ES514795A0 - Procedimiento para la preparacion de derivados substituidos de la piridazina. - Google Patents

Procedimiento para la preparacion de derivados substituidos de la piridazina.

Info

Publication number
ES514795A0
ES514795A0 ES514795A ES514795A ES514795A0 ES 514795 A0 ES514795 A0 ES 514795A0 ES 514795 A ES514795 A ES 514795A ES 514795 A ES514795 A ES 514795A ES 514795 A0 ES514795 A0 ES 514795A0
Authority
ES
Spain
Prior art keywords
piridazine
procedure
preparation
substituted derivatives
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES514795A
Other languages
English (en)
Spanish (es)
Other versions
ES8305738A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi SA filed Critical Sanofi SA
Publication of ES514795A0 publication Critical patent/ES514795A0/es
Publication of ES8305738A1 publication Critical patent/ES8305738A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
ES514795A 1981-08-07 1982-08-06 Procedimiento para la preparacion de derivados substituidos de la piridazina. Expired ES8305738A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8115380A FR2510998B1 (fr) 1981-08-07 1981-08-07 Nouveaux derives amines de la pyridazine, leur procede de preparation et les medicaments, a action desinhibitrice, qui en comportent

Publications (2)

Publication Number Publication Date
ES514795A0 true ES514795A0 (es) 1983-04-16
ES8305738A1 ES8305738A1 (es) 1983-04-16

Family

ID=9261294

Family Applications (2)

Application Number Title Priority Date Filing Date
ES514795A Expired ES8305738A1 (es) 1981-08-07 1982-08-06 Procedimiento para la preparacion de derivados substituidos de la piridazina.
ES514794A Expired ES8305737A1 (es) 1981-08-07 1982-08-06 Procedimiento para la preparacion de compuestos aminados de la piridazina.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES514794A Expired ES8305737A1 (es) 1981-08-07 1982-08-06 Procedimiento para la preparacion de compuestos aminados de la piridazina.

Country Status (30)

Country Link
US (1) US4508720A (enExample)
EP (2) EP0072726B1 (enExample)
JP (2) JPS5877867A (enExample)
KR (2) KR880001624B1 (enExample)
AR (2) AR231637A1 (enExample)
AT (2) ATE12227T1 (enExample)
AU (2) AU548931B2 (enExample)
CA (2) CA1179346A (enExample)
CS (2) CS229940B2 (enExample)
DD (2) DD202549A5 (enExample)
DE (2) DE3269383D1 (enExample)
DK (2) DK148795C (enExample)
EG (2) EG15788A (enExample)
ES (2) ES8305738A1 (enExample)
FI (2) FI72969C (enExample)
FR (1) FR2510998B1 (enExample)
GR (2) GR76430B (enExample)
HU (2) HU189166B (enExample)
IE (2) IE53388B1 (enExample)
IL (2) IL66409A (enExample)
MA (2) MA19560A1 (enExample)
NO (2) NO157102C (enExample)
NZ (2) NZ201518A (enExample)
OA (2) OA07175A (enExample)
PH (1) PH18545A (enExample)
PL (2) PL130647B1 (enExample)
PT (2) PT75351B (enExample)
SU (2) SU1138024A3 (enExample)
YU (2) YU172082A (enExample)
ZA (2) ZA825513B (enExample)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2540113A1 (fr) * 1983-01-27 1984-08-03 Sanofi Sa Acides derives de la pyridazine actifs sur le systeme nerveux central
US4565814A (en) * 1983-01-28 1986-01-21 Sanofi Pyridazine derivatives having a psychotropic action and compositions
US4628088A (en) * 1984-07-17 1986-12-09 Eli Lilly And Company Preparation of substituted pyridazines
EP0190563B1 (de) * 1985-01-14 1989-08-02 Boehringer Ingelheim Kg Neue 12-Amino-pyridazino[4',5':3,4]pyrrolo-[2,1-a]isochinoline, Verfahren zu ihrer Herstellung und ihre Verwendung
FR2642648B1 (fr) * 1989-02-07 1991-06-21 Sanofi Sa Utilisation de derives d'alkyl-5 pyridazine comme medicaments actifs sur le systeme cholinergique
US5461053A (en) * 1989-02-07 1995-10-24 Sanofi Pyridazine derivatives
FR2665442B1 (fr) * 1990-07-31 1992-12-04 Sanofi Sa Derives d'alkyl-6 pyridazine, procede de preparation et compositions pharmaceutiques en contenant.
PT93060B (pt) 1989-02-07 1995-12-29 Sanofi Sa Processo para a obtencao de derivados de piridazina e de composicoes farmaceuticas que os contem
FR2663326B2 (fr) * 1989-11-17 1992-10-16 Sanofi Sa Derives de la pyridazine, procede de preparation et compositions pharmaceutiques en contenant.
FR2642754B1 (fr) * 1989-02-07 1991-05-24 Sanofi Sa Nouveaux derives de la pyridazine, procede de preparation et compositions pharmaceutiques en contenant
US5656631A (en) * 1989-02-07 1997-08-12 Sanofi Pyridazine derivatives
FR2654727B1 (fr) * 1989-11-17 1992-03-27 Sanofi Sa Derives de la pyridazine, procede de preparation et compositions pharmaceutiques en contenant.
FR2676444B1 (fr) * 1991-05-16 1995-03-10 Sanofi Elf Nouveaux derives d'amino-3 pyridazines actifs sur le systeme nerveux central, procede de preparation et compositions pharmaceutiques en contenant.
US20100210590A1 (en) * 1995-09-27 2010-08-19 Northwestern University Compositions and treatments for seizure-related disorders
WO2003018563A1 (en) * 2001-08-31 2003-03-06 Northwestern University Anti-inflammatory and protein kinase inhibitor composition and method of use
WO2004014865A1 (en) * 2002-08-13 2004-02-19 Merck Sharp & Dohme Limited Phenylpyridazine derivatives as ligands for gaba receptors
EP1812007B1 (en) * 2004-11-02 2011-09-07 Northwestern University Pyridazine compounds and methods
EP2592075B1 (en) 2004-11-02 2015-04-29 Northwestern University Pyridazine compounds for the treatment of inflammatory diseases
EP2015751A2 (en) * 2006-04-28 2009-01-21 Northwestern University Salts of pyridazine compounds
CA2650625A1 (en) * 2006-04-28 2007-11-08 Northwestern University Formulations containing pyridazine compounds for treating neuroinflammatory diseases
WO2007127474A2 (en) * 2006-04-28 2007-11-08 Northwestern University Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
RU2555969C1 (ru) * 2014-07-09 2015-07-10 Юлия Алексеевна Щепочкина Керамическая масса для изготовления облицовочной плитки

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1345880A (en) * 1971-06-18 1974-02-06 Cepbepe Pyridazine derivatives

Also Published As

Publication number Publication date
DK148795C (da) 1986-03-10
NO822509L (no) 1983-02-08
JPH0459312B2 (enExample) 1992-09-21
AR231637A1 (es) 1985-01-31
FI72969B (fi) 1987-04-30
CA1174240A (en) 1984-09-11
NZ201518A (en) 1985-04-30
DK354382A (da) 1983-02-08
IL66408A0 (en) 1982-11-30
FI72968C (fi) 1987-08-10
MA19560A1 (fr) 1983-04-01
FR2510998B1 (fr) 1986-01-10
ES514794A0 (es) 1983-04-16
AU8655382A (en) 1983-02-10
PH18545A (en) 1985-08-09
PL130647B1 (en) 1984-08-31
GR76429B (enExample) 1984-08-10
IE53387B1 (en) 1988-10-26
DK148537C (da) 1986-01-13
DK354482A (da) 1983-02-08
ZA825512B (en) 1983-06-29
PT75351B (fr) 1984-08-01
ATE18216T1 (de) 1986-03-15
NO157102C (no) 1988-01-20
YU171882A (en) 1985-03-20
NO157861B (no) 1988-02-22
NZ201520A (en) 1985-04-30
DK148795B (da) 1985-09-30
CS229940B2 (en) 1984-07-16
DK148537B (da) 1985-07-29
SU1140685A3 (ru) 1985-02-15
EG15747A (en) 1986-06-30
PT75351A (fr) 1982-08-01
IE821779L (en) 1983-02-07
FI72968B (fi) 1987-04-30
KR890001569B1 (ko) 1989-05-08
IL66409A (en) 1985-09-29
ATE12227T1 (de) 1985-04-15
HU189166B (en) 1986-06-30
PT75350B (fr) 1984-08-01
SU1138024A3 (ru) 1985-01-30
PL137199B1 (en) 1986-05-31
AU548931B2 (en) 1986-01-09
US4508720A (en) 1985-04-02
AU8655482A (en) 1983-02-10
JPS5877868A (ja) 1983-05-11
AR231441A1 (es) 1984-11-30
KR840001145A (ko) 1984-03-28
ZA825513B (en) 1983-06-29
AU548930B2 (en) 1986-01-09
FR2510998A1 (fr) 1983-02-11
NO157102B (no) 1987-10-12
IE821778L (en) 1983-02-07
OA07175A (fr) 1984-04-30
MA19562A1 (fr) 1983-04-01
FI822748L (fi) 1983-02-08
EP0074863B1 (fr) 1986-02-26
FI72969C (fi) 1987-08-10
NO157861C (no) 1988-06-01
CS229941B2 (en) 1984-07-16
YU172082A (en) 1985-03-20
DE3262671D1 (en) 1985-04-25
KR880001624B1 (ko) 1988-09-02
HU190028B (en) 1986-08-28
DD202549A5 (de) 1983-09-21
IE53388B1 (en) 1988-10-26
IL66409A0 (en) 1982-11-30
DE3269383D1 (en) 1986-04-03
EG15788A (en) 1986-09-30
FI822747A0 (fi) 1982-08-06
OA07176A (fr) 1984-04-30
EP0072726B1 (fr) 1985-03-20
ES8305738A1 (es) 1983-04-16
FI822747L (fi) 1983-02-08
CA1179346A (en) 1984-12-11
PT75350A (fr) 1982-08-01
JPS5877867A (ja) 1983-05-11
PL237808A1 (en) 1983-02-28
DD202715A5 (de) 1983-09-28
ES8305737A1 (es) 1983-04-16
PL237809A1 (en) 1983-02-28
KR840001159A (ko) 1984-03-28
NO822510L (no) 1983-02-08
EP0074863A1 (fr) 1983-03-23
EP0072726A1 (fr) 1983-02-23
IL66408A (en) 1985-12-31
GR76430B (enExample) 1984-08-10
FI822748A0 (fi) 1982-08-06

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19991102