ECSP034540A - Monohidrato cristalino, procedimiento para su preparacion y su utilizacion para la preparacion de un medicamento - Google Patents

Monohidrato cristalino, procedimiento para su preparacion y su utilizacion para la preparacion de un medicamento

Info

Publication number
ECSP034540A
ECSP034540A EC2003004540A ECSP034540A ECSP034540A EC SP034540 A ECSP034540 A EC SP034540A EC 2003004540 A EC2003004540 A EC 2003004540A EC SP034540 A ECSP034540 A EC SP034540A EC SP034540 A ECSP034540 A EC SP034540A
Authority
EC
Ecuador
Prior art keywords
preparation
procedure
crystalline
monohidrate
medicinal product
Prior art date
Application number
EC2003004540A
Other languages
English (en)
Spanish (es)
Inventor
Rolf Banholzer
Peter Sieger
Christian Kulinna
Michael Trunk
Manfred Ludwig August Graulich
Peter Specht
Helmut Meissner
Andreas Mathes
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP034540(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of ECSP034540A publication Critical patent/ECSP034540A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
EC2003004540A 2000-10-12 2003-04-07 Monohidrato cristalino, procedimiento para su preparacion y su utilizacion para la preparacion de un medicamento ECSP034540A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12

Publications (1)

Publication Number Publication Date
ECSP034540A true ECSP034540A (es) 2003-07-25

Family

ID=7659568

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2003004540A ECSP034540A (es) 2000-10-12 2003-04-07 Monohidrato cristalino, procedimiento para su preparacion y su utilizacion para la preparacion de un medicamento

Country Status (46)

Country Link
EP (2) EP1468998A1 (de)
JP (1) JP3764422B2 (de)
KR (1) KR100823860B1 (de)
CN (2) CN1221549C (de)
AP (1) AP1572A (de)
AR (2) AR034389A1 (de)
AT (1) ATE276253T1 (de)
AU (2) AU2002214996B2 (de)
BG (1) BG66161B1 (de)
BR (1) BR0114584A (de)
CA (1) CA2425539C (de)
CR (1) CR6938A (de)
CZ (1) CZ301841B6 (de)
DE (1) DE50103666D1 (de)
DK (1) DK1326862T3 (de)
DZ (1) DZ3478A1 (de)
EA (1) EA004381B1 (de)
EC (1) ECSP034540A (de)
EE (1) EE04567B1 (de)
EG (1) EG24142A (de)
ES (1) ES2228965T3 (de)
GE (1) GEP20063905B (de)
HR (1) HRP20030276B1 (de)
HU (1) HU226830B1 (de)
IL (2) IL155335A0 (de)
IS (1) IS2339B (de)
MA (1) MA25842A1 (de)
ME (2) MEP40008A (de)
MX (1) MXPA03003221A (de)
MY (1) MY126931A (de)
NO (1) NO328465B1 (de)
NZ (1) NZ525733A (de)
OA (1) OA12403A (de)
PE (1) PE20020422A1 (de)
PL (1) PL207870B1 (de)
PT (1) PT1326862E (de)
RS (1) RS50218B (de)
SA (1) SA01220412B1 (de)
SI (1) SI1326862T1 (de)
SK (1) SK287009B6 (de)
TR (1) TR200402579T4 (de)
TW (1) TW589313B (de)
UA (1) UA74215C2 (de)
UY (2) UY26962A1 (de)
WO (1) WO2002030928A1 (de)
ZA (1) ZA200302500B (de)

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US7220742B2 (en) 2004-05-14 2007-05-22 Boehringer Ingelheim International Gmbh Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
DE102004024454A1 (de) 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Enantiomerenreine Betaagonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
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KR20080007645A (ko) 2005-04-28 2008-01-22 베링거 인겔하임 인터내셔날 게엠베하 염증성 질환 치료용 신규 화합물
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KR20080024532A (ko) * 2005-06-15 2008-03-18 베링거 인겔하임 인터내셔날 게엠베하 신규한 티오트로퓸 염의 제조방법, 신규한 티오트로퓸 염및 이의 약제학적 조성물
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Also Published As

Publication number Publication date
CN1733761A (zh) 2006-02-15
EE04567B1 (et) 2005-12-15
AP1572A (en) 2006-02-13
HK1060567A1 (en) 2004-08-13
EA200300457A1 (ru) 2003-10-30
ATE276253T1 (de) 2004-10-15
CA2425539A1 (en) 2003-04-11
EP1326862B1 (de) 2004-09-15
UA74215C2 (uk) 2005-11-15
PT1326862E (pt) 2004-11-30
CZ301841B6 (cs) 2010-07-07
EP1468998A1 (de) 2004-10-20
ES2228965T3 (es) 2005-04-16
UY26962A1 (es) 2002-06-20
NO20031694L (no) 2003-04-11
NZ525733A (en) 2005-01-28
MA25842A1 (fr) 2003-07-01
IS6772A (is) 2003-04-09
OA12403A (en) 2006-04-18
NO328465B1 (no) 2010-02-22
EG24142A (en) 2008-08-06
HRP20030276A2 (en) 2005-02-28
AU1499602A (en) 2002-04-22
TW589313B (en) 2004-06-01
HU226830B1 (en) 2009-11-30
BR0114584A (pt) 2003-08-26
KR100823860B1 (ko) 2008-04-21
HUP0301022A2 (hu) 2003-10-28
CN1221549C (zh) 2005-10-05
EE200300171A (et) 2003-06-16
HUP0301022A3 (en) 2005-12-28
AP2003002775A0 (en) 2003-03-31
AR068527A2 (es) 2009-11-18
CA2425539C (en) 2007-04-03
PE20020422A1 (es) 2002-06-28
UY34901A (es) 2015-02-27
MY126931A (en) 2006-10-31
HK1086557A1 (zh) 2006-09-22
DK1326862T3 (da) 2004-11-22
DE50103666D1 (de) 2004-10-21
YU27303A (sh) 2006-05-25
IS2339B (is) 2008-02-15
SK4362003A3 (en) 2003-08-05
ZA200302500B (en) 2004-04-22
AR034389A1 (es) 2004-02-25
MEP40008A (en) 2011-02-10
TR200402579T4 (tr) 2004-12-21
SI1326862T1 (sl) 2005-02-28
EP1326862A1 (de) 2003-07-16
IL155335A (en) 2009-02-11
BG66161B1 (bg) 2011-09-30
GEP20063905B (en) 2006-08-25
JP3764422B2 (ja) 2006-04-05
EA004381B1 (ru) 2004-04-29
ME00243B (me) 2011-05-10
NO20031694D0 (no) 2003-04-11
KR20030042008A (ko) 2003-05-27
DZ3478A1 (fr) 2002-04-18
SK287009B6 (sk) 2009-09-07
CR6938A (es) 2004-10-28
WO2002030928A1 (de) 2002-04-18
HRP20030276B1 (en) 2006-02-28
RS50218B (sr) 2009-07-15
PL366041A1 (en) 2005-01-24
PL207870B1 (pl) 2011-02-28
AU2002214996B2 (en) 2007-03-15
CN1469877A (zh) 2004-01-21
IL155335A0 (en) 2003-11-23
MXPA03003221A (es) 2004-12-03
BG107687A (bg) 2003-09-30
JP2004526668A (ja) 2004-09-02
CN100519558C (zh) 2009-07-29
SA01220412B1 (ar) 2006-11-05

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