OA12347A - Composés azabicycliques, leur préparation et leur utilisation comme médicaments, notamment comme anti-bactériens. - Google Patents

Composés azabicycliques, leur préparation et leur utilisation comme médicaments, notamment comme anti-bactériens. Download PDF

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Publication number
OA12347A
OA12347A OA1200300019A OA1200300019A OA12347A OA 12347 A OA12347 A OA 12347A OA 1200300019 A OA1200300019 A OA 1200300019A OA 1200300019 A OA1200300019 A OA 1200300019A OA 12347 A OA12347 A OA 12347A
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OA
OAPI
Prior art keywords
group
dichloromethane
added
reduced pressure
trans
Prior art date
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OA1200300019A
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English (en)
French (fr)
Inventor
Maxime Lampilas
Jozsef Aszodi
David Alan Rowlands
Claude Fromentin
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Aventis Pharma Sa
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8853181&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA12347(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of OA12347A publication Critical patent/OA12347A/fr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
OA1200300019A 2000-08-01 2001-07-24 Composés azabicycliques, leur préparation et leur utilisation comme médicaments, notamment comme anti-bactériens. OA12347A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0010121A FR2812635B1 (fr) 2000-08-01 2000-08-01 Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens

Publications (1)

Publication Number Publication Date
OA12347A true OA12347A (fr) 2006-05-15

Family

ID=8853181

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200300019A OA12347A (fr) 2000-08-01 2001-07-24 Composés azabicycliques, leur préparation et leur utilisation comme médicaments, notamment comme anti-bactériens.

Country Status (42)

Country Link
US (5) US7112592B2 (ru)
EP (1) EP1307457B1 (ru)
JP (2) JP4515704B2 (ru)
KR (1) KR100632906B1 (ru)
CN (1) CN1289500C (ru)
AP (1) AP1614A (ru)
AR (1) AR031716A1 (ru)
AT (1) ATE263768T1 (ru)
AU (2) AU2001279905B2 (ru)
BG (1) BG66094B1 (ru)
BR (1) BRPI0112986B8 (ru)
CA (1) CA2417475C (ru)
CR (1) CR6895A (ru)
CZ (1) CZ294956B6 (ru)
DE (1) DE60102702T2 (ru)
DK (1) DK1307457T3 (ru)
DZ (1) DZ3397A1 (ru)
EA (1) EA004920B1 (ru)
EC (1) ECSP034460A (ru)
EE (1) EE05183B1 (ru)
ES (1) ES2220793T3 (ru)
FR (1) FR2812635B1 (ru)
HK (1) HK1060356A1 (ru)
HR (1) HRP20030034B1 (ru)
HU (1) HU226889B1 (ru)
IL (2) IL154187A0 (ru)
MA (1) MA26938A1 (ru)
ME (2) ME00060B (ru)
MX (1) MXPA03000881A (ru)
NO (1) NO324940B1 (ru)
NZ (1) NZ523707A (ru)
OA (1) OA12347A (ru)
PL (2) PL234468B1 (ru)
PT (1) PT1307457E (ru)
RS (1) RS50214B (ru)
SI (1) SI1307457T1 (ru)
SK (1) SK287597B6 (ru)
TR (1) TR200400859T4 (ru)
TW (1) TWI292401B (ru)
UA (1) UA73791C2 (ru)
WO (1) WO2002010172A1 (ru)
ZA (1) ZA200300676B (ru)

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FR2835186B1 (fr) * 2002-01-28 2006-10-20 Aventis Pharma Sa Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases
FR2844273B1 (fr) 2002-09-05 2008-04-04 Aventis Pharma Sa Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens.
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