg
Application granted granted Critical
Publication of FI109453B publication Critical patent/FI109453B/fi
Priority to US10/223,298 priority patent/US6797732B2/en
Priority to JP2008063280A priority patent/JP4885896B2/ja
Priority to NO20110090A priority patent/NO20110090L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
FI991485A 1999-06-30 1999-06-30 Farmaseuttinen koostumus FI109453B (fi)

Priority Applications (47)

Application Number Priority Date Filing Date Title
FI991485A FI109453B (fi) 1999-06-30 1999-06-30 Farmaseuttinen koostumus
TW089110218A TWI241187B (en) 1999-06-30 2000-05-26 Levodopa/carbidopa/entacapone pharmaceutical composition
PE2000000641A PE20010399A1 (es) 1999-06-30 2000-06-27 Composicion solida oral que contiene entacapona, levodopa y carbidopa
IT2000MI001450A ITMI20001450A1 (it) 1999-06-30 2000-06-28 Nuova composizione farmaceutica
SK1923-2001A SK286451B6 (sk) 1999-06-30 2000-06-29 Perorálna pevná kompozícia obsahujúca entakapon, levodopu a karbidopu a spôsoby jej prípravy a použitie
SI200030190T SI1189608T1 (en) 1999-06-30 2000-06-29 Levodopa/carbidopa/entacapone pharmaceutical preparation
ES00944070T ES2203495T3 (es) 1999-06-30 2000-06-29 Preparado farmaceutico de levodopa/carbidopa/entacapona.
CZ20014636A CZ303010B6 (cs) 1999-06-30 2000-06-29 Perorální pevná kompozice obsahující entacapon, levodopu a karbidopu, zpusoby její prípravy a použití
PL352775A PL197818B1 (pl) 1999-06-30 2000-06-29 Stałe doustne kompozycje lewodopa/karbidopa/entakapon, sposób ich wytwarzania oraz ich zastosowanie
TR2001/03763T TR200103763T2 (tr) 1999-06-30 2000-06-29 Levodopa/karbidopa/entakapon farmasötik preparasyonu.
YUP-925/01A RS50368B (sr) 1999-06-30 2000-06-29 Levodopa/karbidopa/entakapon farmaceutski preparat
ARP000103325A AR033796A1 (es) 1999-06-30 2000-06-29 Composicion farmaceutica
CA002378469A CA2378469C (en) 1999-06-30 2000-06-29 An oral solid composition comprising carbidopa, levodopa and entacapone
CZ2011-885A CZ304416B6 (cs) 1999-06-30 2000-06-29 Farmaceutická kompozice obsahující entacapon, levodopu a karbidopu a léčivo pro léčení Parkinsonovy choroby
CO00048944A CO5180579A1 (es) 1999-06-30 2000-06-29 Composicion oral solida que comprende levidopa, carbidopa y entacapone
MEP-2008-863A ME00520B (me) 1999-06-30 2000-06-29 Levodop/karbidop/entakapon farmaceutski preparat
EP00944070A EP1189608B1 (en) 1999-06-30 2000-06-29 Levodopa/carbidopa/entacapone pharmaceutical preparation
KR1020017015737A KR100905428B1 (ko) 1999-06-30 2000-06-29 레보도파/카비도파/엔타카폰 약학적 제제
HR20020088A HRP20020088B1 (hr) 1999-06-30 2000-06-29 Levodopa/karbidopa/entakapon farmaceutski pripravak
PCT/FI2000/000593 WO2001001984A1 (en) 1999-06-30 2000-06-29 Levodopa / carbidopa / entacapone pharmaceutical preparation
HU0202273A HU230395B1 (hu) 1999-06-30 2000-06-29 Levodopa /carbidopa/ entacapone tartalmú orálisan adagolható szilárd készítmény, eljárás ennek előállítására és ezt tartalmazó tabletta
UA2002010771A UA75047C2 (en) 1999-06-30 2000-06-29 Fixed dose composition of levodopa, carbidopa and entacapone
BRPI0011867A BRPI0011867B8 (pt) 1999-06-30 2000-06-29 preparação farmacêutica de levodopa/carbidopa/entacapona e processo para preparação da mesma
EEP200100716A EE05473B1 (et) 1999-06-30 2000-06-29 Levodopa/karbidopa/entakapooni farmatseutiline preparaat, selle valmistamise meetod ja kasutamine
JP2001507476A JP4204783B2 (ja) 1999-06-30 2000-06-29 レボドパ/カルビドパ/エンタカポン医薬製剤
CNB008095868A CN1168440C (zh) 1999-06-30 2000-06-29 左旋多巴/卡比多巴/恩他卡朋药物制剂
NZ515780A NZ515780A (en) 1999-06-30 2000-06-29 Levodopa / carbidopa / entacapone pharmaceutical preparation
AU58306/00A AU765932B2 (en) 1999-06-30 2000-06-29 Levodopa / carbidopa / entacapone pharmaceutical preparation
MYPI20002972A MY127685A (en) 1999-06-30 2000-06-29 Levodopa/carbidopa/entacapone pharmaceutical preparation
US09/605,529 US6500867B1 (en) 1999-06-30 2000-06-29 Pharmaceutical composition comprising entacapone, levodopa, and carbidopa
BR0011867-2A BR0011867A (pt) 1999-06-30 2000-06-29 Preparação farmacêutica de levodopa/carbidopa/entacapona
DK00944070T DK1189608T3 (da) 1999-06-30 2000-06-29 Farmaceutisk fremstilling på basis af levodopa, carbidopa og entacapon
MXPA01013167A MXPA01013167A (es) 1999-06-30 2000-06-29 Preparacion farmaceutica de levodopa / carbidopa / entacapona.
EA200200106A EA004503B1 (ru) 1999-06-30 2000-06-29 Фармацевтическая композиция леводопа/карбидопа/энтакапон
DE60004052T DE60004052T2 (de) 1999-06-30 2000-06-29 Pharmazeutische zubereitungen auf der basis von levodopa, carbidopa und entacapone
HK02108609.4A HK1047040B (zh) 1999-06-30 2000-06-29 左旋多巴/卡比多巴/恩他卡朋藥物製劑
PT00944070T PT1189608E (pt) 1999-06-30 2000-06-29 Preparacao farmaceutica de levodopa/carbidopa/entacapona
GE4619A GEP20043314B (en) 1999-06-30 2000-06-29 Pharmaceutical Composition Comprising Entacapone, Levodopa, and Carbidopa
AT00944070T ATE245417T1 (de) 1999-06-30 2000-06-29 Pharmazeutische zubereitungen auf der basis von levodopa, carbidopa und entacapone
FR0008472A FR2797587A1 (fr) 1999-06-30 2000-06-30 Nouvelle composition pharmaceutique
IL146807A IL146807A (en) 1999-06-30 2001-11-29 Levodopa/carbidopa/entacapone pharmaceutical preparation
ZA200109868A ZA200109868B (en) 1999-06-30 2001-11-29 Levodopa/carbidopa/entacapone pharmaceutical preparation.
NO20016203A NO330260B1 (no) 1999-06-30 2001-12-18 Oral, fast sammensetning omfattende levodopa/carbidopa/entacapon, fremgangsmate for fremstilling derav, samt anvendelse av en sammensetning omfattende levodopa/carbidopa/entacapon for fremstilling av et medikament til behandling av Parkinsons sykdom.
BG106251A BG65364B1 (bg) 1999-06-30 2001-12-20 Фармацевтичен препарат леводопа/карбидопа/ентакапон
US10/223,298 US6797732B2 (en) 1999-06-30 2002-08-20 Pharmaceutical composition comprising entracapone, levodopa, and carbidopa
JP2008063280A JP4885896B2 (ja) 1999-06-30 2008-03-12 レボドパ/カルビドパ/エンタカポン医薬製剤
NO20110090A NO20110090L (no) 1999-06-30 2011-01-19 Stabil fast oral sammensetning omfattende levodopa, carbidopa, og entacapon

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FI991485 1999-06-30
FI991485A FI109453B (fi) 1999-06-30 1999-06-30 Farmaseuttinen koostumus

Publications (3)

Publication Number Publication Date
FI991485A0 FI991485A0 (fi) 1999-06-30
FI991485L FI991485L (fi) 2000-12-31
FI109453B true FI109453B (fi) 2002-08-15

Family

ID=8554988

Family Applications (1)

Application Number Title Priority Date Filing Date
FI991485A FI109453B (fi) 1999-06-30 1999-06-30 Farmaseuttinen koostumus

Country Status (42)

Country Link
US (2) US6500867B1 (cs)
EP (1) EP1189608B1 (cs)
JP (2) JP4204783B2 (cs)
KR (1) KR100905428B1 (cs)
CN (1) CN1168440C (cs)
AR (1) AR033796A1 (cs)
AT (1) ATE245417T1 (cs)
AU (1) AU765932B2 (cs)
BG (1) BG65364B1 (cs)
BR (2) BR0011867A (cs)
CA (1) CA2378469C (cs)
CO (1) CO5180579A1 (cs)
CZ (2) CZ304416B6 (cs)
DE (1) DE60004052T2 (cs)
DK (1) DK1189608T3 (cs)
EA (1) EA004503B1 (cs)
EE (1) EE05473B1 (cs)
ES (1) ES2203495T3 (cs)
FI (1) FI109453B (cs)
FR (1) FR2797587A1 (cs)
GE (1) GEP20043314B (cs)
HK (1) HK1047040B (cs)
HR (1) HRP20020088B1 (cs)
HU (1) HU230395B1 (cs)
IL (1) IL146807A (cs)
IT (1) ITMI20001450A1 (cs)
ME (1) ME00520B (cs)
MX (1) MXPA01013167A (cs)
MY (1) MY127685A (cs)
NO (2) NO330260B1 (cs)
NZ (1) NZ515780A (cs)
PE (1) PE20010399A1 (cs)
PL (1) PL197818B1 (cs)
PT (1) PT1189608E (cs)
RS (1) RS50368B (cs)
SI (1) SI1189608T1 (cs)
SK (1) SK286451B6 (cs)
TR (1) TR200103763T2 (cs)
TW (1) TWI241187B (cs)
UA (1) UA75047C2 (cs)
WO (1) WO2001001984A1 (cs)
ZA (1) ZA200109868B (cs)

Families Citing this family (75)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI109453B (fi) 1999-06-30 2002-08-15 Orion Yhtymae Oyj Farmaseuttinen koostumus
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US20040166159A1 (en) * 2002-05-29 2004-08-26 Chien-Hsuan Han Pharmaceutical dosage forms having immediate and controlled release properties that contain an aromatic amino acid decarboxylase inhibitor and levodopa
US20030224045A1 (en) * 2002-05-29 2003-12-04 Chien-Hsuan Han Combination immediate release sustained release levodopa/carbidopa dosage forms
US20060013875A1 (en) * 2002-05-29 2006-01-19 Impax Laboratories, Inc. Combination immediate release controlled release levodopa/carbidopa dosage forms
US20050147670A1 (en) * 2002-05-29 2005-07-07 Impax Laboratories Inc. Oral disintegrating dosage forms
US20040006072A1 (en) * 2002-06-25 2004-01-08 Franz Robert M. Sustained-release alprazolam composition
EP1560569A4 (en) * 2002-10-11 2006-03-22 Depomed Dev Ltd GASTRORETENTIVE LEVODOPA DELIVERY FORM
AR044007A1 (es) 2003-04-11 2005-08-24 Newron Pharmaceuticals Inc Metodos para el tratamiento de la enfermedad de parkinson
EP1588704A1 (en) * 2004-04-22 2005-10-26 Newron Pharmaceuticals S.p.A. Alpha-aminoamide derivatives useful in the treatment of restless legs syndrome and addictive disorders
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US20060241183A1 (en) * 2004-09-28 2006-10-26 Farouk Karoum Compositions and methods of using D-DOPA to treat Parkinson's disease
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AU2006261893A1 (en) * 2005-06-23 2007-01-04 Combinatorx, Incorporated Improved dosage forms for movement disorder treatment
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US8772346B2 (en) * 2005-11-09 2014-07-08 Torrent Pharmaceuticals Limited Pharmaceutical composition
GB2429645A (en) * 2006-03-10 2007-03-07 Sekhsaria Chemicals Ltd Solid pharmaceutical composition comprising a COMT inhibitor, a starch and a wetting agent
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PT2413912T (pt) 2009-04-01 2019-06-11 Bial Portela & Ca Sa Formulações farmacêuticas compreendendo derivados de nitrocatecol e métodos para as produzir
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