CH621558A5 - Process for the preparation of kanamycin derivatives with antibacterial activity - Google Patents

Process for the preparation of kanamycin derivatives with antibacterial activity Download PDF

Info

Publication number
CH621558A5
CH621558A5 CH1593175A CH1593175A CH621558A5 CH 621558 A5 CH621558 A5 CH 621558A5 CH 1593175 A CH1593175 A CH 1593175A CH 1593175 A CH1593175 A CH 1593175A CH 621558 A5 CH621558 A5 CH 621558A5
Authority
CH
Switzerland
Prior art keywords
formula
compound
amino
water
vii
Prior art date
Application number
CH1593175A
Other languages
German (de)
English (en)
Inventor
Takayuki Naito
Susumu Nakagawa
Yukio Narita
Soichiro Toda
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of CH621558A5 publication Critical patent/CH621558A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
CH1593175A 1974-12-09 1975-12-08 Process for the preparation of kanamycin derivatives with antibacterial activity CH621558A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US53078774A 1974-12-09 1974-12-09

Publications (1)

Publication Number Publication Date
CH621558A5 true CH621558A5 (en) 1981-02-13

Family

ID=24114972

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1593175A CH621558A5 (en) 1974-12-09 1975-12-08 Process for the preparation of kanamycin derivatives with antibacterial activity

Country Status (17)

Country Link
JP (1) JPS51105036A (xx)
BE (1) BE836292A (xx)
CA (1) CA1052780A (xx)
CH (1) CH621558A5 (xx)
CS (1) CS191168B2 (xx)
DE (1) DE2555405A1 (xx)
DK (1) DK149775B (xx)
FR (1) FR2293941A1 (xx)
GB (1) GB1535215A (xx)
HU (1) HU175575B (xx)
IE (1) IE42179B1 (xx)
LU (1) LU73957A1 (xx)
NL (1) NL7514322A (xx)
SE (1) SE435513B (xx)
SU (1) SU581873A3 (xx)
YU (1) YU306475A (xx)
ZA (1) ZA757652B (xx)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2860513D1 (en) * 1977-06-24 1981-04-09 Scherico Ltd Process for preparing aminoglycoside derivatives, novel derivatives obtained and pharmaceutical compositions containing such derivatives
CN101868472B (zh) 2007-11-21 2013-05-29 尔察祯有限公司 抗菌性氨基糖苷类似物
WO2010132765A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132759A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of dibekacin
WO2010132757A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132768A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of sisomicin
WO2010132760A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of tobramycin
CN103228282A (zh) 2010-09-13 2013-07-31 苏黎世大学 细菌感染性疾病的治疗
WO2018004993A1 (en) 2016-07-01 2018-01-04 Res Usa, Llc Reduction of greenhouse gas emission
US9981896B2 (en) 2016-07-01 2018-05-29 Res Usa, Llc Conversion of methane to dimethyl ether
WO2018004994A1 (en) 2016-07-01 2018-01-04 Res Usa, Llc Fluidized bed membrane reactor

Also Published As

Publication number Publication date
YU306475A (en) 1982-05-31
DK551075A (da) 1976-06-10
GB1535215A (en) 1978-12-13
FR2293941B1 (xx) 1978-11-10
ZA757652B (en) 1976-11-24
SE435513B (sv) 1984-10-01
LU73957A1 (xx) 1976-11-11
HU175575B (hu) 1980-09-28
SU581873A3 (ru) 1977-11-25
JPS51105036A (en) 1976-09-17
BE836292A (fr) 1976-06-04
CS191168B2 (en) 1979-06-29
SE7513804L (sv) 1976-06-10
FR2293941A1 (fr) 1976-07-09
CA1052780A (en) 1979-04-17
IE42179L (en) 1976-06-09
AU8688275A (en) 1977-06-02
IE42179B1 (en) 1980-06-18
DE2555405A1 (de) 1976-06-10
DK149775B (da) 1986-09-29
NL7514322A (nl) 1976-06-11

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