CO7071131A2 - Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluor-3-fenilquinazolin-4(3h)-ona - Google Patents

Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluor-3-fenilquinazolin-4(3h)-ona

Info

Publication number
CO7071131A2
CO7071131A2 CO14202424A CO14202424A CO7071131A2 CO 7071131 A2 CO7071131 A2 CO 7071131A2 CO 14202424 A CO14202424 A CO 14202424A CO 14202424 A CO14202424 A CO 14202424A CO 7071131 A2 CO7071131 A2 CO 7071131A2
Authority
CO
Colombia
Prior art keywords
phenylquinazolin
purin
ylamino
fluor
propyl
Prior art date
Application number
CO14202424A
Other languages
English (en)
Spanish (es)
Inventor
Ernest Carra
Michael Gerber
Bing Shi
Keiko Sujino
Duong Tran
Fang Wang
Jerry B Evarts
Original Assignee
Gilead Calistoga Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO7071131(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Calistoga Llc filed Critical Gilead Calistoga Llc
Publication of CO7071131A2 publication Critical patent/CO7071131A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32Nitrogen atom
    • C07D473/34Nitrogen atom attached in position 6, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
CO14202424A 2012-03-05 2014-09-12 Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluor-3-fenilquinazolin-4(3h)-ona CO7071131A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05

Publications (1)

Publication Number Publication Date
CO7071131A2 true CO7071131A2 (es) 2014-09-30

Family

ID=49117265

Family Applications (1)

Application Number Title Priority Date Filing Date
CO14202424A CO7071131A2 (es) 2012-03-05 2014-09-12 Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluor-3-fenilquinazolin-4(3h)-ona

Country Status (31)

Country Link
US (3) US8865730B2 (enExample)
EP (1) EP2834241B1 (enExample)
JP (2) JP2015509537A (enExample)
KR (1) KR20140133590A (enExample)
CN (2) CN106146506A (enExample)
AP (1) AP2014007875A0 (enExample)
AR (1) AR090253A1 (enExample)
AU (1) AU2013203620B2 (enExample)
BR (1) BR112014021935A2 (enExample)
CA (1) CA2864305C (enExample)
CL (1) CL2014002358A1 (enExample)
CO (1) CO7071131A2 (enExample)
CR (1) CR20140460A (enExample)
EA (3) EA025407B1 (enExample)
EC (1) ECSP14020478A (enExample)
ES (1) ES2848273T3 (enExample)
IN (1) IN2014DN07105A (enExample)
MA (1) MA37379A1 (enExample)
MD (1) MD20140100A2 (enExample)
MX (1) MX2014010656A (enExample)
NZ (1) NZ629684A (enExample)
PE (1) PE20141792A1 (enExample)
PH (1) PH12014501920A1 (enExample)
PL (1) PL2834241T3 (enExample)
PT (1) PT2834241T (enExample)
SG (1) SG11201405446PA (enExample)
SI (1) SI2834241T1 (enExample)
TW (1) TW201350486A (enExample)
UY (1) UY34656A (enExample)
WO (1) WO2013134288A1 (enExample)
ZA (1) ZA201405870B (enExample)

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TWI649326B (zh) 2015-07-02 2019-02-01 瑞士商赫孚孟拉羅股份公司 苯并氧氮呯噁唑啶酮化合物及其製備方法
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CZ2015575A3 (cs) * 2015-08-26 2017-03-08 Zentiva, K.S. Soli 5-fluoro-3-fenyl-2-[(1S)-1-(9H-purin-6-ylamino)propyl]quinazolin-4-onu a jejich příprava
CN106565716B (zh) * 2015-10-10 2021-06-15 上海创诺制药有限公司 一种Idelalisib晶型A及其制备方法
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CN106632337B (zh) * 2016-10-18 2018-11-20 湖北生物医药产业技术研究院有限公司 艾代拉里斯的晶型、药物组合物、制备方法和用途
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CN107573345B (zh) * 2017-09-12 2020-01-10 浙江乐普药业股份有限公司 一种艾代拉利司及其中间体的制备方法
CN109575027A (zh) * 2017-09-29 2019-04-05 宁波爱诺医药科技有限公司 一种抗肿瘤药物艾德力布的一水合物及其制备方法
WO2019178596A1 (en) 2018-03-16 2019-09-19 Johnson Matthey Public Limited Company Pyridine or n,n-dimethyl acetamide solvated solid state forms of solvated idelalisib, their use and preparation
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GB202109006D0 (en) 2021-06-23 2021-08-04 Anglo American Minerio De Ferro Brasil S/A Method of and system for operating a grinding mill
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