AR068402A1 - Combinaciones de compuestos inhibidores de fosfoinositida 3-quinasa y agentes quimioterapeuticos y los metodos de uso - Google Patents

Combinaciones de compuestos inhibidores de fosfoinositida 3-quinasa y agentes quimioterapeuticos y los metodos de uso

Info

Publication number
AR068402A1
AR068402A1 ARP080103927A ARP080103927A AR068402A1 AR 068402 A1 AR068402 A1 AR 068402A1 AR P080103927 A ARP080103927 A AR P080103927A AR P080103927 A ARP080103927 A AR P080103927A AR 068402 A1 AR068402 A1 AR 068402A1
Authority
AR
Argentina
Prior art keywords
nr10r11
cr14r15
nr12c
alkyl
heteroaryl
Prior art date
Application number
ARP080103927A
Other languages
English (en)
Spanish (es)
Original Assignee
Genentech Inc
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39942941&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR068402(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Genentech Inc, Hoffmann La Roche filed Critical Genentech Inc
Publication of AR068402A1 publication Critical patent/AR068402A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T436/00—Chemistry: analytical and immunological testing
    • Y10T436/14—Heterocyclic carbon compound [i.e., O, S, N, Se, Te, as only ring hetero atom]

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ARP080103927A 2007-09-12 2008-09-10 Combinaciones de compuestos inhibidores de fosfoinositida 3-quinasa y agentes quimioterapeuticos y los metodos de uso AR068402A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US97177307P 2007-09-12 2007-09-12

Publications (1)

Publication Number Publication Date
AR068402A1 true AR068402A1 (es) 2009-11-18

Family

ID=39942941

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080103927A AR068402A1 (es) 2007-09-12 2008-09-10 Combinaciones de compuestos inhibidores de fosfoinositida 3-quinasa y agentes quimioterapeuticos y los metodos de uso

Country Status (18)

Country Link
US (3) US8247397B2 (enExample)
EP (1) EP2205242B1 (enExample)
JP (1) JP5658565B2 (enExample)
KR (1) KR101584823B1 (enExample)
CN (1) CN101939006B (enExample)
AR (1) AR068402A1 (enExample)
AU (1) AU2008298948B2 (enExample)
BR (1) BRPI0816769A2 (enExample)
CA (1) CA2699202C (enExample)
CL (1) CL2008002687A1 (enExample)
ES (1) ES2537352T3 (enExample)
IL (1) IL204333A (enExample)
MX (1) MX338504B (enExample)
PE (2) PE20090678A1 (enExample)
RU (1) RU2523890C2 (enExample)
TW (1) TWI471134B (enExample)
WO (1) WO2009036082A2 (enExample)
ZA (1) ZA201002475B (enExample)

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KR20100085912A (ko) 2010-07-29
JP5658565B2 (ja) 2015-01-28
US8604014B2 (en) 2013-12-10
CL2008002687A1 (es) 2009-01-16
BRPI0816769A2 (pt) 2016-11-29
CN101939006A (zh) 2011-01-05
US20110223619A1 (en) 2011-09-15
US20090098135A1 (en) 2009-04-16
EP2205242B1 (en) 2015-04-15
EP2205242A2 (en) 2010-07-14
US8247397B2 (en) 2012-08-21
RU2523890C2 (ru) 2014-07-27
IL204333A (en) 2016-08-31
WO2009036082A3 (en) 2009-11-19
AU2008298948B2 (en) 2014-09-04
CA2699202A1 (en) 2009-03-19
PE20090678A1 (es) 2009-06-27
TW200920377A (en) 2009-05-16
TWI471134B (zh) 2015-02-01
HK1145287A1 (en) 2011-04-15
MX2010002543A (es) 2010-03-29
ES2537352T3 (es) 2015-06-05
JP2010539177A (ja) 2010-12-16
ZA201002475B (en) 2011-06-29
CN101939006B (zh) 2015-09-16
CA2699202C (en) 2016-09-27
PE20140100A1 (es) 2014-02-12
RU2010112837A (ru) 2011-10-20
US20130345217A1 (en) 2013-12-26

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