BR9408450A - Antagonistas da neuroquinina diazabiciclicos - Google Patents

Antagonistas da neuroquinina diazabiciclicos

Info

Publication number
BR9408450A
BR9408450A BR9408450A BR9408450A BR9408450A BR 9408450 A BR9408450 A BR 9408450A BR 9408450 A BR9408450 A BR 9408450A BR 9408450 A BR9408450 A BR 9408450A BR 9408450 A BR9408450 A BR 9408450A
Authority
BR
Brazil
Prior art keywords
diazabicyclic
neurokinin antagonists
compounds
formula
disorders
Prior art date
Application number
BR9408450A
Other languages
English (en)
Inventor
Harry R Howard
Kevin D Shenk
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of BR9408450A publication Critical patent/BR9408450A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR9408450A 1993-12-29 1994-11-14 Antagonistas da neuroquinina diazabiciclicos BR9408450A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17503493A 1993-12-29 1993-12-29
PCT/IB1994/000352 WO1995018129A1 (en) 1993-12-29 1994-11-14 Diazabicyclic neurokinin antagonists

Publications (1)

Publication Number Publication Date
BR9408450A true BR9408450A (pt) 1997-08-05

Family

ID=22638565

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9408450A BR9408450A (pt) 1993-12-29 1994-11-14 Antagonistas da neuroquinina diazabiciclicos

Country Status (26)

Country Link
US (2) US5854239A (pt)
EP (1) EP0737194B1 (pt)
JP (1) JP2895630B2 (pt)
KR (1) KR100197454B1 (pt)
CN (1) CN1046515C (pt)
AT (1) ATE177099T1 (pt)
AU (1) AU699465B2 (pt)
BR (1) BR9408450A (pt)
CA (1) CA2180263C (pt)
CO (1) CO4230019A1 (pt)
CZ (1) CZ282567B6 (pt)
DE (1) DE69416869T2 (pt)
DK (1) DK0737194T3 (pt)
ES (1) ES2127946T3 (pt)
FI (1) FI108296B (pt)
GR (1) GR3029853T3 (pt)
HU (1) HUT74682A (pt)
IL (1) IL112118A (pt)
NO (1) NO305600B1 (pt)
NZ (1) NZ274915A (pt)
PE (1) PE49395A1 (pt)
PL (1) PL179435B1 (pt)
RU (1) RU2124014C1 (pt)
TW (1) TW369526B (pt)
WO (1) WO1995018129A1 (pt)
ZA (1) ZA9410339B (pt)

Families Citing this family (67)

* Cited by examiner, † Cited by third party
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BR9408450A (pt) * 1993-12-29 1997-08-05 Pfizer Antagonistas da neuroquinina diazabiciclicos
FR2786770B1 (fr) * 1998-12-04 2001-01-19 Synthelabo Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique
AU7552401A (en) * 2000-06-12 2001-12-24 Univ Rochester Method of treating symptoms of hormonal variation, including hot flashes, using tachykinin receptor antagonist
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FR2825705B1 (fr) * 2001-06-08 2005-05-20 Aventis Pharma Sa Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens
FR2835186B1 (fr) * 2002-01-28 2006-10-20 Aventis Pharma Sa Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases
FR2844273B1 (fr) 2002-09-05 2008-04-04 Aventis Pharma Sa Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens.
FR2848210B1 (fr) * 2002-12-06 2007-10-19 Aventis Pharma Sa Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens et inhibiteurs de beta-lactamases
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US20110218176A1 (en) 2006-11-01 2011-09-08 Barbara Brooke Jennings-Spring Compounds, methods, and treatments for abnormal signaling pathways for prenatal and postnatal development
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US3494923A (en) * 1965-05-28 1970-02-10 Sterling Drug Inc 1,2,3,4,5,8-hexahydro-1,5-methanobenzo (f)(1,4)diazocine
WO1992015585A1 (en) * 1991-03-01 1992-09-17 Pfizer Inc. 1-azabicyclo[3.2.2]nonan-3-amine derivatives
BR9408450A (pt) * 1993-12-29 1997-08-05 Pfizer Antagonistas da neuroquinina diazabiciclicos

Also Published As

Publication number Publication date
US6110919A (en) 2000-08-29
FI946140A0 (fi) 1994-12-28
US5854239A (en) 1998-12-29
PE49395A1 (es) 1996-01-06
PL315193A1 (en) 1996-10-14
PL179435B1 (pl) 2000-09-29
CZ188696A3 (en) 1996-10-16
RU2124014C1 (ru) 1998-12-27
JP2895630B2 (ja) 1999-05-24
NZ274915A (en) 1997-11-24
GR3029853T3 (en) 1999-07-30
DK0737194T3 (da) 1999-09-27
NO962742L (no) 1996-06-28
HU9601790D0 (en) 1996-09-30
ATE177099T1 (de) 1999-03-15
NO305600B1 (no) 1999-06-28
ZA9410339B (en) 1996-06-28
DE69416869T2 (de) 1999-07-01
FI946140A (fi) 1995-06-30
KR100197454B1 (ko) 1999-06-15
DE69416869D1 (de) 1999-04-08
HUT74682A (en) 1997-01-28
CN1046515C (zh) 1999-11-17
IL112118A0 (en) 1995-03-15
CN1139434A (zh) 1997-01-01
EP0737194A1 (en) 1996-10-16
CA2180263C (en) 2000-05-16
FI108296B (fi) 2001-12-31
CZ282567B6 (cs) 1997-08-13
ES2127946T3 (es) 1999-05-01
JPH09500904A (ja) 1997-01-28
AU699465B2 (en) 1998-12-03
WO1995018129A1 (en) 1995-07-06
CO4230019A1 (es) 1995-10-19
EP0737194B1 (en) 1999-03-03
TW369526B (en) 1999-09-11
IL112118A (en) 1998-10-30
AU8002194A (en) 1995-07-17
NO962742D0 (no) 1996-06-28

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