AU2013290100A1 - Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk - Google Patents
Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk Download PDFInfo
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- AU2013290100A1 AU2013290100A1 AU2013290100A AU2013290100A AU2013290100A1 AU 2013290100 A1 AU2013290100 A1 AU 2013290100A1 AU 2013290100 A AU2013290100 A AU 2013290100A AU 2013290100 A AU2013290100 A AU 2013290100A AU 2013290100 A1 AU2013290100 A1 AU 2013290100A1
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- metformin
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- 239000003795 chemical substances by application Substances 0.000 title description 41
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- -1 biguanide compound Chemical class 0.000 claims abstract description 181
- 238000000034 method Methods 0.000 claims abstract description 107
- 239000013543 active substance Substances 0.000 claims abstract description 48
- 208000024172 Cardiovascular disease Diseases 0.000 claims abstract description 24
- 229940000425 combination drug Drugs 0.000 claims abstract description 9
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- 229960003105 metformin Drugs 0.000 claims description 158
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- 239000003112 inhibitor Substances 0.000 claims description 27
- XNCOSPRUTUOJCJ-UHFFFAOYSA-N Biguanide Chemical compound NC(N)=NC(N)=N XNCOSPRUTUOJCJ-UHFFFAOYSA-N 0.000 claims description 21
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13/547,022 | 2012-07-11 | ||
| US13/547,022 US8796338B2 (en) | 2011-01-07 | 2012-07-11 | Biguanide compositions and methods of treating metabolic disorders |
| US13/734,966 US9211263B2 (en) | 2012-01-06 | 2013-01-05 | Compositions and methods of treating metabolic disorders |
| US13/734,966 | 2013-01-05 | ||
| PCT/US2013/050142 WO2014011926A1 (en) | 2012-07-11 | 2013-07-11 | Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk |
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| AU2013290100A1 true AU2013290100A1 (en) | 2015-01-29 |
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| AU2013290100A Abandoned AU2013290100A1 (en) | 2012-07-11 | 2013-07-11 | Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk |
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| EP (1) | EP2872127A1 (enExample) |
| JP (2) | JP2015522080A (enExample) |
| CN (1) | CN104780915A (enExample) |
| AR (1) | AR091739A1 (enExample) |
| AU (1) | AU2013290100A1 (enExample) |
| CA (1) | CA2878625A1 (enExample) |
| HK (1) | HK1210825A1 (enExample) |
| IL (1) | IL236647A0 (enExample) |
| WO (1) | WO2014011926A1 (enExample) |
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| UY33937A (es) | 2011-03-07 | 2012-09-28 | Boehringer Ingelheim Int | Composiciones farmacéuticas que contienen inhibidores de dpp-4 y/o sglt-2 y metformina |
| US11813275B2 (en) | 2013-04-05 | 2023-11-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, methods for treating and uses thereof |
| CA2812519A1 (en) | 2013-04-05 | 2014-10-05 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, methods for treating and uses thereof |
| HK1213818A1 (zh) | 2013-04-05 | 2016-07-15 | 勃林格殷格翰国际有限公司 | 依帕列净的治疗用途 |
| ES2702174T3 (es) | 2013-04-05 | 2019-02-27 | Boehringer Ingelheim Int | Usos terapéuticos de empagliflozina |
| JP2016520564A (ja) | 2013-04-18 | 2016-07-14 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 医薬組成物、治療方法及びその使用 |
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| WO2012154009A2 (ko) | 2011-05-12 | 2012-11-15 | 한국화학연구원 | 티에노피리미딘 유도체, 이의 약학적으로 허용가능한 이의 제조방법 및 이를 유효성분으로 함유하는 당뇨 관련 질환의 또는 치료용 약학적 조성물 |
| WO2012170702A1 (en) | 2011-06-08 | 2012-12-13 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| EP2718288B1 (en) | 2011-06-09 | 2015-03-11 | Boehringer Ingelheim International GmbH | Substituted piperidines as gpr119 modulators for the treatment of metabolic disorders |
| JP2014159376A (ja) | 2011-06-17 | 2014-09-04 | Taisho Pharmaceutical Co Ltd | アザスピロアルカン化合物 |
| CA2841757A1 (en) | 2011-07-15 | 2013-01-24 | Etzer Darout | Gpr 119 modulators |
| WO2013055910A1 (en) | 2011-10-12 | 2013-04-18 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| CN102357088A (zh) * | 2011-10-26 | 2012-02-22 | 河北山姆士药业有限公司 | 盐酸二甲双胍肠溶片 |
-
2013
- 2013-07-11 AR ARP130102472 patent/AR091739A1/es unknown
- 2013-07-11 CA CA2878625A patent/CA2878625A1/en not_active Abandoned
- 2013-07-11 HK HK15111491.4A patent/HK1210825A1/xx unknown
- 2013-07-11 JP JP2015521822A patent/JP2015522080A/ja active Pending
- 2013-07-11 EP EP13739919.2A patent/EP2872127A1/en not_active Withdrawn
- 2013-07-11 AU AU2013290100A patent/AU2013290100A1/en not_active Abandoned
- 2013-07-11 CN CN201380046376.XA patent/CN104780915A/zh active Pending
- 2013-07-11 WO PCT/US2013/050142 patent/WO2014011926A1/en not_active Ceased
-
2015
- 2015-01-11 IL IL236647A patent/IL236647A0/en unknown
-
2018
- 2018-02-01 JP JP2018016141A patent/JP2018087214A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| WO2014011926A1 (en) | 2014-01-16 |
| AR091739A1 (es) | 2015-02-25 |
| EP2872127A1 (en) | 2015-05-20 |
| CN104780915A (zh) | 2015-07-15 |
| JP2018087214A (ja) | 2018-06-07 |
| HK1210825A1 (en) | 2016-05-06 |
| CA2878625A1 (en) | 2014-01-16 |
| JP2015522080A (ja) | 2015-08-03 |
| IL236647A0 (en) | 2015-02-26 |
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