DK166498B1 - Macrolidforbindelser, fremgangsmaade til fremstilling deraf, praeparater indeholdende saadanne forbindelser samt en ikke-terapeutisk fremgangsmaade til bekaempelse af skadedyr under anvendelse af en saadan forbindelse - Google Patents

Macrolidforbindelser, fremgangsmaade til fremstilling deraf, praeparater indeholdende saadanne forbindelser samt en ikke-terapeutisk fremgangsmaade til bekaempelse af skadedyr under anvendelse af en saadan forbindelse Download PDF

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Publication number
DK166498B1
DK166498B1 DK290287A DK290287A DK166498B1 DK 166498 B1 DK166498 B1 DK 166498B1 DK 290287 A DK290287 A DK 290287A DK 290287 A DK290287 A DK 290287A DK 166498 B1 DK166498 B1 DK 166498B1
Authority
DK
Denmark
Prior art keywords
compound
hydroxy
compounds
general formula
alkyl
Prior art date
Application number
DK290287A
Other languages
Danish (da)
English (en)
Other versions
DK290287D0 (da
DK290287A (da
Inventor
Derek R Sutherland
Michael V J Ramsay
Edward P Tiley
Oswy Z Pereira
John B Ward
Neil Porter
Hazel M Noble
Richard A Fletton
David Noble
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB868613790A external-priority patent/GB8613790D0/en
Priority claimed from GB868625854A external-priority patent/GB8625854D0/en
Priority claimed from GB878708423A external-priority patent/GB8708423D0/en
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of DK290287D0 publication Critical patent/DK290287D0/da
Publication of DK290287A publication Critical patent/DK290287A/da
Application granted granted Critical
Publication of DK166498B1 publication Critical patent/DK166498B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N49/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds containing the group, wherein m+n>=1, both X together may also mean —Y— or a direct carbon-to-carbon bond, and the carbon atoms marked with an asterisk are not part of any ring system other than that which may be formed by the atoms X, the carbon atoms in square brackets being part of any acyclic or cyclic structure, or the group, wherein A means a carbon atom or Y, n>=0, and not more than one of these carbon atoms being a member of the same ring system, e.g. juvenile insect hormones or mimics thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Public Health (AREA)
  • Insects & Arthropods (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK290287A 1986-06-06 1987-06-04 Macrolidforbindelser, fremgangsmaade til fremstilling deraf, praeparater indeholdende saadanne forbindelser samt en ikke-terapeutisk fremgangsmaade til bekaempelse af skadedyr under anvendelse af en saadan forbindelse DK166498B1 (da)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GB8613790 1986-06-06
GB868613790A GB8613790D0 (en) 1986-06-06 1986-06-06 Chemical compounds
GB868625854A GB8625854D0 (en) 1986-10-29 1986-10-29 Chemical process
GB8625854 1986-10-29
GB8708423 1987-04-08
GB878708423A GB8708423D0 (en) 1987-04-08 1987-04-08 Chemical compounds

Publications (3)

Publication Number Publication Date
DK290287D0 DK290287D0 (da) 1987-06-04
DK290287A DK290287A (da) 1987-12-07
DK166498B1 true DK166498B1 (da) 1993-06-01

Family

ID=27263057

Family Applications (1)

Application Number Title Priority Date Filing Date
DK290287A DK166498B1 (da) 1986-06-06 1987-06-04 Macrolidforbindelser, fremgangsmaade til fremstilling deraf, praeparater indeholdende saadanne forbindelser samt en ikke-terapeutisk fremgangsmaade til bekaempelse af skadedyr under anvendelse af en saadan forbindelse

Country Status (35)

Country Link
US (1) US4900753A (zh)
JP (1) JP2648147B2 (zh)
KR (1) KR950010077B1 (zh)
CN (1) CN1023858C (zh)
AR (1) AR244691A1 (zh)
AT (1) AT398571B (zh)
AU (1) AU609399B2 (zh)
BE (1) BE1000201A4 (zh)
BR (1) BR8702866A (zh)
CA (1) CA1296329C (zh)
CH (1) CH677670A5 (zh)
DE (3) DE3745133C2 (zh)
DK (1) DK166498B1 (zh)
EG (1) EG18752A (zh)
ES (1) ES2006479A6 (zh)
FI (2) FI90663C (zh)
FR (1) FR2599742B1 (zh)
GB (1) GB2192630B (zh)
GE (1) GEP19981388B (zh)
GR (1) GR870891B (zh)
HU (1) HU199847B (zh)
IE (1) IE60411B1 (zh)
IL (1) IL82776A (zh)
IT (1) IT1206015B (zh)
LU (2) LU86908A1 (zh)
LV (2) LV10280A (zh)
NL (2) NL193376C (zh)
NZ (1) NZ220587A (zh)
OA (1) OA08606A (zh)
PH (1) PH23948A (zh)
PL (3) PL155723B1 (zh)
PT (1) PT85018B (zh)
SE (1) SE503399C2 (zh)
TR (1) TR28970A (zh)
UA (1) UA45300C2 (zh)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4886828A (en) * 1986-09-12 1989-12-12 American Cyanamid Company Δ22 -derivatives of LL-F28249 compounds
EP0259779B1 (en) * 1986-09-12 1994-08-10 American Cyanamid Company 23-Oxo (Keto) and 23-imino Derivatives of LL-F28249 Compounds
EP0260537A1 (en) * 1986-09-12 1988-03-23 American Cyanamid Company 13-Deoxy-23-oxo(keto) and 23-imino derivatives of 13-deoxy C-076-aglycone compounds
GB8721377D0 (en) * 1987-09-11 1987-10-21 Glaxo Group Ltd Chemical compounds
GB8811036D0 (en) * 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
GB8813150D0 (en) * 1988-06-03 1988-07-06 American Cyanamid Co Chemical compounds
GB8905605D0 (en) * 1989-03-11 1989-04-26 Beecham Group Plc Novel compounds
NZ233680A (en) * 1989-05-17 1995-02-24 Beecham Group Plc Avermectins and milbemycins and compositions thereof
US4988824A (en) * 1989-09-11 1991-01-29 Maulding Donald R Process for the preparation of 23-(C1-C6 alkyloxime)-LL-F28249 compounds
WO1992010170A1 (en) * 1990-12-07 1992-06-25 Temple University - Of The Commonwealth System Of Higher Education Stabilized insect nematode compositions
JP2855181B2 (ja) 1993-12-10 1999-02-10 敏雄 鈴木 松類の枯損防止用組成物及び防止方法
DE60118132T2 (de) 2000-10-10 2006-10-19 Wyeth Anthelmintika
US7348417B2 (en) * 2003-08-07 2008-03-25 Wyeth Method of purifying moxidectin through crystallization
US20090214676A1 (en) * 2005-04-30 2009-08-27 Tissuetech, Inc. Method for treating ocular demodex
JP4939025B2 (ja) * 2005-09-30 2012-05-23 三菱電線工業株式会社 電熱ヒータ付きハンドル用グリップ部材
EP1849363A1 (en) * 2006-03-09 2007-10-31 Cheminova A/S Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin
US8128968B2 (en) 2007-08-29 2012-03-06 Tissuetech, Inc. Compositions and methods for treating Demodex infestations
AU2012345813B2 (en) * 2011-12-02 2017-02-02 Boehringer lngelheim Vetmedica GMBH Long-acting injectable moxidectin formulations and novel moxidectin crystal forms
FR2995605B1 (fr) * 2012-09-18 2014-09-19 Sanofi Sa Derives de macrolides, leur preparation et leur application therapeutique.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH15982A (en) * 1977-10-03 1983-05-18 Merck & Co Inc Selective hydrogenation producta of c-076 compounds and derivatives thereof
US4289760A (en) * 1980-05-02 1981-09-15 Merck & Co., Inc. 23-Keto derivatives of C-076 compounds
US4423209A (en) * 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
JPS59108785A (ja) * 1982-11-25 1984-06-23 Sankyo Co Ltd ミルベマイシン類の５−オキシム誘導体
JPS60126289A (ja) * 1983-11-14 1985-07-05 Sankyo Co Ltd ミルベマイシン類の５−カ−ボネ−ト誘導体
EP0170006B1 (en) * 1984-06-05 1992-07-08 American Cyanamid Company Method and compositions for helmintic, arthropod ectoparasitic and acaridal infections with novel agents
US4579864A (en) * 1984-06-11 1986-04-01 Merck & Co., Inc. Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives
CH666690A5 (de) * 1984-09-14 1988-08-15 Glaxo Group Ltd Antibiotisch wirkende verbindungen der makrolidgruppe aus streptomyces-mikroorganismen, ihre herstellung und verwendung.
IL78621A (en) * 1985-04-30 1991-06-30 American Cyanamid Co Mylbemycin analogs,their preparation and pesticidal compositions containing them
EP0259779B1 (en) * 1986-09-12 1994-08-10 American Cyanamid Company 23-Oxo (Keto) and 23-imino Derivatives of LL-F28249 Compounds

Also Published As

Publication number Publication date
LU88790I2 (fr) 1997-03-18
LU86908A1 (fr) 1988-01-20
GB2192630A (en) 1988-01-20
BE1000201A4 (fr) 1988-08-23
PT85018A (en) 1987-07-01
EG18752A (en) 1993-12-30
PH23948A (en) 1990-01-23
NL990026I2 (nl) 1999-12-01
TR28970A (tr) 1997-07-21
GB8713239D0 (en) 1987-07-08
LV10280A (lv) 1994-10-20
PL153226B1 (en) 1991-03-29
ES2006479A6 (es) 1989-05-01
DK290287D0 (da) 1987-06-04
NL990026I1 (nl) 1999-11-01
DE3745133C2 (de) 1998-01-02
DE19875029I2 (de) 2001-11-22
OA08606A (en) 1988-11-30
AR244691A1 (es) 1993-11-30
GR870891B (en) 1987-10-02
CN87104431A (zh) 1987-12-30
JP2648147B2 (ja) 1997-08-27
ATA143887A (de) 1994-05-15
HU199847B (en) 1990-03-28
FI90549C (fi) 1994-02-25
DK290287A (da) 1987-12-07
SE8702361D0 (sv) 1987-06-05
NZ220587A (en) 1990-05-28
AU7387387A (en) 1987-12-10
CH677670A5 (zh) 1991-06-14
FI90549B (fi) 1993-11-15
NL193376B (nl) 1999-04-01
HUT44254A (en) 1988-02-29
KR880000441A (ko) 1988-03-25
CN1023858C (zh) 1994-02-23
IE60411B1 (en) 1994-07-13
GB2192630B (en) 1990-05-23
IL82776A (en) 1992-02-16
DE3718926C2 (de) 1998-01-15
FR2599742B1 (fr) 1989-05-19
AU609399B2 (en) 1991-05-02
NL8701322A (nl) 1988-01-04
CA1296329C (en) 1992-02-25
IT8748023A0 (it) 1987-06-05
FI90663B (fi) 1993-11-30
DE3718926A1 (de) 1987-12-10
PL155723B1 (en) 1991-12-31
SE503399C2 (sv) 1996-06-10
FI90663C (fi) 1994-03-10
PL266100A1 (en) 1988-07-21
JPS6354375A (ja) 1988-03-08
PL153036B1 (en) 1991-02-28
BR8702866A (pt) 1988-03-01
LV10781B (en) 1996-10-20
FI872517A (fi) 1987-12-07
FI923445A (fi) 1992-07-30
LV10781A (lv) 1995-08-20
NL193376C (nl) 1999-08-03
SE8702361L (sv) 1987-12-07
FR2599742A1 (fr) 1987-12-11
IL82776A0 (en) 1987-12-20
IT1206015B (it) 1989-04-05
AT398571B (de) 1994-12-27
GEP19981388B (en) 1998-11-10
PT85018B (pt) 1990-03-08
FI923445A0 (fi) 1992-07-30
US4900753A (en) 1990-02-13
IE871496L (en) 1987-12-06
KR950010077B1 (ko) 1995-09-06
FI872517A0 (fi) 1987-06-04
UA45300C2 (uk) 2002-04-15

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
CTFF Application for supplementary protection certificate (spc) filed

Free format text: CA 1995 00018, 951109

CTFG Supplementary protection certificate (spc) issued

Free format text: CA 1995 00018, 951109, EXPIRES: 20091230

PUP Patent expired