BE876732A - Nouveaux aminothiazoles et composition pharmaceutique les contenant - Google Patents
Nouveaux aminothiazoles et composition pharmaceutique les contenantInfo
- Publication number
- BE876732A BE876732A BE0/195534A BE195534A BE876732A BE 876732 A BE876732 A BE 876732A BE 0/195534 A BE0/195534 A BE 0/195534A BE 195534 A BE195534 A BE 195534A BE 876732 A BE876732 A BE 876732A
- Authority
- BE
- Belgium
- Prior art keywords
- aminothiazoles
- new
- pharmaceutical composition
- composition containing
- pharmaceutical
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
-
- F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
- F16—ENGINEERING ELEMENTS AND UNITS; GENERAL MEASURES FOR PRODUCING AND MAINTAINING EFFECTIVE FUNCTIONING OF MACHINES OR INSTALLATIONS; THERMAL INSULATION IN GENERAL
- F16B—DEVICES FOR FASTENING OR SECURING CONSTRUCTIONAL ELEMENTS OR MACHINE PARTS TOGETHER, e.g. NAILS, BOLTS, CIRCLIPS, CLAMPS, CLIPS OR WEDGES; JOINTS OR JOINTING
- F16B15/00—Nails; Staples
- F16B15/0023—Nail plates
- F16B2015/0076—Nail plates with provisions for additional fastening means, e.g. hooks, holes for separate screws or nails, adhesive
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Immunology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US91183078A | 1978-06-02 | 1978-06-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE876732A true BE876732A (fr) | 1979-12-03 |
Family
ID=25430923
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/195534A BE876732A (fr) | 1978-06-02 | 1979-06-01 | Nouveaux aminothiazoles et composition pharmaceutique les contenant |
Country Status (36)
Country | Link |
---|---|
JP (1) | JPS5936988B2 (fr) |
AR (1) | AR226285A1 (fr) |
AT (1) | AT373248B (fr) |
AU (1) | AU511242B2 (fr) |
BE (1) | BE876732A (fr) |
CA (1) | CA1117949A (fr) |
CH (1) | CH639653A5 (fr) |
CS (1) | CS216927B2 (fr) |
DD (1) | DD144055A5 (fr) |
DE (1) | DE2922523C2 (fr) |
DK (1) | DK150068C (fr) |
EG (1) | EG14354A (fr) |
ES (1) | ES481220A1 (fr) |
FI (1) | FI68820C (fr) |
FR (1) | FR2427333A1 (fr) |
GB (1) | GB2022085B (fr) |
GR (1) | GR73142B (fr) |
HK (1) | HK66487A (fr) |
HU (1) | HU180045B (fr) |
IE (1) | IE48426B1 (fr) |
IL (1) | IL57450A (fr) |
IT (1) | IT1121238B (fr) |
KE (1) | KE3459A (fr) |
LU (1) | LU81349A1 (fr) |
MY (1) | MY8500318A (fr) |
NL (1) | NL178421C (fr) |
NO (1) | NO150760C (fr) |
NZ (1) | NZ190623A (fr) |
PH (1) | PH17020A (fr) |
PL (1) | PL117515B1 (fr) |
PT (1) | PT69718A (fr) |
SE (1) | SE438333B (fr) |
SG (1) | SG56184G (fr) |
SU (1) | SU843746A3 (fr) |
YU (1) | YU40997B (fr) |
ZA (1) | ZA792729B (fr) |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0063575A4 (fr) * | 1980-10-24 | 1983-02-14 | Ronald Peter Hansen | System de reduction de la poussiere. |
WO1982002384A1 (fr) * | 1981-01-08 | 1982-07-22 | Sakano Isao | Derives de n-(4-phenyl-2-thiazolyl) carbamate, procede de preparation et composition medicinale les contenant |
JPS57136579A (en) * | 1981-01-21 | 1982-08-23 | Mitsui Toatsu Chem Inc | Thiazolylurea derivative, its preparation, and pharmaceutical composition containing the same |
JPS57116067A (en) * | 1981-01-12 | 1982-07-19 | Sankyo Kagaku Kk | Novel 8-quinolinesulfonyl derivative, its synthesis and use |
DE3273781D1 (en) * | 1981-01-13 | 1986-11-20 | Mitsui Toatsu Chemicals | Novel thiazole compounds, process for their preparation, and medicinal composition containing same |
WO1982002386A1 (fr) * | 1981-01-13 | 1982-07-22 | Sakano Isao | Derives d'aminothiazoles, procede de preparation et composition medicinale les contenant |
JPS57154175A (en) * | 1981-03-16 | 1982-09-22 | Mitsui Toatsu Chem Inc | 2-thiazoleamine derivative, its preparation, and drug composition comprising it |
DE3227329A1 (de) * | 1982-07-22 | 1984-01-26 | Basf Ag, 6700 Ludwigshafen | Verfahren zur herstellung von 2-n,n-disubstituierten aminothiazolen |
WO1986003203A1 (fr) * | 1984-11-22 | 1986-06-05 | Yoshitomi Pharmaceutical Industries, Ltd. | Derives de thienylthiazole |
FR2581063B1 (fr) * | 1985-04-30 | 1987-07-17 | Chauvin Blache Lab | Amino-2 thiazoles n-substitues, leur procede de preparation et leur application en therapeutique |
JPS63152368A (ja) * | 1986-06-03 | 1988-06-24 | Sumitomo Pharmaceut Co Ltd | 新規なアミノアゾ−ル誘導体およびその酸付加塩 |
JPH075579B2 (ja) * | 1986-09-01 | 1995-01-25 | 吉富製薬株式会社 | アミノチアゾ−ル化合物 |
JPH0753666B2 (ja) * | 1987-09-14 | 1995-06-07 | 久光製薬株式会社 | 置換ジフェニルチアゾール誘導体からなる抗炎症剤 |
DE69031624T2 (de) * | 1989-08-10 | 1998-05-14 | Commw Scient Ind Res Org | Verfahren zur herstellung von einer elektrosuspension von mikropartikeln |
DE69132293D1 (de) * | 1991-03-07 | 2000-08-10 | Hisamitsu Pharmaceutical Co | Diphenylthiazolderivate mit antiinflammatorischer aktivität |
FR2692893B1 (fr) * | 1992-06-24 | 1994-09-02 | Sanofi Elf | Dérivés alkylamino ramifiés du thiazole, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent. |
WO1996003392A1 (fr) * | 1994-07-27 | 1996-02-08 | G.D. Searle & Co. | Thiazoles substitues destines au traitement de l'inflammation |
FR2754258B1 (fr) | 1996-10-08 | 1998-12-31 | Sanofi Sa | Derives d'aminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
WO2001064674A1 (fr) | 2000-03-01 | 2001-09-07 | Janssen Pharmaceutica N.V. | Derives de thiazolyle 2,4-disubstitue |
EP1423113A4 (fr) * | 2001-08-13 | 2007-04-18 | Phenex Pharmaceuticals Ag | Composes de liaison au recepteur nucleaire nr1h4 |
WO2003027095A1 (fr) * | 2001-09-26 | 2003-04-03 | Bayer Pharmaceuticals Corporation | 3-pyridyl tetrazoles substitues en tant qu'inhibiteurs de la lyase c17,20 de la steroide |
BR0306811A (pt) | 2002-01-11 | 2004-10-26 | Sankyo Co | Composto, éster farmacologicamente aceitável do mesmo, composição farmacêutica e métodos para prevenção ou tratamento de doenças autoimunes, da artrite reumatóide e da rejeição causada pelo transplante de vários órgãos em um mamìfero |
EP1555264A1 (fr) * | 2004-01-15 | 2005-07-20 | Sireen AG | Hétérocycles à cinq chaínons comme inhibiteurs de la famille des SRC proteines kinases |
AU2005215320B2 (en) | 2004-02-24 | 2008-04-17 | Sankyo Company, Limited | Amino alcohol compound |
AU2006244203B2 (en) * | 2005-05-09 | 2012-05-03 | Achillion Pharmaceuticals, Inc. | Thiazole compounds and methods of use |
CA2636077C (fr) | 2006-01-18 | 2012-01-03 | Amgen Inc. | Composes thiazole et procedes d'utilisation |
CA2692713A1 (fr) | 2007-07-17 | 2009-01-22 | Amgen Inc. | Modulateurs heterocycliques de pkb |
CA2693473A1 (fr) | 2007-07-17 | 2009-01-22 | Amgen Inc. | Thiadiazoles modulateurs de l'activite de pkb |
WO2012170951A2 (fr) * | 2011-06-10 | 2012-12-13 | Calcimedica, Inc. | Composés modulant le calcium intracellulaire |
US20120316182A1 (en) | 2011-06-10 | 2012-12-13 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
WO2013059677A1 (fr) | 2011-10-19 | 2013-04-25 | Calcimedica, Inc. | Composés qui modulent le calcium intracellulaire |
CN110590785B (zh) * | 2019-09-23 | 2021-02-02 | 武汉大学 | 一种氨基噻唑类化合物及其制备方法与抗肠道病毒71型的应用 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3458526A (en) * | 1966-09-26 | 1969-07-29 | Upjohn Co | Certain 2-amino-4,5-bis(p-methoxyphenyl)thiazoles |
-
1979
- 1979-04-30 DK DK177679A patent/DK150068C/da not_active IP Right Cessation
- 1979-05-23 GB GB7917872A patent/GB2022085B/en not_active Expired
- 1979-05-29 CH CH501679A patent/CH639653A5/fr not_active IP Right Cessation
- 1979-05-30 CS CS793728A patent/CS216927B2/cs unknown
- 1979-05-30 EG EG333/79A patent/EG14354A/xx active
- 1979-05-31 SE SE7904798A patent/SE438333B/sv not_active IP Right Cessation
- 1979-05-31 CA CA000328805A patent/CA1117949A/fr not_active Expired
- 1979-05-31 YU YU1288/79A patent/YU40997B/xx unknown
- 1979-05-31 LU LU81349A patent/LU81349A1/fr unknown
- 1979-05-31 PH PH22588A patent/PH17020A/en unknown
- 1979-05-31 SU SU792773929A patent/SU843746A3/ru active
- 1979-05-31 HU HU79PI679A patent/HU180045B/hu not_active IP Right Cessation
- 1979-05-31 AU AU47634/79A patent/AU511242B2/en not_active Ceased
- 1979-05-31 IL IL57450A patent/IL57450A/xx unknown
- 1979-06-01 AT AT0401679A patent/AT373248B/de not_active IP Right Cessation
- 1979-06-01 IT IT23228/79A patent/IT1121238B/it active
- 1979-06-01 NL NLAANVRAGE7904337,A patent/NL178421C/xx not_active IP Right Cessation
- 1979-06-01 ZA ZA792729A patent/ZA792729B/xx unknown
- 1979-06-01 JP JP54068781A patent/JPS5936988B2/ja not_active Expired
- 1979-06-01 DD DD79213371A patent/DD144055A5/de not_active IP Right Cessation
- 1979-06-01 FR FR7914164A patent/FR2427333A1/fr active Granted
- 1979-06-01 GR GR59240A patent/GR73142B/el unknown
- 1979-06-01 PL PL1979216030A patent/PL117515B1/pl unknown
- 1979-06-01 ES ES481220A patent/ES481220A1/es not_active Expired
- 1979-06-01 FI FI791754A patent/FI68820C/fi not_active IP Right Cessation
- 1979-06-01 AR AR276782A patent/AR226285A1/es active
- 1979-06-01 BE BE0/195534A patent/BE876732A/fr not_active IP Right Cessation
- 1979-06-01 NZ NZ190623A patent/NZ190623A/en unknown
- 1979-06-01 DE DE2922523A patent/DE2922523C2/de not_active Expired
- 1979-06-01 PT PT69718A patent/PT69718A/pt unknown
- 1979-06-01 NO NO791831A patent/NO150760C/no unknown
- 1979-08-08 IE IE1069/79A patent/IE48426B1/en unknown
-
1984
- 1984-08-13 SG SG561/84A patent/SG56184G/en unknown
- 1984-09-24 KE KE3459A patent/KE3459A/xx unknown
-
1985
- 1985-12-30 MY MY318/85A patent/MY8500318A/xx unknown
-
1987
- 1987-09-17 HK HK664/87A patent/HK66487A/xx unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: PFIZER INC. Effective date: 19930630 |