EA200300211A1 - Азабициклические соединения, способ их получения и их применение в качестве лекарственных средств, в частности в качестве антибактериальных средств - Google Patents

Азабициклические соединения, способ их получения и их применение в качестве лекарственных средств, в частности в качестве антибактериальных средств

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Publication number
EA200300211A1
EA200300211A1 EA200300211A EA200300211A EA200300211A1 EA 200300211 A1 EA200300211 A1 EA 200300211A1 EA 200300211 A EA200300211 A EA 200300211A EA 200300211 A EA200300211 A EA 200300211A EA 200300211 A1 EA200300211 A1 EA 200300211A1
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EA
Eurasian Patent Office
Prior art keywords
compounds
application
azabiccal
medicine
production
Prior art date
Application number
EA200300211A
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English (en)
Other versions
EA004920B1 (ru
Inventor
Максим Лампила
Жозеф Асзоди
Дэвид Ален Роулендс
Клод Фроментэн
Original Assignee
Авентис Фарма Са
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8853181&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200300211(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Авентис Фарма Са filed Critical Авентис Фарма Са
Publication of EA200300211A1 publication Critical patent/EA200300211A1/ru
Publication of EA004920B1 publication Critical patent/EA004920B1/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Изобретение относится к новым гетероциклическим соединениям общей формулы (I) и их солям с основанием или с кислотой. Изобретение также относится к способу получения этих соединений, а также к их применению в качестве лекарственных средств, в частности в качестве антибактериальных средств.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200300211A 2000-08-01 2001-07-24 Азабициклические соединения, способ их получения и их применение в качестве лекарственных средств, в частности в качестве антибактериальных средств EA004920B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0010121A FR2812635B1 (fr) 2000-08-01 2000-08-01 Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens
PCT/FR2001/002418 WO2002010172A1 (fr) 2000-08-01 2001-07-24 Composes azabicycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens

Publications (2)

Publication Number Publication Date
EA200300211A1 true EA200300211A1 (ru) 2003-06-26
EA004920B1 EA004920B1 (ru) 2004-10-28

Family

ID=8853181

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200300211A EA004920B1 (ru) 2000-08-01 2001-07-24 Азабициклические соединения, способ их получения и их применение в качестве лекарственных средств, в частности в качестве антибактериальных средств

Country Status (42)

Country Link
US (5) US7112592B2 (ru)
EP (1) EP1307457B1 (ru)
JP (2) JP4515704B2 (ru)
KR (1) KR100632906B1 (ru)
CN (1) CN1289500C (ru)
AP (1) AP1614A (ru)
AR (1) AR031716A1 (ru)
AT (1) ATE263768T1 (ru)
AU (2) AU7990501A (ru)
BG (1) BG66094B1 (ru)
BR (1) BRPI0112986B8 (ru)
CA (1) CA2417475C (ru)
CR (1) CR6895A (ru)
CZ (1) CZ294956B6 (ru)
DE (1) DE60102702T2 (ru)
DK (1) DK1307457T3 (ru)
DZ (1) DZ3397A1 (ru)
EA (1) EA004920B1 (ru)
EC (1) ECSP034460A (ru)
EE (1) EE05183B1 (ru)
ES (1) ES2220793T3 (ru)
FR (1) FR2812635B1 (ru)
HK (1) HK1060356A1 (ru)
HR (1) HRP20030034B1 (ru)
HU (1) HU226889B1 (ru)
IL (2) IL154187A0 (ru)
MA (1) MA26938A1 (ru)
ME (2) MEP17108A (ru)
MX (1) MXPA03000881A (ru)
NO (1) NO324940B1 (ru)
NZ (1) NZ523707A (ru)
OA (1) OA12347A (ru)
PL (2) PL216028B1 (ru)
PT (1) PT1307457E (ru)
RS (1) RS50214B (ru)
SI (1) SI1307457T1 (ru)
SK (1) SK287597B6 (ru)
TR (1) TR200400859T4 (ru)
TW (1) TWI292401B (ru)
UA (1) UA73791C2 (ru)
WO (1) WO2002010172A1 (ru)
ZA (1) ZA200300676B (ru)

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* Cited by examiner, † Cited by third party
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