DK177679A - Fremgangsmaade til fremstilling af hidtil ukendte aminothiazoler - Google Patents

Fremgangsmaade til fremstilling af hidtil ukendte aminothiazoler

Info

Publication number
DK177679A
DK177679A DK177679A DK177679A DK177679A DK 177679 A DK177679 A DK 177679A DK 177679 A DK177679 A DK 177679A DK 177679 A DK177679 A DK 177679A DK 177679 A DK177679 A DK 177679A
Authority
DK
Denmark
Prior art keywords
aminothiazoles
procedure
preparation
now unknown
unknown
Prior art date
Application number
DK177679A
Other languages
English (en)
Other versions
DK150068B (da
DK150068C (da
Inventor
J G Lombardino
J S Bindra
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK177679A publication Critical patent/DK177679A/da
Publication of DK150068B publication Critical patent/DK150068B/da
Application granted granted Critical
Publication of DK150068C publication Critical patent/DK150068C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/42Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
    • FMECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F16ENGINEERING ELEMENTS AND UNITS; GENERAL MEASURES FOR PRODUCING AND MAINTAINING EFFECTIVE FUNCTIONING OF MACHINES OR INSTALLATIONS; THERMAL INSULATION IN GENERAL
    • F16BDEVICES FOR FASTENING OR SECURING CONSTRUCTIONAL ELEMENTS OR MACHINE PARTS TOGETHER, e.g. NAILS, BOLTS, CIRCLIPS, CLAMPS, CLIPS OR WEDGES; JOINTS OR JOINTING
    • F16B15/00Nails; Staples
    • F16B15/0023Nail plates
    • F16B2015/0076Nail plates with provisions for additional fastening means, e.g. hooks, holes for separate screws or nails, adhesive

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK177679A 1978-06-02 1979-04-30 Analogifremgangsmaade til fremstilling af aminothiazoler DK150068C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US91183078A 1978-06-02 1978-06-02
US91183078 1978-06-02

Publications (3)

Publication Number Publication Date
DK177679A true DK177679A (da) 1979-12-03
DK150068B DK150068B (da) 1986-12-01
DK150068C DK150068C (da) 1987-06-29

Family

ID=25430923

Family Applications (1)

Application Number Title Priority Date Filing Date
DK177679A DK150068C (da) 1978-06-02 1979-04-30 Analogifremgangsmaade til fremstilling af aminothiazoler

Country Status (36)

Country Link
JP (1) JPS5936988B2 (da)
AR (1) AR226285A1 (da)
AT (1) AT373248B (da)
AU (1) AU511242B2 (da)
BE (1) BE876732A (da)
CA (1) CA1117949A (da)
CH (1) CH639653A5 (da)
CS (1) CS216927B2 (da)
DD (1) DD144055A5 (da)
DE (1) DE2922523C2 (da)
DK (1) DK150068C (da)
EG (1) EG14354A (da)
ES (1) ES481220A1 (da)
FI (1) FI68820C (da)
FR (1) FR2427333A1 (da)
GB (1) GB2022085B (da)
GR (1) GR73142B (da)
HK (1) HK66487A (da)
HU (1) HU180045B (da)
IE (1) IE48426B1 (da)
IL (1) IL57450A (da)
IT (1) IT1121238B (da)
KE (1) KE3459A (da)
LU (1) LU81349A1 (da)
MY (1) MY8500318A (da)
NL (1) NL178421C (da)
NO (1) NO150760C (da)
NZ (1) NZ190623A (da)
PH (1) PH17020A (da)
PL (1) PL117515B1 (da)
PT (1) PT69718A (da)
SE (1) SE438333B (da)
SG (1) SG56184G (da)
SU (1) SU843746A3 (da)
YU (1) YU40997B (da)
ZA (1) ZA792729B (da)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1982001481A1 (en) * 1980-10-24 1982-05-13 Ronald P Hansen Dust mitigation system
JPS57136579A (en) * 1981-01-21 1982-08-23 Mitsui Toatsu Chem Inc Thiazolylurea derivative, its preparation, and pharmaceutical composition containing the same
WO1982002384A1 (en) * 1981-01-08 1982-07-22 Sakano Isao Their preparation,and medicinal composition containing same
JPS57116067A (en) * 1981-01-12 1982-07-19 Sankyo Kagaku Kk Novel 8-quinolinesulfonyl derivative, its synthesis and use
EP0069154B1 (en) * 1981-01-13 1986-10-15 Mitsui Toatsu Kagaku Kabushiki Kaisha Novel thiazole compounds, process for their preparation, and medicinal composition containing same
WO1982002386A1 (en) * 1981-01-13 1982-07-22 Sakano Isao Aminothiazole derivatives,process for their preparation,and medicinal composition containing same
JPS57154175A (en) * 1981-03-16 1982-09-22 Mitsui Toatsu Chem Inc 2-thiazoleamine derivative, its preparation, and drug composition comprising it
DE3227329A1 (de) * 1982-07-22 1984-01-26 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von 2-n,n-disubstituierten aminothiazolen
WO1986003203A1 (en) * 1984-11-22 1986-06-05 Yoshitomi Pharmaceutical Industries, Ltd. Thienylthiazole derivatives
FR2581063B1 (fr) * 1985-04-30 1987-07-17 Chauvin Blache Lab Amino-2 thiazoles n-substitues, leur procede de preparation et leur application en therapeutique
JPS63152368A (ja) * 1986-06-03 1988-06-24 Sumitomo Pharmaceut Co Ltd 新規なアミノアゾ−ル誘導体およびその酸付加塩
JPH075579B2 (ja) * 1986-09-01 1995-01-25 吉富製薬株式会社 アミノチアゾ−ル化合物
JPH0753666B2 (ja) * 1987-09-14 1995-06-07 久光製薬株式会社 置換ジフェニルチアゾール誘導体からなる抗炎症剤
EP0486543B1 (en) * 1989-08-10 1997-10-22 Commonwealth Scientific And Industrial Research Organisation Method for producing an electrosuspension of micronised particles
ATE194338T1 (de) * 1991-03-07 2000-07-15 Hisamitsu Pharmaceutical Co Diphenylthiazolderivate mit antiinflammatorischer aktivität
FR2692893B1 (fr) * 1992-06-24 1994-09-02 Sanofi Elf Dérivés alkylamino ramifiés du thiazole, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent.
CA2195847A1 (en) * 1994-07-27 1996-02-08 John J. Talley Substituted thiazoles for the treatment of inflammation
FR2754258B1 (fr) 1996-10-08 1998-12-31 Sanofi Sa Derives d'aminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant
ES2317889T3 (es) 2000-03-01 2009-05-01 Janssen Pharmaceutica Nv Derivados de tiazolilo 2,4-disustituido.
EP1423113A4 (en) * 2001-08-13 2007-04-18 Phenex Pharmaceuticals Ag NR1H4 NUCLEAR RECEPTOR BINDING COMPOUNDS
WO2003027094A2 (en) * 2001-09-26 2003-04-03 Bayer Pharmaceuticals Corporation Substituted 3-pyridyl indoles and indazoles as c17,20 lyase inhibitors
KR100836547B1 (ko) 2002-01-11 2008-06-10 상꾜 가부시키가이샤 아미노 알코올 유도체 또는 포스폰산 유도체 및 이들을함유하는 의약 조성물
EP1555264A1 (en) * 2004-01-15 2005-07-20 Sireen AG Five-membered heterocyclic compounds as inhibitors of SRC family protein kinase.
WO2005079788A1 (ja) 2004-02-24 2005-09-01 Sankyo Company, Limited アミノアルコール化合物
US8088806B2 (en) * 2005-05-09 2012-01-03 Achillion Pharmaceuticals, Inc. Thiazole compounds and methods of use
KR20080091369A (ko) 2006-01-18 2008-10-10 암젠 인크 단백질 키나제 b (pkb) 억제제로서 티아졸 화합물
AU2008276521B2 (en) 2007-07-17 2011-11-03 Amgen Inc. Heterocyclic modulators of PKB
CA2693473A1 (en) 2007-07-17 2009-01-22 Amgen Inc. Thiadiazole modulators of pkb
US20130143927A1 (en) * 2011-06-10 2013-06-06 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2012170931A2 (en) 2011-06-10 2012-12-13 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9856240B2 (en) 2011-10-19 2018-01-02 Calcimedica, Inc. Compounds that modulate intracellular calcium
CN110590785B (zh) * 2019-09-23 2021-02-02 武汉大学 一种氨基噻唑类化合物及其制备方法与抗肠道病毒71型的应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3458526A (en) * 1966-09-26 1969-07-29 Upjohn Co Certain 2-amino-4,5-bis(p-methoxyphenyl)thiazoles

Also Published As

Publication number Publication date
NZ190623A (en) 1984-07-06
MY8500318A (en) 1985-12-31
AU4763479A (en) 1979-12-06
SE438333B (sv) 1985-04-15
NO150760B (no) 1984-09-03
NO150760C (no) 1984-12-12
KE3459A (en) 1984-10-12
NL7904337A (nl) 1979-12-04
FR2427333A1 (fr) 1979-12-28
IE48426B1 (en) 1985-01-23
NO791831L (no) 1979-12-04
GB2022085B (en) 1983-01-12
SE7904798L (sv) 1979-12-03
SU843746A3 (ru) 1981-06-30
AR226285A1 (es) 1982-06-30
PL216030A1 (da) 1980-03-10
FI68820C (fi) 1985-11-11
IT1121238B (it) 1986-03-26
ES481220A1 (es) 1980-09-01
LU81349A1 (fr) 1979-12-07
IL57450A0 (en) 1979-09-30
DE2922523A1 (de) 1979-12-06
CS216927B2 (en) 1982-12-31
FI791754A (fi) 1979-11-26
PH17020A (en) 1984-05-11
ATA401679A (de) 1983-05-15
CA1117949A (en) 1982-02-09
DD144055A5 (de) 1980-09-24
CH639653A5 (fr) 1983-11-30
DK150068B (da) 1986-12-01
NL178421B (nl) 1985-10-16
PL117515B1 (en) 1981-08-31
PT69718A (en) 1979-07-01
AU511242B2 (en) 1980-08-07
BE876732A (fr) 1979-12-03
EG14354A (en) 1984-06-30
JPS5936988B2 (ja) 1984-09-06
NL178421C (nl) 1986-03-17
JPS54160369A (en) 1979-12-19
FR2427333B1 (da) 1983-05-20
HK66487A (en) 1987-09-25
FI68820B (fi) 1985-07-31
IE791069L (en) 1979-12-02
ZA792729B (en) 1981-03-25
YU40997B (en) 1986-10-31
DK150068C (da) 1987-06-29
IL57450A (en) 1982-11-30
GB2022085A (en) 1979-12-12
HU180045B (en) 1983-01-28
IT7923228A0 (it) 1979-06-01
DE2922523C2 (de) 1982-10-21
YU128879A (en) 1982-10-31
AT373248B (de) 1983-12-27
SG56184G (en) 1985-03-08
GR73142B (da) 1984-02-09

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Legal Events

Date Code Title Description
PBP Patent lapsed