DK3174868T3 - Forbindelser, der er aktive mod bromodomæner - Google Patents
Forbindelser, der er aktive mod bromodomæner Download PDFInfo
- Publication number
- DK3174868T3 DK3174868T3 DK15744908.3T DK15744908T DK3174868T3 DK 3174868 T3 DK3174868 T3 DK 3174868T3 DK 15744908 T DK15744908 T DK 15744908T DK 3174868 T3 DK3174868 T3 DK 3174868T3
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- DK
- Denmark
- Prior art keywords
- bromodomains
- active against
- compounds active
- compounds
- against bromodomains
- Prior art date
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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| AU2017245641A1 (en) * | 2016-04-07 | 2018-09-13 | Glaxosmithkline Intellectual Property (No.2) Limited | Pyridyl derivatives as bromodomain inhibitors |
| TW202413340A (zh) | 2016-07-12 | 2024-04-01 | 美商銳新醫藥公司 | 作為異位shp2抑制劑之2,5-雙取代型3-甲基吡嗪及2,5,6-三取代型3-甲基吡嗪 |
| US20190247302A1 (en) * | 2016-10-21 | 2019-08-15 | University Of Miami | Materials and methods for treating ophthalmic inflammation |
| AU2017385292B2 (en) * | 2016-12-27 | 2020-05-14 | Fujifilm Corporation | Antitumor agent and bromodomain inhibitor |
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| RU2020123241A (ru) | 2017-12-15 | 2022-01-17 | Революшн Медсинз, Инк. | Полициклические соединения в качестве аллостерических ингибиторов shp2 |
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