AU2011290126B2 - Heterocyclic compound and use thereof - Google Patents

Heterocyclic compound and use thereof Download PDF

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Publication number
AU2011290126B2
AU2011290126B2 AU2011290126A AU2011290126A AU2011290126B2 AU 2011290126 B2 AU2011290126 B2 AU 2011290126B2 AU 2011290126 A AU2011290126 A AU 2011290126A AU 2011290126 A AU2011290126 A AU 2011290126A AU 2011290126 B2 AU2011290126 B2 AU 2011290126B2
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Australia
Prior art keywords
optionally substituted
halogen atom
alkyl
group
substituted
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AU2011290126A
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AU2011290126A1 (en
Inventor
Yasutomi Asano
Eiji Honda
Toshihiro Imaeda
Masakuni Kori
Michiyo Mochizuki
Shinji Nakamura
Masashi Toyofuku
Osamu Ujikawa
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Takeda Pharmaceutical Co Ltd
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Takeda Pharmaceutical Co Ltd
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Publication of AU2011290126A1 publication Critical patent/AU2011290126A1/en
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
AU2011290126A 2010-08-10 2011-08-09 Heterocyclic compound and use thereof Active AU2011290126B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2010179577 2010-08-10
JP2010-179577 2010-08-10
PCT/JP2011/068497 WO2012020848A1 (en) 2010-08-10 2011-08-09 Heterocyclic compound and use thereof

Publications (2)

Publication Number Publication Date
AU2011290126A1 AU2011290126A1 (en) 2013-03-07
AU2011290126B2 true AU2011290126B2 (en) 2016-01-07

Family

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AU2011290126A Active AU2011290126B2 (en) 2010-08-10 2011-08-09 Heterocyclic compound and use thereof

Country Status (39)

Country Link
US (11) US9150591B2 (OSRAM)
EP (1) EP2603513B1 (OSRAM)
JP (2) JP5788496B2 (OSRAM)
KR (1) KR101852215B1 (OSRAM)
CN (2) CN103180326B (OSRAM)
AR (1) AR082618A1 (OSRAM)
AU (1) AU2011290126B2 (OSRAM)
BR (1) BR112013002250B1 (OSRAM)
CA (1) CA2807460C (OSRAM)
CL (1) CL2013000380A1 (OSRAM)
CO (1) CO6680700A2 (OSRAM)
CR (1) CR20130066A (OSRAM)
CY (1) CY1123507T1 (OSRAM)
DK (1) DK2603513T3 (OSRAM)
DO (1) DOP2013000030A (OSRAM)
EA (1) EA022078B1 (OSRAM)
EC (1) ECSP13012478A (OSRAM)
ES (1) ES2793723T3 (OSRAM)
GE (1) GEP20156216B (OSRAM)
HR (1) HRP20200844T1 (OSRAM)
HU (1) HUE049460T2 (OSRAM)
IL (1) IL224452A (OSRAM)
LT (1) LT2603513T (OSRAM)
MA (1) MA34509B1 (OSRAM)
MX (1) MX349470B (OSRAM)
MY (1) MY165908A (OSRAM)
NZ (1) NZ607593A (OSRAM)
PE (1) PE20131116A1 (OSRAM)
PH (1) PH12013500247A1 (OSRAM)
PL (1) PL2603513T3 (OSRAM)
PT (1) PT2603513T (OSRAM)
RS (1) RS60311B1 (OSRAM)
SG (1) SG187656A1 (OSRAM)
SI (1) SI2603513T1 (OSRAM)
TW (1) TWI504604B (OSRAM)
UA (1) UA111594C2 (OSRAM)
UY (1) UY33551A (OSRAM)
WO (1) WO2012020848A1 (OSRAM)
ZA (1) ZA201301120B (OSRAM)

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EP3164386B1 (en) 2014-07-02 2020-10-07 FMC Corporation Piperidinone herbicides
SG11201702924WA (en) 2014-12-08 2017-05-30 Du Pont 3-oxo-3-(arylamino)propanoates, a process for their preparation, and their use in preparing pyrrolidinones
RU2710379C2 (ru) 2015-04-10 2019-12-26 ЭфЭмСи Корпорейшн Замещенные циклические амиды в качестве гербицидов
EP3288928B1 (en) 2015-04-27 2021-10-13 FMC Corporation Butyrolactones as herbicides
DK3288940T5 (da) 2015-04-29 2021-09-20 Janssen Pharmaceutica Nv Azabenzimidazoler og deres anvendelse som ampa-receptormodulatorer
WO2016176457A1 (en) * 2015-04-29 2016-11-03 Janssen Pharmaceutica Nv Imidazopyrazines and pyrazolopyrimidines and their use as ampa receptor modulators
CA2980643C (en) 2015-05-12 2023-10-17 E I Du Pont De Nemours And Company Aryl substituted bicyclic compounds as herbicides
JP6869192B2 (ja) 2015-05-29 2021-05-12 エフ エム シー コーポレーションFmc Corporation 除草剤としての置換環状アミド
RU2017142979A (ru) 2015-06-02 2019-07-15 ЭфЭмСи Корпорейшн Замещенные циклические амиды и их применение в качестве гербицидов
JP6937290B2 (ja) 2015-07-31 2021-09-22 エフ エム シー コーポレーションFmc Corporation 除草剤として有用な環状n−カルボキサミド化合物
CN107709342B (zh) * 2015-08-06 2021-09-03 豪夫迈·罗氏有限公司 制备乙酰半乳糖胺酸衍生物的方法
US20170181292A1 (en) * 2015-12-16 2017-06-22 Rohm And Haas Electronic Materials Llc Method for forming organic coating on nickel surface
CN105669731B (zh) * 2016-01-10 2017-06-30 沧州普瑞东方科技有限公司 一种4‑(4‑烷基环己氧基)苯硼酸的合成方法
CN110312712B (zh) 2016-12-21 2023-06-23 Fmc公司 硝酮除草剂
CN107892697B (zh) 2016-12-26 2020-11-03 郑州泰基鸿诺医药股份有限公司 一种[1,3]噻嗪-2-胺类化合物及应用,药物组合物
JP7201609B2 (ja) 2017-03-21 2023-01-10 エフ エム シー コーポレーション ピロリジノン及びこれらを調製するためのプロセス
US11919859B2 (en) 2017-03-21 2024-03-05 Fmc Corporation Herbicidal mixture, composition and method
AR111967A1 (es) 2017-05-30 2019-09-04 Fmc Corp Amidas herbicidas
AR111839A1 (es) 2017-05-30 2019-08-21 Fmc Corp Lactamas 3-sustituidas herbicidas
US11407748B2 (en) 2017-10-06 2022-08-09 Takeda Pharmaceutical Company Limited Substituted pyrido[1,2-a]pyrimidines and pyrazino[1,2-a]pyrimidines for enhancing AMPA receptor function
ES2971497T3 (es) 2017-10-06 2024-06-05 Takeda Pharmaceuticals Co Compuestos heterocíclicos
PH12022550597A1 (en) 2019-09-16 2024-03-04 Takeda Pharmaceuticals Co Azole-fused pyridazin-3(2h)-one derivatives
JP2023526249A (ja) * 2020-05-15 2023-06-21 武田薬品工業株式会社 うつ病の処置
CN113943294A (zh) * 2020-07-15 2022-01-18 成都海博为药业有限公司 一种作为btk抑制剂的化合物及其制备方法与用途
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Also Published As

Publication number Publication date
US9884875B2 (en) 2018-02-06
US20120077799A1 (en) 2012-03-29
KR20130138738A (ko) 2013-12-19
PE20131116A1 (es) 2013-10-24
HRP20200844T1 (hr) 2020-08-21
ES2793723T3 (es) 2020-11-16
CA2807460C (en) 2018-09-18
US20170022222A1 (en) 2017-01-26
NZ607593A (en) 2015-01-30
KR101852215B1 (ko) 2018-04-25
US11279713B2 (en) 2022-03-22
WO2012020848A8 (en) 2012-09-27
BR112013002250A2 (pt) 2016-05-24
EP2603513A1 (en) 2013-06-19
US20190263832A1 (en) 2019-08-29
JP5788496B2 (ja) 2015-09-30
EP2603513B1 (en) 2020-03-11
US20140080817A1 (en) 2014-03-20
MY165908A (en) 2018-05-18
PT2603513T (pt) 2020-06-08
US9150591B2 (en) 2015-10-06
AR082618A1 (es) 2012-12-19
US20240360156A1 (en) 2024-10-31
US8916551B2 (en) 2014-12-23
SI2603513T1 (sl) 2020-07-31
UA111594C2 (uk) 2016-05-25
US20150353578A1 (en) 2015-12-10
DOP2013000030A (es) 2013-03-15
LT2603513T (lt) 2020-05-25
US20200317692A1 (en) 2020-10-08
GEP20156216B (en) 2015-01-12
MX349470B (es) 2017-07-31
CA2807460A1 (en) 2012-02-16
ECSP13012478A (es) 2013-04-30
US20130184266A1 (en) 2013-07-18
JP2013535408A (ja) 2013-09-12
MA34509B1 (fr) 2013-09-02
EA022078B1 (ru) 2015-10-30
US9499568B2 (en) 2016-11-22
PH12013500247A1 (en) 2013-03-11
DK2603513T3 (da) 2020-06-15
CY1123507T1 (el) 2022-03-24
TWI504604B (zh) 2015-10-21
US8575154B2 (en) 2013-11-05
WO2012020848A1 (en) 2012-02-16
CL2013000380A1 (es) 2013-05-31
IL224452A (en) 2017-11-30
US10654874B2 (en) 2020-05-19
BR112013002250B1 (pt) 2020-10-27
RS60311B1 (sr) 2020-07-31
MX2013001614A (es) 2013-07-05
SG187656A1 (en) 2013-03-28
PL2603513T3 (pl) 2020-07-27
CN103180326A (zh) 2013-06-26
CO6680700A2 (es) 2013-05-31
UY33551A (es) 2012-03-30
CN104926837A (zh) 2015-09-23
EA201390222A1 (ru) 2013-08-30
CN103180326B (zh) 2015-06-10
US20130190291A1 (en) 2013-07-25
ZA201301120B (en) 2014-04-30
JP2016006080A (ja) 2016-01-14
HUE049460T2 (hu) 2020-09-28
AU2011290126A1 (en) 2013-03-07
US20150073137A1 (en) 2015-03-12
TW201217386A (en) 2012-05-01
US8778934B2 (en) 2014-07-15
JP6113789B2 (ja) 2017-04-12
US20180162875A1 (en) 2018-06-14
CR20130066A (es) 2013-05-03

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