AR016432A1 - Derivados de la equinocandina, su procedimiento de preparacion, compuestos intermediarios y composiciones farmaceuticas. - Google Patents

Derivados de la equinocandina, su procedimiento de preparacion, compuestos intermediarios y composiciones farmaceuticas.

Info

Publication number
AR016432A1
AR016432A1 ARP980106281A ARP980106281A AR016432A1 AR 016432 A1 AR016432 A1 AR 016432A1 AR P980106281 A ARP980106281 A AR P980106281A AR P980106281 A ARP980106281 A AR P980106281A AR 016432 A1 AR016432 A1 AR 016432A1
Authority
AR
Argentina
Prior art keywords
radical
atom
atoms
eventually
cyclic
Prior art date
Application number
ARP980106281A
Other languages
English (en)
Spanish (es)
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9715628A external-priority patent/FR2772028B1/fr
Priority claimed from FR9813361A external-priority patent/FR2784993B1/fr
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of AR016432A1 publication Critical patent/AR016432A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/18Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Detergent Compositions (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
ARP980106281A 1997-12-10 1998-12-10 Derivados de la equinocandina, su procedimiento de preparacion, compuestos intermediarios y composiciones farmaceuticas. AR016432A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9715628A FR2772028B1 (fr) 1997-12-10 1997-12-10 Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides
FR9813361A FR2784993B1 (fr) 1998-10-26 1998-10-26 Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides

Publications (1)

Publication Number Publication Date
AR016432A1 true AR016432A1 (es) 2001-07-04

Family

ID=26233984

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980106281A AR016432A1 (es) 1997-12-10 1998-12-10 Derivados de la equinocandina, su procedimiento de preparacion, compuestos intermediarios y composiciones farmaceuticas.

Country Status (43)

Country Link
US (3) US6677429B1 (enExample)
EP (1) EP1036090B1 (enExample)
JP (1) JP4361679B2 (enExample)
KR (1) KR100564872B1 (enExample)
CN (1) CN1284084A (enExample)
AP (2) AP1260A (enExample)
AR (1) AR016432A1 (enExample)
AT (1) ATE321772T1 (enExample)
AU (1) AU755033B2 (enExample)
BG (1) BG65033B1 (enExample)
BR (1) BR9813531A (enExample)
CA (1) CA2311295A1 (enExample)
CO (1) CO4980875A1 (enExample)
CU (1) CU22962A3 (enExample)
CY (1) CY1105695T1 (enExample)
CZ (1) CZ301919B6 (enExample)
DE (1) DE69834057T2 (enExample)
DK (1) DK1036090T3 (enExample)
DZ (1) DZ2670A1 (enExample)
EA (1) EA002706B1 (enExample)
EE (1) EE04837B1 (enExample)
ES (1) ES2259462T3 (enExample)
GE (1) GEP20032975B (enExample)
HR (1) HRP20000384B1 (enExample)
HU (1) HUP0100263A3 (enExample)
IL (4) IL136647A0 (enExample)
MA (1) MA26575A1 (enExample)
NO (1) NO327498B1 (enExample)
NZ (1) NZ504614A (enExample)
OA (1) OA11899A (enExample)
PA (1) PA8464201A1 (enExample)
PE (1) PE130099A1 (enExample)
PL (1) PL196889B1 (enExample)
PT (1) PT1036090E (enExample)
RS (1) RS49905B (enExample)
SA (1) SA99191248B1 (enExample)
SK (1) SK286916B6 (enExample)
TN (1) TNSN98222A1 (enExample)
TR (1) TR200001655T2 (enExample)
TW (1) TW446541B (enExample)
UA (1) UA72200C2 (enExample)
UY (1) UY25292A1 (enExample)
WO (1) WO1999029716A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
WO2000024694A1 (en) * 1998-10-28 2000-05-04 Eli Lilly And Company Photochemical process for making 1-deoxy-2-keto derivatives
FR2794746B1 (fr) 1999-06-09 2002-12-06 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2794747B1 (fr) 1999-06-09 2004-04-16 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2833596B1 (fr) * 2001-12-14 2005-02-18 Aventis Pharma Sa Procede de preparation de derives d'echinocandine
CN101659692B (zh) * 2008-08-27 2012-07-04 上海医药工业研究院 制备棘球康定b的方法
CN101659693B (zh) * 2008-08-27 2012-11-21 上海医药工业研究院 制备纽莫康定b0的方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2241955A (en) * 1990-03-16 1991-09-18 Merck & Co Inc Cyclohexapeptide compounds
NZ247149A (en) * 1992-03-19 1996-10-28 Lilly Co Eli Cyclic peptide antifungal agents and compositions thereof
US5516757A (en) * 1994-09-16 1996-05-14 Merck & Co., Inc. Semi-synthetic lipopeptides, compositions containing said lipopeptides, and methods of use
US5516756A (en) * 1994-10-31 1996-05-14 Merck & Co., Inc. Aza cyclohexapeptide compounds
DE69615535T2 (de) * 1995-01-26 2002-05-02 Merck & Co., Inc. Neue fungizide cyclohexapeptide
US5646111A (en) * 1995-04-07 1997-07-08 Eli Lilly And Company Cyclic peptide antifungal Agents
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
FR2794747B1 (fr) * 1999-06-09 2004-04-16 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques

Also Published As

Publication number Publication date
DE69834057T2 (de) 2006-12-14
CY1105695T1 (el) 2010-12-22
CZ20002113A3 (cs) 2000-11-15
AP1567A (en) 2006-02-08
NZ504614A (en) 2002-12-20
NO20002959L (no) 2000-08-09
EA002706B1 (ru) 2002-08-29
ES2259462T3 (es) 2006-10-01
EE04837B1 (et) 2007-06-15
PL196889B1 (pl) 2008-02-29
TNSN98222A1 (fr) 2005-03-15
UY25292A1 (es) 2000-12-29
AP2000001826A0 (en) 2000-06-30
SA99191248B1 (ar) 2006-08-12
PL341012A1 (en) 2001-03-12
AU1565999A (en) 1999-06-28
JP4361679B2 (ja) 2009-11-11
PT1036090E (pt) 2006-06-30
HRP20000384B1 (en) 2010-02-28
DK1036090T3 (da) 2006-07-24
US20050267019A1 (en) 2005-12-01
AU755033B2 (en) 2002-11-28
WO1999029716A1 (fr) 1999-06-17
BG65033B1 (bg) 2006-12-29
CO4980875A1 (es) 2000-11-27
US7285619B2 (en) 2007-10-23
OA11899A (fr) 2006-04-10
KR20010032924A (ko) 2001-04-25
IL136647A0 (en) 2001-06-14
UA72200C2 (uk) 2005-02-15
ATE321772T1 (de) 2006-04-15
TW446541B (en) 2001-07-21
AP1260A (en) 2004-03-16
CU22962A3 (es) 2004-06-21
PA8464201A1 (es) 2000-09-29
NO20002959D0 (no) 2000-06-09
SK286916B6 (sk) 2009-07-06
CA2311295A1 (fr) 1999-06-17
EP1036090B1 (fr) 2006-03-29
KR100564872B1 (ko) 2006-03-30
US6677429B1 (en) 2004-01-13
CZ301919B6 (cs) 2010-07-28
PE130099A1 (es) 1999-12-16
HUP0100263A3 (en) 2002-11-28
IL136647A (en) 2007-06-03
BR9813531A (pt) 2000-10-10
MA26575A1 (fr) 2004-12-20
YU33900A (sh) 2002-08-12
GEP20032975B (en) 2003-05-27
HUP0100263A1 (hu) 2001-08-28
US7160983B2 (en) 2007-01-09
DZ2670A1 (fr) 2003-03-22
EA200000625A1 (ru) 2000-12-25
BG104494A (en) 2001-01-31
SK8392000A3 (en) 2001-10-08
HRP20000384A2 (en) 2000-10-31
JP2001525421A (ja) 2001-12-11
TR200001655T2 (tr) 2000-11-21
IL184171A0 (en) 2007-10-31
US20040072737A1 (en) 2004-04-15
NO327498B1 (no) 2009-07-20
IL172412A (en) 2008-11-26
AP2003002874A0 (en) 2003-09-30
CN1284084A (zh) 2001-02-14
EE200000336A (et) 2001-08-15
DE69834057D1 (de) 2006-05-18
EP1036090A1 (fr) 2000-09-20
RS49905B (sr) 2008-08-07

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Legal Events

Date Code Title Description
FG Grant, registration