ES2609987T3 - Piridinonas bicíclicas novedosas - Google Patents

Piridinonas bicíclicas novedosas Download PDF

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Publication number
ES2609987T3
ES2609987T3 ES13792085.6T ES13792085T ES2609987T3 ES 2609987 T3 ES2609987 T3 ES 2609987T3 ES 13792085 T ES13792085 T ES 13792085T ES 2609987 T3 ES2609987 T3 ES 2609987T3
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ES
Spain
Prior art keywords
methyl
alkyl
mmol
phenyl
tetrahydrofuran
Prior art date
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Active
Application number
ES13792085.6T
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English (en)
Spanish (es)
Inventor
Christopher William Am Ende
Michael Eric GREEN
Douglas Scott Johnson
Gregory Wayne KAUFFMAN
Christopher John O'donnell
Nandini Chaturbhai Patel
Martin Youngjin Pettersson
Antonia Friederike STEPAN
Cory Michael Stiff
Chakrapani Subramanyam
Tuan Phong Tran
Patrick Robert Verhoest
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Pfizer Inc
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Pfizer Inc
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Publication of ES2609987T3 publication Critical patent/ES2609987T3/es
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Epidemiology (AREA)
ES13792085.6T 2012-09-21 2013-09-06 Piridinonas bicíclicas novedosas Active ES2609987T3 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261703969P 2012-09-21 2012-09-21
US201261703969P 2012-09-21
PCT/IB2013/058347 WO2014045156A1 (en) 2012-09-21 2013-09-06 Novel bicyclic pyridinones

Publications (1)

Publication Number Publication Date
ES2609987T3 true ES2609987T3 (es) 2017-04-25

Family

ID=49585452

Family Applications (1)

Application Number Title Priority Date Filing Date
ES13792085.6T Active ES2609987T3 (es) 2012-09-21 2013-09-06 Piridinonas bicíclicas novedosas

Country Status (46)

Country Link
US (3) US8916564B2 (enExample)
EP (1) EP2897956B1 (enExample)
JP (1) JP5844018B2 (enExample)
KR (1) KR101725696B1 (enExample)
CN (1) CN104662021B (enExample)
AP (1) AP2015008277A0 (enExample)
AR (1) AR092628A1 (enExample)
AU (1) AU2013319845B2 (enExample)
BR (1) BR112015006436A2 (enExample)
CA (1) CA2882386C (enExample)
CL (1) CL2015000717A1 (enExample)
CR (1) CR20150053A (enExample)
CU (1) CU20150021A7 (enExample)
CY (1) CY1118662T1 (enExample)
DK (1) DK2897956T3 (enExample)
DO (1) DOP2015000069A (enExample)
EA (1) EA026668B1 (enExample)
EC (1) ECSP15015594A (enExample)
ES (1) ES2609987T3 (enExample)
GE (1) GEP201706659B (enExample)
GT (1) GT201500069A (enExample)
HR (1) HRP20161558T1 (enExample)
HU (1) HUE031248T2 (enExample)
IL (1) IL237163A (enExample)
IN (1) IN2015DN01119A (enExample)
LT (1) LT2897956T (enExample)
MA (1) MA37886B1 (enExample)
MD (1) MD4583B1 (enExample)
ME (1) ME02571B (enExample)
MX (1) MX360599B (enExample)
MY (1) MY181891A (enExample)
NI (1) NI201500038A (enExample)
NZ (1) NZ704863A (enExample)
PE (1) PE20150686A1 (enExample)
PH (1) PH12015500376A1 (enExample)
PL (1) PL2897956T3 (enExample)
PT (1) PT2897956T (enExample)
RS (1) RS55426B1 (enExample)
SG (1) SG11201501074WA (enExample)
SI (1) SI2897956T1 (enExample)
TN (1) TN2015000084A1 (enExample)
TW (1) TWI500616B (enExample)
UA (1) UA110688C2 (enExample)
UY (1) UY35039A (enExample)
WO (1) WO2014045156A1 (enExample)
ZA (1) ZA201501195B (enExample)

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CN113402490B (zh) * 2021-03-29 2023-01-03 白银京宇新药业有限公司 一种1，2，6，7-四氢-8H-茚并[5，4-b]呋喃-8-酮的制备方法
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