DK0733635T3 - Krystalformer af et thieno[2,3-b] [1,5]benzodiazepin-derivat og fremgangsmåde til deres fremstilling - Google Patents

Krystalformer af et thieno[2,3-b] [1,5]benzodiazepin-derivat og fremgangsmåde til deres fremstilling

Info

Publication number
DK0733635T3
DK0733635T3 DK96302000T DK96302000T DK0733635T3 DK 0733635 T3 DK0733635 T3 DK 0733635T3 DK 96302000 T DK96302000 T DK 96302000T DK 96302000 T DK96302000 T DK 96302000T DK 0733635 T3 DK0733635 T3 DK 0733635T3
Authority
DK
Denmark
Prior art keywords
thieno
preparation
crystal forms
benzodiazepine derivative
benzodiazepine
Prior art date
Application number
DK96302000T
Other languages
Danish (da)
English (en)
Inventor
Charles Arthur Bunnell
Samuel Dean Larsen
Barry Arnold Hendriksen
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23621056&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0733635(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK0733635T3 publication Critical patent/DK0733635T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicinal Preparation (AREA)
DK96302000T 1995-03-24 1996-03-22 Krystalformer af et thieno[2,3-b] [1,5]benzodiazepin-derivat og fremgangsmåde til deres fremstilling DK0733635T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40956695A 1995-03-24 1995-03-24

Publications (1)

Publication Number Publication Date
DK0733635T3 true DK0733635T3 (da) 2001-10-08

Family

ID=23621056

Family Applications (4)

Application Number Title Priority Date Filing Date
DK96302000T DK0733635T3 (da) 1995-03-24 1996-03-22 Krystalformer af et thieno[2,3-b] [1,5]benzodiazepin-derivat og fremgangsmåde til deres fremstilling
DK00203573T DK1095941T3 (da) 1995-03-24 1996-03-22 Fremgangsmåde og krystalformer for 2-methyl-thieno-benzodiazepin
DK03077455T DK1445259T3 (da) 1995-03-24 1996-03-22 Anvendelse af krystalformer for 2-methyl-thieno-benzodiazepin
DK108997A DK108997A (da) 1995-03-24 1997-09-23 Fremstilling og krystalformer af 2-methylthien-benzodiazepin

Family Applications After (3)

Application Number Title Priority Date Filing Date
DK00203573T DK1095941T3 (da) 1995-03-24 1996-03-22 Fremgangsmåde og krystalformer for 2-methyl-thieno-benzodiazepin
DK03077455T DK1445259T3 (da) 1995-03-24 1996-03-22 Anvendelse af krystalformer for 2-methyl-thieno-benzodiazepin
DK108997A DK108997A (da) 1995-03-24 1997-09-23 Fremstilling og krystalformer af 2-methylthien-benzodiazepin

Country Status (49)

Country Link
US (1) US5736541A (no)
EP (3) EP1445259B1 (no)
JP (1) JPH11502535A (no)
KR (1) KR100399688B1 (no)
CN (1) CN1065536C (no)
AP (1) AP828A (no)
AR (2) AR002719A1 (no)
AT (4) AT406771B (no)
AU (1) AU706471B2 (no)
BG (1) BG62619B1 (no)
BR (1) BR9607790A (no)
CA (1) CA2214005C (no)
CH (1) CH690579A5 (no)
CO (1) CO4650278A1 (no)
CZ (1) CZ292688B6 (no)
DE (4) DE69636313T2 (no)
DK (4) DK0733635T3 (no)
EA (1) EA000149B1 (no)
EE (1) EE03489B1 (no)
EG (1) EG23659A (no)
ES (3) ES2208220T3 (no)
FI (1) FI973750A (no)
GB (1) GB2313835B (no)
HK (1) HK1013988A1 (no)
HU (1) HU224989B1 (no)
IL (1) IL117610A (no)
IS (1) IS1896B (no)
LT (1) LT4349B (no)
LU (1) LU90096B1 (no)
LV (1) LV12018B (no)
MY (1) MY114701A (no)
NO (1) NO314663B1 (no)
NZ (1) NZ306110A (no)
OA (1) OA10510A (no)
PA (1) PA8353701A1 (no)
PE (1) PE44897A1 (no)
PL (1) PL183723B1 (no)
PT (3) PT1095941E (no)
RO (1) RO118872B1 (no)
SE (1) SE9703205D0 (no)
SI (4) SI9620040B (no)
SK (1) SK284143B6 (no)
SV (1) SV1996000031A (no)
TR (1) TR199701017T1 (no)
TW (2) TW442488B (no)
UA (1) UA44765C2 (no)
WO (1) WO1996030375A1 (no)
YU (1) YU49478B (no)
ZA (2) ZA962342B (no)

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Also Published As

Publication number Publication date
HK1013988A1 (en) 1999-09-17
NO974365D0 (no) 1997-09-22
WO1996030375A1 (en) 1996-10-03
EP1445259B1 (en) 2006-06-28
AP9701065A0 (en) 1997-10-31
AR010448A1 (es) 2000-06-28
YU49478B (sh) 2006-05-25
CN1179160A (zh) 1998-04-15
EA000149B1 (ru) 1998-10-29
DE69636313T2 (de) 2007-05-31
CA2214005C (en) 2001-07-03
ES2208220T3 (es) 2004-06-16
CO4650278A1 (es) 1998-09-03
LV12018B (en) 1998-09-20
LU90096B1 (fr) 1997-07-22
EP1095941B1 (en) 2003-10-08
HUP9802824A2 (hu) 1999-06-28
LT4349B (lt) 1998-05-25
ES2266719T3 (es) 2007-03-01
US5736541A (en) 1998-04-07
AU5427996A (en) 1996-10-16
MX9707183A (es) 1997-11-29
BG101900A (en) 1999-03-31
IL117610A (en) 2001-08-26
DE69614426D1 (de) 2001-09-20
FI973750A0 (fi) 1997-09-22
HUP9802824A3 (en) 2000-01-28
UA44765C2 (uk) 2002-03-15
SI9620040A (sl) 1998-06-30
PL183723B1 (pl) 2002-07-31
DE69630324T2 (de) 2004-07-29
EE03489B1 (et) 2001-08-15
AT406771B (de) 2000-08-25
DE69614426T2 (de) 2002-05-23
IS4564A (is) 1997-09-22
EE9700232A (et) 1998-04-15
GB9719819D0 (en) 1997-11-19
HU224989B1 (en) 2006-05-29
EG23659A (en) 2007-03-26
KR19980703188A (ko) 1998-10-15
OA10510A (en) 2002-04-24
TW513432B (en) 2002-12-11
ATE204280T1 (de) 2001-09-15
CH690579A5 (de) 2000-10-31
SV1996000031A (es) 1998-03-27
ES2159346T3 (es) 2001-10-01
SI9620040B (sl) 2002-02-28
GB2313835A (en) 1997-12-10
IL117610A0 (en) 1996-07-23
DK108997A (da) 1997-11-12
TW442488B (en) 2001-06-23
AP828A (en) 2000-04-28
LT97148A (en) 1998-01-26
CN1065536C (zh) 2001-05-09
EP1445259A1 (en) 2004-08-11
BR9607790A (pt) 1998-07-07
SI1445259T1 (sl) 2006-10-31
ATE331719T1 (de) 2006-07-15
SK284143B6 (sk) 2004-10-05
LV12018A (lv) 1998-04-20
RO118872B1 (ro) 2003-12-30
EP0733635B1 (en) 2001-08-16
SI0733635T1 (en) 2002-06-30
CZ300097A3 (en) 1997-12-17
MY114701A (en) 2002-12-31
SE9703205L (sv) 1997-09-05
YU17796A (sh) 1999-03-04
DE19681286T1 (de) 1998-04-02
CZ292688B6 (cs) 2003-11-12
BG62619B1 (bg) 2000-03-31
SE9703205D0 (sv) 1997-09-05
AR002719A1 (es) 1998-04-29
NO314663B1 (no) 2003-04-28
DE69630324D1 (de) 2003-11-13
KR100399688B1 (ko) 2004-02-18
NZ306110A (en) 1998-09-24
DE69636313D1 (de) 2006-08-10
PA8353701A1 (es) 1998-09-18
PT1445259E (pt) 2006-10-31
JPH11502535A (ja) 1999-03-02
ATE251627T1 (de) 2003-10-15
CA2214005A1 (en) 1996-10-03
EA199700262A1 (ru) 1998-02-26
SI1095941T1 (en) 2003-12-31
AU706471B2 (en) 1999-06-17
FI973750A (fi) 1997-09-22
SK121897A3 (en) 1998-03-04
TR199701017T1 (xx) 1998-01-21
ZA962342B (en) 1997-09-22
EP0733635A1 (en) 1996-09-25
DK1445259T3 (da) 2006-10-16
ATA902196A (de) 2000-01-15
PT733635E (pt) 2001-12-28
PT1095941E (pt) 2004-02-27
ZA962344B (en) 1997-09-22
EP1095941A1 (en) 2001-05-02
PE44897A1 (es) 1997-10-22
NO974365L (no) 1997-09-22
PL322501A1 (en) 1998-02-02
DK1095941T3 (da) 2004-02-16
IS1896B (is) 2003-10-20
GB2313835B (en) 1998-09-16

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