AU511242B2 - Novel aminothiazoles - Google Patents

Novel aminothiazoles

Info

Publication number
AU511242B2
AU511242B2 AU47634/79A AU4763479A AU511242B2 AU 511242 B2 AU511242 B2 AU 511242B2 AU 47634/79 A AU47634/79 A AU 47634/79A AU 4763479 A AU4763479 A AU 4763479A AU 511242 B2 AU511242 B2 AU 511242B2
Authority
AU
Australia
Prior art keywords
aminothiazoles
novel
novel aminothiazoles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU47634/79A
Other languages
English (en)
Other versions
AU4763479A (en
Inventor
Jasjit Singh Bindra
Joseph George Lombardino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of AU4763479A publication Critical patent/AU4763479A/en
Application granted granted Critical
Publication of AU511242B2 publication Critical patent/AU511242B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
    • F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F16—ENGINEERING ELEMENTS AND UNITS; GENERAL MEASURES FOR PRODUCING AND MAINTAINING EFFECTIVE FUNCTIONING OF MACHINES OR INSTALLATIONS; THERMAL INSULATION IN GENERAL
    • F16B—DEVICES FOR FASTENING OR SECURING CONSTRUCTIONAL ELEMENTS OR MACHINE PARTS TOGETHER, e.g. NAILS, BOLTS, CIRCLIPS, CLAMPS, CLIPS OR WEDGES; JOINTS OR JOINTING
    • F16B15/00—Nails; Staples
    • F16B15/0023—Nail plates
    • F16B2015/0076—Nail plates with provisions for additional fastening means, e.g. hooks, holes for separate screws or nails, adhesive

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU47634/79A 1978-06-02 1979-05-31 Novel aminothiazoles Ceased AU511242B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US91183078A 1978-06-02 1978-06-02
US911830 1978-06-02

Publications (2)

Publication Number Publication Date
AU4763479A AU4763479A (en) 1979-12-06
AU511242B2 true AU511242B2 (en) 1980-08-07

Family

ID=25430923

Family Applications (1)

Application Number Title Priority Date Filing Date
AU47634/79A Ceased AU511242B2 (en) 1978-06-02 1979-05-31 Novel aminothiazoles

Country Status (36)

Country Link
JP (1) JPS5936988B2 (da)
AR (1) AR226285A1 (da)
AT (1) AT373248B (da)
AU (1) AU511242B2 (da)
BE (1) BE876732A (da)
CA (1) CA1117949A (da)
CH (1) CH639653A5 (da)
CS (1) CS216927B2 (da)
DD (1) DD144055A5 (da)
DE (1) DE2922523C2 (da)
DK (1) DK150068C (da)
EG (1) EG14354A (da)
ES (1) ES481220A1 (da)
FI (1) FI68820C (da)
FR (1) FR2427333A1 (da)
GB (1) GB2022085B (da)
GR (1) GR73142B (da)
HK (1) HK66487A (da)
HU (1) HU180045B (da)
IE (1) IE48426B1 (da)
IL (1) IL57450A (da)
IT (1) IT1121238B (da)
KE (1) KE3459A (da)
LU (1) LU81349A1 (da)
MY (1) MY8500318A (da)
NL (1) NL178421C (da)
NO (1) NO150760C (da)
NZ (1) NZ190623A (da)
PH (1) PH17020A (da)
PL (1) PL117515B1 (da)
PT (1) PT69718A (da)
SE (1) SE438333B (da)
SG (1) SG56184G (da)
SU (1) SU843746A3 (da)
YU (1) YU40997B (da)
ZA (1) ZA792729B (da)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1982001481A1 (en) * 1980-10-24 1982-05-13 Ronald P Hansen Dust mitigation system
WO1991002394A1 (en) * 1989-08-10 1991-02-21 Commonwealth Scientific And Industrial Research Organisation Producing electrosuspensions

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57136579A (en) * 1981-01-21 1982-08-23 Mitsui Toatsu Chem Inc Thiazolylurea derivative, its preparation, and pharmaceutical composition containing the same
WO1982002384A1 (en) * 1981-01-08 1982-07-22 Sakano Isao Their preparation,and medicinal composition containing same
JPS57116067A (en) * 1981-01-12 1982-07-19 Sankyo Kagaku Kk Novel 8-quinolinesulfonyl derivative, its synthesis and use
EP0069154B1 (en) * 1981-01-13 1986-10-15 Mitsui Toatsu Kagaku Kabushiki Kaisha Novel thiazole compounds, process for their preparation, and medicinal composition containing same
WO1982002386A1 (en) * 1981-01-13 1982-07-22 Sakano Isao Aminothiazole derivatives,process for their preparation,and medicinal composition containing same
JPS57154175A (en) * 1981-03-16 1982-09-22 Mitsui Toatsu Chem Inc 2-thiazoleamine derivative, its preparation, and drug composition comprising it
DE3227329A1 (de) * 1982-07-22 1984-01-26 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von 2-n,n-disubstituierten aminothiazolen
WO1986003203A1 (en) * 1984-11-22 1986-06-05 Yoshitomi Pharmaceutical Industries, Ltd. Thienylthiazole derivatives
FR2581063B1 (fr) * 1985-04-30 1987-07-17 Chauvin Blache Lab Amino-2 thiazoles n-substitues, leur procede de preparation et leur application en therapeutique
JPS63152368A (ja) * 1986-06-03 1988-06-24 Sumitomo Pharmaceut Co Ltd 新規なアミノアゾ−ル誘導体およびその酸付加塩
JPH075579B2 (ja) * 1986-09-01 1995-01-25 吉富製薬株式会社 アミノチアゾ−ル化合物
JPH0753666B2 (ja) * 1987-09-14 1995-06-07 久光製薬株式会社 置換ジフェニルチアゾール誘導体からなる抗炎症剤
ATE194338T1 (de) * 1991-03-07 2000-07-15 Hisamitsu Pharmaceutical Co Diphenylthiazolderivate mit antiinflammatorischer aktivität
FR2692893B1 (fr) * 1992-06-24 1994-09-02 Sanofi Elf Dérivés alkylamino ramifiés du thiazole, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent.
CA2195847A1 (en) * 1994-07-27 1996-02-08 John J. Talley Substituted thiazoles for the treatment of inflammation
FR2754258B1 (fr) 1996-10-08 1998-12-31 Sanofi Sa Derives d'aminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant
ES2317889T3 (es) 2000-03-01 2009-05-01 Janssen Pharmaceutica Nv Derivados de tiazolilo 2,4-disustituido.
EP1423113A4 (en) * 2001-08-13 2007-04-18 Phenex Pharmaceuticals Ag NR1H4 NUCLEAR RECEPTOR BINDING COMPOUNDS
WO2003027094A2 (en) * 2001-09-26 2003-04-03 Bayer Pharmaceuticals Corporation Substituted 3-pyridyl indoles and indazoles as c17,20 lyase inhibitors
KR100836547B1 (ko) 2002-01-11 2008-06-10 상꾜 가부시키가이샤 아미노 알코올 유도체 또는 포스폰산 유도체 및 이들을함유하는 의약 조성물
EP1555264A1 (en) * 2004-01-15 2005-07-20 Sireen AG Five-membered heterocyclic compounds as inhibitors of SRC family protein kinase.
WO2005079788A1 (ja) 2004-02-24 2005-09-01 Sankyo Company, Limited アミノアルコール化合物
US8088806B2 (en) * 2005-05-09 2012-01-03 Achillion Pharmaceuticals, Inc. Thiazole compounds and methods of use
KR20080091369A (ko) 2006-01-18 2008-10-10 암젠 인크 단백질 키나제 ｂ （ｐｋｂ） 억제제로서 티아졸 화합물
AU2008276521B2 (en) 2007-07-17 2011-11-03 Amgen Inc. Heterocyclic modulators of PKB
CA2693473A1 (en) 2007-07-17 2009-01-22 Amgen Inc. Thiadiazole modulators of pkb
US20130143927A1 (en) * 2011-06-10 2013-06-06 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2012170931A2 (en) 2011-06-10 2012-12-13 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9856240B2 (en) 2011-10-19 2018-01-02 Calcimedica, Inc. Compounds that modulate intracellular calcium
CN110590785B (zh) * 2019-09-23 2021-02-02 武汉大学 一种氨基噻唑类化合物及其制备方法与抗肠道病毒71型的应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3458526A (en) * 1966-09-26 1969-07-29 Upjohn Co Certain 2-amino-4,5-bis(p-methoxyphenyl)thiazoles

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1982001481A1 (en) * 1980-10-24 1982-05-13 Ronald P Hansen Dust mitigation system
WO1991002394A1 (en) * 1989-08-10 1991-02-21 Commonwealth Scientific And Industrial Research Organisation Producing electrosuspensions

Also Published As

Publication number Publication date
NZ190623A (en) 1984-07-06
MY8500318A (en) 1985-12-31
AU4763479A (en) 1979-12-06
SE438333B (sv) 1985-04-15
NO150760B (no) 1984-09-03
NO150760C (no) 1984-12-12
KE3459A (en) 1984-10-12
NL7904337A (nl) 1979-12-04
FR2427333A1 (fr) 1979-12-28
IE48426B1 (en) 1985-01-23
NO791831L (no) 1979-12-04
GB2022085B (en) 1983-01-12
SE7904798L (sv) 1979-12-03
SU843746A3 (ru) 1981-06-30
AR226285A1 (es) 1982-06-30
PL216030A1 (da) 1980-03-10
FI68820C (fi) 1985-11-11
IT1121238B (it) 1986-03-26
ES481220A1 (es) 1980-09-01
LU81349A1 (fr) 1979-12-07
IL57450A0 (en) 1979-09-30
DE2922523A1 (de) 1979-12-06
CS216927B2 (en) 1982-12-31
FI791754A (fi) 1979-11-26
PH17020A (en) 1984-05-11
ATA401679A (de) 1983-05-15
CA1117949A (en) 1982-02-09
DD144055A5 (de) 1980-09-24
CH639653A5 (fr) 1983-11-30
DK150068B (da) 1986-12-01
NL178421B (nl) 1985-10-16
PL117515B1 (en) 1981-08-31
PT69718A (en) 1979-07-01
BE876732A (fr) 1979-12-03
EG14354A (en) 1984-06-30
JPS5936988B2 (ja) 1984-09-06
NL178421C (nl) 1986-03-17
JPS54160369A (en) 1979-12-19
FR2427333B1 (da) 1983-05-20
HK66487A (en) 1987-09-25
FI68820B (fi) 1985-07-31
IE791069L (en) 1979-12-02
ZA792729B (en) 1981-03-25
DK177679A (da) 1979-12-03
YU40997B (en) 1986-10-31
DK150068C (da) 1987-06-29
IL57450A (en) 1982-11-30
GB2022085A (en) 1979-12-12
HU180045B (en) 1983-01-28
IT7923228A0 (it) 1979-06-01
DE2922523C2 (de) 1982-10-21
YU128879A (en) 1982-10-31
AT373248B (de) 1983-12-27
SG56184G (en) 1985-03-08
GR73142B (da) 1984-02-09

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