CN1826322B - 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物 - Google Patents

用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物 Download PDF

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CN1826322B
CN1826322B CN2004800210095A CN200480021009A CN1826322B CN 1826322 B CN1826322 B CN 1826322B CN 2004800210095 A CN2004800210095 A CN 2004800210095A CN 200480021009 A CN200480021009 A CN 200480021009A CN 1826322 B CN1826322 B CN 1826322B
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phenyl
pyrazole
urea
methyl
group
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CN1826322A (zh
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布拉德利·特加登
洪纳帕·贾亚库马尔
李红梅
索尼娅·斯特拉-普莱内特
彼得·伊恩·多萨
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Arena Pharmaceuticals Inc
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CN2004800210095A 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物 Expired - Fee Related CN1826322B (zh)

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Application Number Priority Date Filing Date Title
US48957203P 2003-07-22 2003-07-22
US60/489,572 2003-07-22
US50358603P 2003-09-16 2003-09-16
US60/503,586 2003-09-16
PCT/US2004/023488 WO2005012254A1 (en) 2003-07-22 2004-07-21 Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of disorders related therto

Related Child Applications (2)

Application Number Title Priority Date Filing Date
CN201010199162.4A Division CN101875961B (zh) 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物
CN201010200790A Division CN101871931A (zh) 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物

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CN1826322A CN1826322A (zh) 2006-08-30
CN1826322B true CN1826322B (zh) 2012-04-18

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CN2004800210095A Expired - Fee Related CN1826322B (zh) 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物
CN201010200790A Pending CN101871931A (zh) 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物
CN201010199162.4A Expired - Fee Related CN101875961B (zh) 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物

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CN201010200790A Pending CN101871931A (zh) 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物
CN201010199162.4A Expired - Fee Related CN101875961B (zh) 2003-07-22 2004-07-21 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物

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DK1558582T3 (da) 2003-07-22 2006-05-08 Arena Pharm Inc Diaryl og arylheteroarylureaderivater som modulatorer af aktiviteten af 5-HT2A-serotoninreceptoren anvendelige til profylakse eller behandling af forstyrrelser relateret dertil
WO2005103011A1 (en) * 2004-03-23 2005-11-03 Arena Pharmaceuticals, Inc. Processes for preparing substituted n-aryl-n’-[3-(1h-pyrazol-5-yl) phenyl] ureas and intermediates thereof
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US20150073141A1 (en) 2015-03-12
US20160374990A1 (en) 2016-12-29
US9775829B2 (en) 2017-10-03
EA200600295A1 (ru) 2006-08-25
NO20060877L (no) 2006-02-22
ECSP066269A (es) 2006-07-28
KR101157272B1 (ko) 2012-06-15
HK1072943A1 (en) 2005-09-16
TNSN06017A1 (en) 2007-10-03
NZ544331A (en) 2010-03-26
MXPA06000795A (es) 2006-08-23
CN101875961A (zh) 2010-11-03
EP1558582B1 (en) 2005-12-21
JP2007039461A (ja) 2007-02-15
DK1558582T3 (da) 2006-05-08
TW200523253A (en) 2005-07-16
ATE313532T1 (de) 2006-01-15
US20070072857A1 (en) 2007-03-29

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