EE04567B1 - Kristalliline monohdraat, meetod selle valmistamiseks ja selle kasutamine ravimi valmistamiseks - Google Patents

Kristalliline monohdraat, meetod selle valmistamiseks ja selle kasutamine ravimi valmistamiseks

Info

Publication number
EE04567B1
EE04567B1 EEP200300171A EEP200300171A EE04567B1 EE 04567 B1 EE04567 B1 EE 04567B1 EE P200300171 A EEP200300171 A EE P200300171A EE P200300171 A EEP200300171 A EE P200300171A EE 04567 B1 EE04567 B1 EE 04567B1
Authority
EE
Estonia
Prior art keywords
monoh
drape
medicament
crystalline
manufacture
Prior art date
Application number
EEP200300171A
Other languages
English (en)
Estonian (et)
Inventor
Banholzer Rolf
Sieger Peter
Kulinna Christian
Trunk Michael
Ludwig August Graulich Manfred
Specht Peter
Meissner Helmut
Mathes Andreas
Original Assignee
Boehringer Ingelheim Pharma Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE04567(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma Gmbh & Co. Kg filed Critical Boehringer Ingelheim Pharma Gmbh & Co. Kg
Publication of EE200300171A publication Critical patent/EE200300171A/xx
Publication of EE04567B1 publication Critical patent/EE04567B1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06Oxygen atoms
    • C07D451/10Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
EEP200300171A 2000-10-12 2001-09-28 Kristalliline monohdraat, meetod selle valmistamiseks ja selle kasutamine ravimi valmistamiseks EE04567B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12
PCT/EP2001/011225 WO2002030928A1 (de) 2000-10-12 2001-09-28 Kristallines monohydrat, verfahren zu dessen herstellung und dessen verwendung zur herstellung eines arzneimittels

Publications (2)

Publication Number Publication Date
EE200300171A EE200300171A (et) 2003-06-16
EE04567B1 true EE04567B1 (et) 2005-12-15

Family

ID=7659568

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300171A EE04567B1 (et) 2000-10-12 2001-09-28 Kristalliline monohdraat, meetod selle valmistamiseks ja selle kasutamine ravimi valmistamiseks

Country Status (47)

Country Link
EP (2) EP1326862B1 (ru)
JP (1) JP3764422B2 (ru)
KR (1) KR100823860B1 (ru)
CN (2) CN100519558C (ru)
AP (1) AP1572A (ru)
AR (2) AR034389A1 (ru)
AT (1) ATE276253T1 (ru)
AU (2) AU2002214996B2 (ru)
BG (1) BG66161B1 (ru)
BR (1) BR0114584A (ru)
CA (1) CA2425539C (ru)
CR (1) CR6938A (ru)
CZ (1) CZ301841B6 (ru)
DE (1) DE50103666D1 (ru)
DK (1) DK1326862T3 (ru)
DZ (1) DZ3478A1 (ru)
EA (1) EA004381B1 (ru)
EC (1) ECSP034540A (ru)
EE (1) EE04567B1 (ru)
EG (1) EG24142A (ru)
ES (1) ES2228965T3 (ru)
GE (1) GEP20063905B (ru)
HK (2) HK1060567A1 (ru)
HR (1) HRP20030276B1 (ru)
HU (1) HU226830B1 (ru)
IL (2) IL155335A0 (ru)
IS (1) IS2339B (ru)
MA (1) MA25842A1 (ru)
ME (2) ME00243B (ru)
MX (1) MXPA03003221A (ru)
MY (1) MY126931A (ru)
NO (1) NO328465B1 (ru)
NZ (1) NZ525733A (ru)
OA (1) OA12403A (ru)
PE (1) PE20020422A1 (ru)
PL (1) PL207870B1 (ru)
PT (1) PT1326862E (ru)
RS (1) RS50218B (ru)
SA (1) SA01220412B1 (ru)
SI (1) SI1326862T1 (ru)
SK (1) SK287009B6 (ru)
TR (1) TR200402579T4 (ru)
TW (1) TW589313B (ru)
UA (1) UA74215C2 (ru)
UY (2) UY26962A1 (ru)
WO (1) WO2002030928A1 (ru)
ZA (1) ZA200302500B (ru)

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Also Published As

Publication number Publication date
TR200402579T4 (tr) 2004-12-21
PT1326862E (pt) 2004-11-30
DE50103666D1 (de) 2004-10-21
BG66161B1 (bg) 2011-09-30
IS2339B (is) 2008-02-15
HRP20030276B1 (en) 2006-02-28
AR068527A2 (es) 2009-11-18
PE20020422A1 (es) 2002-06-28
UY26962A1 (es) 2002-06-20
EP1326862A1 (de) 2003-07-16
HUP0301022A2 (hu) 2003-10-28
CN1733761A (zh) 2006-02-15
SK287009B6 (sk) 2009-09-07
AP1572A (en) 2006-02-13
HRP20030276A2 (en) 2005-02-28
DK1326862T3 (da) 2004-11-22
NO20031694D0 (no) 2003-04-11
YU27303A (sh) 2006-05-25
UY34901A (es) 2015-02-27
ME00243B (me) 2011-05-10
AR034389A1 (es) 2004-02-25
IL155335A0 (en) 2003-11-23
HU226830B1 (en) 2009-11-30
IS6772A (is) 2003-04-09
ECSP034540A (es) 2003-07-25
GEP20063905B (en) 2006-08-25
HK1060567A1 (en) 2004-08-13
WO2002030928A1 (de) 2002-04-18
AU2002214996B2 (en) 2007-03-15
MY126931A (en) 2006-10-31
CA2425539C (en) 2007-04-03
CA2425539A1 (en) 2003-04-11
JP2004526668A (ja) 2004-09-02
EA004381B1 (ru) 2004-04-29
HUP0301022A3 (en) 2005-12-28
CN1469877A (zh) 2004-01-21
MEP40008A (en) 2011-02-10
CZ301841B6 (cs) 2010-07-07
EG24142A (en) 2008-08-06
IL155335A (en) 2009-02-11
RS50218B (sr) 2009-07-15
EA200300457A1 (ru) 2003-10-30
OA12403A (en) 2006-04-18
NO20031694L (no) 2003-04-11
CR6938A (es) 2004-10-28
MXPA03003221A (es) 2004-12-03
EP1468998A1 (de) 2004-10-20
HK1086557A1 (en) 2006-09-22
NZ525733A (en) 2005-01-28
DZ3478A1 (fr) 2002-04-18
SK4362003A3 (en) 2003-08-05
NO328465B1 (no) 2010-02-22
PL207870B1 (pl) 2011-02-28
KR20030042008A (ko) 2003-05-27
PL366041A1 (en) 2005-01-24
BR0114584A (pt) 2003-08-26
BG107687A (bg) 2003-09-30
JP3764422B2 (ja) 2006-04-05
CN100519558C (zh) 2009-07-29
EP1326862B1 (de) 2004-09-15
UA74215C2 (ru) 2005-11-15
SA01220412B1 (ar) 2006-11-05
KR100823860B1 (ko) 2008-04-21
ZA200302500B (en) 2004-04-22
ES2228965T3 (es) 2005-04-16
SI1326862T1 (en) 2005-02-28
MA25842A1 (fr) 2003-07-01
CN1221549C (zh) 2005-10-05
EE200300171A (et) 2003-06-16
AP2003002775A0 (en) 2003-03-31
AU1499602A (en) 2002-04-22
TW589313B (en) 2004-06-01
ATE276253T1 (de) 2004-10-15

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