AR054191A1 - Compuestos de 3 aminopirrolidina sustituidos utiles como inhibidores de la recaptacion de monoamina - Google Patents

Compuestos de 3 aminopirrolidina sustituidos utiles como inhibidores de la recaptacion de monoamina

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Publication number
AR054191A1
AR054191A1 ARP060101917A ARP060101917A AR054191A1 AR 054191 A1 AR054191 A1 AR 054191A1 AR P060101917 A ARP060101917 A AR P060101917A AR P060101917 A ARP060101917 A AR P060101917A AR 054191 A1 AR054191 A1 AR 054191A1
Authority
AR
Argentina
Prior art keywords
group
lower alkyl
groups
substituted
optionally substituted
Prior art date
Application number
ARP060101917A
Other languages
English (en)
Spanish (es)
Inventor
Nobuaki Ito
Kuninori Tai
Noriaki Takemura
Yasuhiro Menjo
Shin Miyamura
Yohji Sakurai
Yasuyo Sakata
Takumi Masumoto
Kohei Akazawa
Naoki Amada
Satoshi Ohashi
Tomoichi Shinohara
Hirofumi Sasaki
Junko Yamashita
Satoko Nakajima
Muneaki Kurimura
Shinichi Taira
Haruhiko Sugino
Takahiro Tomoyasu
Takayuki Matsuzaki
Akihito Watanabe
Chisako Morita
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36693623&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR054191(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of AR054191A1 publication Critical patent/AR054191A1/es

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    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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ARP060101917A 2005-05-13 2006-05-12 Compuestos de 3 aminopirrolidina sustituidos utiles como inhibidores de la recaptacion de monoamina AR054191A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2005141230 2005-05-13

Publications (1)

Publication Number Publication Date
AR054191A1 true AR054191A1 (es) 2007-06-06

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ID=36693623

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ARP060101917A AR054191A1 (es) 2005-05-13 2006-05-12 Compuestos de 3 aminopirrolidina sustituidos utiles como inhibidores de la recaptacion de monoamina

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Country Link
US (6) US8084442B2 (en:Method)
EP (2) EP1881975B8 (en:Method)
JP (1) JP4776631B2 (en:Method)
KR (2) KR20100038453A (en:Method)
CN (3) CN101175748A (en:Method)
AR (1) AR054191A1 (en:Method)
AU (2) AU2006244851B2 (en:Method)
BR (1) BRPI0610279A2 (en:Method)
CA (1) CA2608184C (en:Method)
CY (1) CY1114767T1 (en:Method)
DK (1) DK2407451T3 (en:Method)
ES (2) ES2446375T3 (en:Method)
IL (1) IL187311A (en:Method)
IN (1) IN2012DN00758A (en:Method)
MX (1) MX2007014252A (en:Method)
MY (1) MY148653A (en:Method)
PL (1) PL2407451T3 (en:Method)
PT (1) PT2407451E (en:Method)
RU (1) RU2414454C2 (en:Method)
SG (1) SG162722A1 (en:Method)
SI (1) SI2407451T1 (en:Method)
TW (3) TWI410406B (en:Method)
WO (1) WO2006121218A1 (en:Method)
ZA (1) ZA200709691B (en:Method)

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GEP20115290B (en) 2002-11-27 2011-09-26 Incyte Corp 3-aminopyrrolidine derivatives as modulators of chemokine receptors
TWI410406B (zh) 2005-05-13 2013-10-01 Otsuka Pharma Co Ltd 吡咯烷化合物
BRPI0619263A2 (pt) * 2005-11-30 2011-09-27 Hoffmann La Roche indóis de 3-amino-1-arilpropila e indóis aza-substituìdos, métodos para prepará-los, composição farmacêutica e uso dos referidos indóis
US20100216813A1 (en) * 2005-11-30 2010-08-26 Smithkline Beecham Corporation Pyrrolidineanilines
JP5219465B2 (ja) * 2006-11-10 2013-06-26 大塚製薬株式会社 医薬
ES2370593T3 (es) 2008-03-20 2011-12-20 F. Hoffmann-La Roche Ag Derivados de pirrolidinilo y usos de los mismos.
JP5827627B2 (ja) * 2009-11-07 2015-12-02 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung TGF−β受容体キナーゼ阻害剤としてのヘテロアリールアミノキノリン
EP2560953B1 (en) * 2010-04-21 2016-01-06 Probiodrug AG Inhibitors of glutaminyl cyclase
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