CL2017000240A1 - Compuestos activos hacia bromodominios - Google Patents

Compuestos activos hacia bromodominios

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Publication number
CL2017000240A1
CL2017000240A1 CL2017000240A CL2017000240A CL2017000240A1 CL 2017000240 A1 CL2017000240 A1 CL 2017000240A1 CL 2017000240 A CL2017000240 A CL 2017000240A CL 2017000240 A CL2017000240 A CL 2017000240A CL 2017000240 A1 CL2017000240 A1 CL 2017000240A1
Authority
CL
Chile
Prior art keywords
bromodominiums
active compounds
compounds towards
compounds
towards
Prior art date
Application number
CL2017000240A
Other languages
English (en)
Spanish (es)
Inventor
Seitzberg Jimmi Gerner
Akinleminu Kronborg Tine Titilola
Visnha Poljak
Gitte Friberg
Lene Teuber
Original Assignee
Nuevolution As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nuevolution As filed Critical Nuevolution As
Publication of CL2017000240A1 publication Critical patent/CL2017000240A1/es

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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08—Bridged systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4704—2-Quinolinones, e.g. carbostyril
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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