NI201500038A - Piridinonas bicíclicas novedosas - Google Patents

Piridinonas bicíclicas novedosas

Info

Publication number
NI201500038A
NI201500038A NI201500038A NI201500038A NI201500038A NI 201500038 A NI201500038 A NI 201500038A NI 201500038 A NI201500038 A NI 201500038A NI 201500038 A NI201500038 A NI 201500038A NI 201500038 A NI201500038 A NI 201500038A
Authority
NI
Nicaragua
Prior art keywords
new bicyclic
compounds
pyridinones
bicyclic pyridinones
new
Prior art date
Application number
NI201500038A
Other languages
English (en)
Spanish (es)
Inventor
William Am Ende Christopher
Eric Green Michael
Scott Johnson Douglas
Wayne Kauffmann Gregory
John O'donnell Christopher
Chaturbhai Patel Nandini
Youngjin Pettersson Martin
Friederike Stepan Antonia
Michael Stiff Cory
Subramanyam Chakrapani
Phong Tran Tuan
Robert Verhoest Patrick
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NI201500038A publication Critical patent/NI201500038A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epidemiology (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
NI201500038A 2012-09-21 2015-03-19 Piridinonas bicíclicas novedosas NI201500038A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261703969P 2012-09-21 2012-09-21

Publications (1)

Publication Number Publication Date
NI201500038A true NI201500038A (es) 2015-06-05

Family

ID=49585452

Family Applications (1)

Application Number Title Priority Date Filing Date
NI201500038A NI201500038A (es) 2012-09-21 2015-03-19 Piridinonas bicíclicas novedosas

Country Status (46)

Country Link
US (3) US8916564B2 (enExample)
EP (1) EP2897956B1 (enExample)
JP (1) JP5844018B2 (enExample)
KR (1) KR101725696B1 (enExample)
CN (1) CN104662021B (enExample)
AP (1) AP2015008277A0 (enExample)
AR (1) AR092628A1 (enExample)
AU (1) AU2013319845B2 (enExample)
BR (1) BR112015006436A2 (enExample)
CA (1) CA2882386C (enExample)
CL (1) CL2015000717A1 (enExample)
CR (1) CR20150053A (enExample)
CU (1) CU20150021A7 (enExample)
CY (1) CY1118662T1 (enExample)
DK (1) DK2897956T3 (enExample)
DO (1) DOP2015000069A (enExample)
EA (1) EA026668B1 (enExample)
EC (1) ECSP15015594A (enExample)
ES (1) ES2609987T3 (enExample)
GE (1) GEP201706659B (enExample)
GT (1) GT201500069A (enExample)
HR (1) HRP20161558T1 (enExample)
HU (1) HUE031248T2 (enExample)
IL (1) IL237163A (enExample)
IN (1) IN2015DN01119A (enExample)
LT (1) LT2897956T (enExample)
MA (1) MA37886B1 (enExample)
MD (1) MD4583B1 (enExample)
ME (1) ME02571B (enExample)
MX (1) MX360599B (enExample)
MY (1) MY181891A (enExample)
NI (1) NI201500038A (enExample)
NZ (1) NZ704863A (enExample)
PE (1) PE20150686A1 (enExample)
PH (1) PH12015500376A1 (enExample)
PL (1) PL2897956T3 (enExample)
PT (1) PT2897956T (enExample)
RS (1) RS55426B1 (enExample)
SG (1) SG11201501074WA (enExample)
SI (1) SI2897956T1 (enExample)
TN (1) TN2015000084A1 (enExample)
TW (1) TWI500616B (enExample)
UA (1) UA110688C2 (enExample)
UY (1) UY35039A (enExample)
WO (1) WO2014045156A1 (enExample)
ZA (1) ZA201501195B (enExample)

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DK3126361T3 (da) * 2014-04-01 2020-01-02 Pfizer Chromen og 1,1a,2,7b-tetrahydrocyclopropa[c]chromen- pyridopyrazindioner som gamma-sekretase-modulatorer
EA033423B1 (ru) * 2015-02-03 2019-10-31 Pfizer Циклопропанбензофуранилпиридопиразиндионы
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JP6904612B2 (ja) * 2016-12-16 2021-07-21 パイプライン セラピューティクス， インコーポレイテッド 蝸牛シナプス障害を処置する方法
TW202034900A (zh) 2018-10-02 2020-10-01 美商頻率醫療公司 有關耳用治療劑之醫藥組成物及方法
US20210393621A1 (en) 2018-10-26 2021-12-23 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
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PH12022551379A1 (en) 2019-12-06 2023-05-03 Vertex Pharma Substituted tetrahydrofurans as modulators of sodium channels
CN113402490B (zh) * 2021-03-29 2023-01-03 白银京宇新药业有限公司 一种1，2，6，7-四氢-8H-茚并[5，4-b]呋喃-8-酮的制备方法
DK4347031T3 (da) 2021-06-04 2025-12-01 Vertex Pharma N-(hydroxyalkyl-(hetero)aryl)-tetrahydrofuran-carboxamider som modulatorer af natriumkanaler
CN114034792B (zh) * 2021-11-09 2024-06-25 山东新华制药股份有限公司 检测氯酮含量的液相色谱分析方法

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