AU2014298051B2 - Novel quinazolinones as bromodomain inhibitors - Google Patents

Novel quinazolinones as bromodomain inhibitors Download PDF

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AU2014298051B2
AU2014298051B2 AU2014298051A AU2014298051A AU2014298051B2 AU 2014298051 B2 AU2014298051 B2 AU 2014298051B2 AU 2014298051 A AU2014298051 A AU 2014298051A AU 2014298051 A AU2014298051 A AU 2014298051A AU 2014298051 B2 AU2014298051 B2 AU 2014298051B2
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amino
cancer
mmol
dimethoxy
pyridin
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AU2014298051A1 (en
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Vladimir Khlebnikov
John Frederick Quinn
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Zenith Epigenetics Ltd
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Zenith Epigenetics Ltd
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    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
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AU2014298051A 2013-07-31 2014-07-30 Novel quinazolinones as bromodomain inhibitors Ceased AU2014298051B2 (en)

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US201361860403P 2013-07-31 2013-07-31
US61/860,403 2013-07-31
PCT/IB2014/002510 WO2015015318A2 (en) 2013-07-31 2014-07-30 Novel quinazolinones as bromodomain inhibitors

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AU2014298051A1 AU2014298051A1 (en) 2016-01-28
AU2014298051B2 true AU2014298051B2 (en) 2018-11-15

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US (2) US9855271B2 (enExample)
EP (1) EP3027604B1 (enExample)
JP (1) JP6542212B2 (enExample)
KR (1) KR20160038008A (enExample)
CN (1) CN105593224B (enExample)
AU (1) AU2014298051B2 (enExample)
CA (1) CA2919948C (enExample)
EA (1) EA201690087A1 (enExample)
IL (1) IL243479B (enExample)
WO (1) WO2015015318A2 (enExample)

Families Citing this family (60)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9073878B2 (en) 2012-11-21 2015-07-07 Zenith Epigenetics Corp. Cyclic amines as bromodomain inhibitors
WO2014080291A2 (en) 2012-11-21 2014-05-30 Rvx Therapeutics Inc. Biaryl derivatives as bromodomain inhibitors
US9271978B2 (en) 2012-12-21 2016-03-01 Zenith Epigenetics Corp. Heterocyclic compounds as bromodomain inhibitors
WO2014159837A1 (en) 2013-03-14 2014-10-02 Convergene Llc Methods and compositions for inhibition of bromodomain-containing proteins
SG11201510409QA (en) 2013-06-21 2016-01-28 Zenith Epigenetics Corp Novel bicyclic bromodomain inhibitors
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